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Holiday Notification: Cayman Chemical will be closed Monday, May 28, 2012, in observance of the Memorial Day holiday. More…
Please feel free to continue placing orders via our website or via fax at 734-971-3640. You may send an email to customer service at custserv@caymanchem.com , or to technical support at techserv@caymanchem.com which we will respond to the next business day. Cayman will resume regular business hours and shipping schedules on Tuesday, May 29, 2012. Thank you for your patience and understanding.

Epigenetics & Assay Kits

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Item Number Product Sizes & Pricing CAS Purity Image Exclusive Introduction Date Mojo Plain Text Name Synonyms Keywords Interest
600520 BRD4 bromodomain 1 TR-FRET Assay Kit New - 2012-04-25 87.870599080453 brd4-bromodomain-1-tr-fret-assay-kit kits assays measures measurements acetylations histones lysines epigenetics regulations genes transcriptions acetylated residues small proteins bromodomains nucleosomes chromatins structures expression BET family tandem Extra Terminal BRD2 BRD3 BRDT cells cellular inflammatory inflammation mitosis viral host virus viral/host interactions binds binding tails couples marks transcriptional targets promoters molecules inhibitors bromodomain/histone I-BET JQ-1 therapeutics human diseases complexes activated macrophages protection protects bacteria-induced sepsis lipopolysaccharides lipopolysaccharide-triggered endotoxic shock enantiomerically pure (+)-JQ1 (+)-JQ-1 2 bromodomain-peptides displacement inhibits inhibitors probes oncogenesis oncology cancers homogeneous TR-FRET time-resolved fluorescence resonance energy transfer characterization bromodomain/acetylated interactions fluorophores europium Eu3+ chelates biotinylated ligands allophycocyanin APC-labeled avidins biotins 87.870599080453
600530 BRD4 bromodomain 2 TR-FRET Assay Kit New - 2012-04-26 88.919981796503 brd4-bromodomain-2-tr-fret-assay-kit kits assays measures measurements acetylations histones lysines epigenetics regulations genes transcriptions acetylated residues small proteins bromodomains nucleosomes chromatins structures expression BET family tandem Extra Terminal BRD2 BRD3 BRDT cells cellular inflammatory inflammation mitosis viral host virus viral/host interactions binds binding tails couples marks transcriptional targets promoters molecules inhibitors bromodomain/histone I-BET JQ-1 therapeutics human diseases complexes activated macrophages protection protects bacteria-induced sepsis lipopolysaccharides lipopolysaccharide-triggered endotoxic shock enantiomerically pure (+)-JQ1 (+)-JQ-1 1 bromodomain-peptides displacement inhibits inhibitors probes oncogenesis oncology cancers homogeneous TR-FRET time-resolved fluorescence resonance energy transfer characterization bromodomain/acetylated interactions fluorophores europium Eu3+ chelates biotinylated ligands allophycocyanin APC-labeled avidins biotins 88.919981796503
700390 Demethylase (Jumonji-type) Activity Assay Kit - 2010-05-26 28.154262474787 demethylase-jumonji-type-activity-assay-kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC JHDM1 JHDM2 JHDM3 JARID1 UTX/UTY cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 28.154262474787
700400 Demethylase (LSD-type) Activity Assay Kit - 2010-08-05 17.725588003157 demethylase-lsd-type-activity-assay-kit kits assays measures measurements histones proteins nucleoproteins chromatins structures DNA deoxyribonuclease eukaryotics nucleus nucleosomals core particles H3 H4 H2B H2A octamers amino termini post-translationally acetylation phosphorylations ubiquitination methylations replication repair transcriptional activation repression dysregulation tumor suppressor genes cancers enzymes catalyze epigenetic marks therapeutics drugs development lysine-specific demethylases LSD1 KDM1 p110b BHC110 NPAO LSD2 flavin adenines dinucleotides FAD-dependent amines oxidases monoamines MAOs polyamines PAOs demethylates monomethylateds dimethylateds lysines 4 K4 repression deacetylases co-repressor complexes 1/2 CtBP neuronal CoREST p53 LYS370 53BP1 apoptosis C-terminal domains CW-type zinc finger motif zince-binding sites chromatin-remodeling fluorescence-based formaldehyde N-terminal tail acetoacetanilides ammonia 17.725588003157
589324 DNA Methylation EIA Kit - 2009-04-23 86.454575966850 dna-methylation-eia-kit 5-methyl-2-deoxy Cytidine ELISA Kit solid plates DNA deoxyribonucleic acids CpG islands dinucleotides genes genomes cancers genomic hypomethylation hypermethylation tumors suppressors malignancy carcinogenesis plasma blood urine leukemia tissues differentiation aging methyltransferases DNMTs DNMT1 DNMT3a DNMT3b nucleosides analogs azacitidine decitabine zebularine drugs suppression competitive assays EIAs ELISAs culture supernatants sample matrices 86.454575966850
