Cayman Chemical | CB-52

10010117 CB-52

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• See more Cannabinoids; Inflammation; Neuroscience

Chemical structure definitions are available for many Cayman products. See Chemical Structure Database for details.

CB-52 is a stable analog of Δ⁹-tetrahydrocannabinol (THC) and anandamide (AEA). It exhibits high affinity for the central cannabinoid (CB₁) and peripheral cannabinoid (CB₂) receptor with K_i values of 210 and 30 nM, respectively.¹ In vitro, CB-52 behaves primarily as a CB₁ receptor partial agonist and a CB₂ receptor neutral antagonist.²

1 Brizzi, A., Brizzi, V., Cascio, M.G., et al. Design, synthesis, and binding studies of new potent ligands of cannabinoid receptors. J Med Chem 48 7343-7350 (2005).

2 Cascio, M.G., Bisogno, T., Palazzo, E., et al. In vitro and in vivo pharmacology of synthetic olivetol- or resorcinol-derived cannabinoid receptor ligands. Br J Pharmacol 149 431-440 (2006).

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Purchase 10010117 CB-52

Pricing is for North America only. Other customers should contact a distributor in their region.

This product is also available to buy in bulk quantities. Please contact our Sales Department for a quote or to purchase.

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Warning This product is not for human or veterinary use.

Pricing updated 2010-03-17.
Prices are subject to change without notice.

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Stability of this item is suitable for room temperature overnight shipping. If shipment on ice is desired, it must be requested when the order is placed.