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HU-210

Cayman Chemical Item Number 90082

(CAS 112830-95-2)

HU-210 (CAS 112830-95-2)

See more	Cannabinoids (296) Endocrinology (335) Forensic Science (306) Neuroscience (654)

Description

HU-210 is a synthetic agonist analog of Δ⁹-THC, which is the primary psychoactive component of marijuana. HU-210 is a potent central cannabinoid (CB₁) and peripheral cannabinoid (CB₂) receptor agonist. It binds to neuroblastoma cell membrane CB₁ receptors with about the same affinity as CP-55940.¹ In mouse behavior models (hypothermia, analgesia, hypoactivity, and catalepsy) the ED₅₀ is 5-20 µg/kg.²

1 Slipetz, D.M., O'Neill, G.P., Gavreau, L., et al. Activation of the human peripheral cannabinoid receptor results in inhibition of adenylyl cyclase. Mol Pharmacol 48 352-361 (1995).

2 Howlett, A.C., Berglund, B., and Melvin, L.S. Cannabinoid receptor agonists and antagonists. Curr Pharm Des 1 343-354 (1995).

Formal Name	3-(1,1'-dimethylheptyl)-6aR,7,10,10aR-tetrahydro-1-hydroxy-6,6-dimethyl-6H-dibenzo[b,d]pyran-9-methanol
CAS Number	112830-95-2
Molecular Formula	C₂₅H₃₈O₃
Formula Weight	386.6
Formulation	A crystalline solid
Purity	>98%
λ_max	207 nm
Stability	2 years
Storage	-20°C
Shipping	Room temperature in continental US; may vary elsewhere
SMILES	Copy SMILES to clipboard CCCCCCC(C)(C)c1cc(O)c2c(c1)OC(C)(C)[C@@H]1CCC(CO)CC21

Background Reading

Slipetz, D.M., O'Neill, G.P., Gavreau, L., et al. Activation of the human peripheral cannabinoid receptor results in inhibition of adenylyl cyclase. Mol Pharmacol 48 352-361 (1995).

Howlett, A.C., Berglund, B., and Melvin, L.S. Cannabinoid receptor agonists and antagonists. Curr Pharm Des 1 343-354 (1995).

HU-210 is available in the following screening library:

Cannabinoid Agonist Screening Library (96-Well)

Size	Price	Quantity	Subtotal
1 mg	$24.00		$0.00
5 mg	$112.00		$0.00
10 mg	$199.00		$0.00
25 mg	$430.00		$0.00
Bulk	Contact
		Cart Total	$0.00

Pricing updated 2012-02-12. Prices are subject to change without notice.

To ask for assistance with one of our products please contact a Technical Support Scientist.

This product requires special processing and/or additional information before it can be shipped. A Customer Service representative will contact you within 24 hours of receipt of your order.

Warning This product is not for human or veterinary use.

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JWH 018 Selective agonist of the CB2 receptor	39.860919038187
JWH 018 (solution) Selective agonist of the CB2 receptor	68.923268613605
JWH 073 Selective agonist of the CB1 receptor	40.353743785596
JWH 073 (solution) Selective agonist of the CB1 receptor	44.560786731709
JWH 200 Potent cannabinoid receptor agonist	47.054774727766
JWH 200 (solution) Potent cannabinoid receptor agonist	45.758690559580
(±)-CP 47,497 A potent CB1 receptor agonist	29.260334883041
(±)-CP 47,497 (solution) A potent CB1 receptor agonist	40.643750448281
(±)-CP 47,497-C8-homolog Exclusive A potent bicyclic CB analog	33.211843073581
(±)-CP 47,497-C8-homolog (solution) Exclusive A potent bicyclic CB analog	43.502412536909
HU-210 (solution) A potent synthetic cannabinoid	26.336929755327
Cannabidiol A neuroprotective phenolic compound from marijuana	26.647332280978
Cannabidiol (solution) A neuroprotective phenolic compound from marijuana	33.602882973380
Synthetic Cannabinoid HPLC Mixture II	39.551017802333

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