700500 G9a Methyltransferase Inhibitor Screening Assay Kit - 2011-03-10 42.864293560789 g9a-methyltransferase-inhibitor-screening-assay-kit EHMT2 Methyltransferase Inhibitor Screening Assay Kit kits assays measures measurements methylations molecules proteins signals transductions biosynthesis proteins repair genes silencing chromatin regulation S-adenosylmethionine SAM methyltransferases enzymes enzymatic cofactors ATP adenosine triphosphates AdoMet donors methyls groups DNA deoxyribonucleic acids Alzheimer's diseases depression Parkinson's multiple sclerosis livers failures cancers methylations lysines transcriptional activation respression histones functions SET domain-containing mammalian monomethylates dimethylates 9 27 H3 embryogenesis genomic imprinting lymphocytes lung cells HIV-1 H3K9 viral latency GLP G9a-like EHMT1 tumors suppressors p53 373 feedback inhibition methylation reactions 42.864293560789
10006515 HAT Inhibitor Screening Assay Kit - 2006-12-06 14.105470800027 hat-inhibitor-screening-assay-kit Histone Acetyltransferase Inhibitor Screening Assay Kit therapeutics histones p300/CBP-Associated Factors pCAF GNAT GCN5-related N-acetyltransferases acetylates lysines N-terminal terminus tails H3 H4 tumors suppressor genes PTEN human cancers apoptosis fluorescence fluorescent inhibitors fluorometric assays 14.105470800027
700230 HDAC8 Inhibitor Screening Assay Kit - 2009-05-15 21.721975138121 hdac8-inhibitor-screening-assay-kit Histone Deacetylase 8 Inhibitor Screening Assay Kit histone deacetylases inhibits inhibitors inhibition angiogenesis cycling apoptosis differentiation tumors proliferation anticancers genes epigenetic trichostatin A human class I tissues nucleus cytosolic smooth muscle neuroblastoma pathogenesis kits assays measures measurement fluorescent fluorescence-based 21.721975138121
600150 HDAC Cell-Based Activity Assay Kit - 2009-11-09 26.370505361597 hdac-cell-based-activity-assay-kit Histone Deacetylase Cell-Based Activity Assay Kit assays kits measuring measurement histones deacetylases lysines residues chromatin condensation transcriptional repression fluorescence deacetylation fluorescent inhibits inhibition enzymes fluorometric assays cancer modulators whole cells proteins lysine-specific HDAC1 homogenous inhibitor/activator TSA 26.370505361597
700360 JMJD2A Inhibitor Screening Assay Kit - 2010-05-25 19.047282813814 jmjd2a-inhibitor-screening-assay-kit Jumonji Domain Containing 2A Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC JHDM1 JHDM2 JHDM3 JARID1 UTX/UTY cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated 19.047282813814
700370 JMJD2D Inhibitor Screening Assay Kit - 2010-05-25 19.603553147282 jmjd2d-inhibitor-screening-assay-kit Jumonji Domain Containing 2D Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation FLJ10251 replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated 19.603553147282
700120 LSD1 Inhibitor Screening Assay Kit - 2008-10-16 24.063191420214 lsd1-inhibitor-screening-assay-kit Lysine-Specific Demethylase 1 lysines 4 demethylases histones residues repression transcription chromosomal DNA chromosomes inhibits inhibitors inhibition tumors suppressors activity cells cycles progression cancers fluorescent fluorescence enzymes enzymatic reactions H2O2 hydrogens peroxides peptides N-terminal tails H3 horseradish peroxidases ADHP resorufins assays 24.063191420214
700140 Methyltransferase Colorimetric Assay Kit - 2009-04-07 30.225331001137 methyltransferase-colorimetric-assay-kit MT Colorimetric Assay Kit assays kits measures measuring monitoring monitors MTs methylation signal transduction biosynthesis repair gene silencing chromatin regulation S-adenosylmethionine SAM-dependent methyltransferases enzymatic cofactors AdoMet donor modifications DNA Alzheimer's diseases depression Parkinson's multiple sclerosis liver failure cancers enzyme-coupled AdoHcy positive control S-adenosylhomocysteine 30.225331001137
700150 Methyltransferase Fluorometric Assay Kit - 2009-04-08 26.105699252585 methyltransferase-fluorometric-assay-kit MT Fluorometric Assay Kit assays kits measures measuring monitoring monitors MTs methylation signal transduction biosynthesis proteins repair gene silencing chromatin regulation S-adenosylmethionine SAM-dependent methyltransferases enzymes enzymatic cofactors AdoMet donor proteins modifications DNA Alzheimer's diseases depression Parkinson's multiple sclerosis liver failure cancers enzyme-coupled AdoHcy positive control S-adenosylhomocysteine 26.105699252585
700560 PAD4 Inhibitor Screening Assay Kit - 2011-05-04 49.092011970534 pad4-inhibitor-screening-assay-kit Protein Arginine Deiminase 4; Peptidylarginine Deiminase 4 kits assays measures measurements proteins arginines deiminases PADs guanidine-modifying enzymes peptidylarginine deiminase amidinotransferases nucleus homodimers transcriptional coregulator catalyzes residues citrulline calcium-dependent substrates histones H2A H3 H4 post-translational modifications genes regulations autocitrullination inhibits enzymatic activity cells rheumatoid arthritis citrulline-containing immune response autoantibodies tissues multiple sclerosis Alzheimer's diseases glaucoma cancers human deiminates N-α-benzoyl-L-arginine ethyl esters BAEE kinetic ammonia detectors fluorescent fluorescence 49.092011970534
700270 SET7/9 Methyltransferase Inhibitor Screening Assay Kit - 2009-12-04 24.872556970425 set7-9-methyltransferase-inhibitor-screening-assay-kit methyltransferases SET Domain-containing Protein 7/9 lysines 7 KMT7 methylation signal transduction biosynthesis proteins repair genes silencing chromatins S-adenosylmethionine SAM AdoMet methyl donors Alzheimer's depression Parkinson's Diseases multiple sclerosis liver cancers substrates histones histone 3 lysine residue 4 H3K4 p53 transcription factors TAF10 mono-methylated mono-methylase DNA damage acetylation human tumorigenesis inhibitors acceptor peptides S-adenosylhomocysteine S-ribosylhomocysteine adenine nucleosidase hypoxanthine deaminase urate hydrogen peroxide H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin fluorescence measures measurement assays kits 24.872556970425
600490 SET7/9 SAM-Screener Assay Kit New - 2011-12-21 41.633066544674 set7-9-sam-screener-assay-kit SET7/9 SAM-Binding Site Inhibitor Screening kits assays measures measurements chromatins posttranslational modifications histones DNA deoxyribonucleic acids lysines methylations epigenetics regulations genomes mono-methyltransferases MTs domains S-adenosyl-L-methionines SAM AdoMet co-factors epsilons amino groups Dot1 KMT7 domain-containing non-histones H3 TAF10 p53 viral Tat estrogens receptors alpha .alpha. α substrates humans diseases catalytic catabolism fluorescence EpiTrek polarizations fluorescent probes binding pockets endogenous cofactors sinefungin peptides high-throughput 41.633066544674
700350 SET8 Methyltransferase Inhibitor Screening Assay Kit - 2010-03-09 21.155178831055 set8-methyltransferase-inhibitor-screening-assay-kit SET domain-containing (lysine methyltransferase) 8; PR-Set7; SETD8 assays kits measures measurement methyltransferases MTs inhibits inhibitors inhibition methylation signal transduction biosynthesis protein repair genes silencing chromatins regulation S-adenosylmethionine (SAM)-dependent AdoMet DNA deoxyribonucleic acids Alzheimer's diseases depression Parkinson's multiple sclerosis livers cancers KMT5A lysines PR-Set 7 methylates histones H4 residues 20 H4K20 transcriptional p53 tumors suppressors tumorigenesis inhibits inhibition inhibitors peptides S-adenosylhomocysteines S-ribosylhomocysteines adenines nucleosidases hypoxanthines deaminases hydrogen peroxides H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazines fluorescent fluorescence resorufin 21.155178831055
10010401 SIRT1 Direct Fluorescent Screening Assay Kit - 2008-02-26 51.236933701657 sirt1-direct-fluorescent-screening-assay-kit SIRT 1 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human homologs yeast SIR2 silent information regulators 2 tumors cancers suppressors inhibits inhitors inhibition apoptosis screening fluorescence activators fluorescent fluorometric 51.236933701657
10010991 SIRT1 FRET-Based Screening Assay Kit - 2008-02-19 20.010414364640 sirt1-fret-based-screening-assay-kit SIRT 1 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human homologs yeast SIR2 silent information regulators 2 tumors cancers suppressors inhibits inhitors inhibition apoptosis screening fluorescence activators fluorescent fluorometric 20.010414364640
700280 SIRT2 Direct Fluorescent Screening Assay Kit - 2009-12-10 40.755135213724 sirt2-direct-fluorescent-screening-assay-kit Nucleosomes chromosomal deoxyribonucleases DNA histones H2A H2B H3 H4 octameric cores transcription amino termini acetylation phosphorylation methylation ε-amino lysines acetyltransferases HATs chromatins genes activation deacetylases HDACs catalyzes hydrolytic acetyls sirtuins trichostatins A-insensitive lysyl-deacetylases class III catalyzes deacetylation nicotinamides O-acetyl-ADP-ribose NAD+ human SIRT1 SIRT2 SIRT3 SIRT4 SIRT5 SIRT6 SIRT7 cytoplasmic proteins H4 lysine-16 lysine-40 α-tubulin a-tubulin alpha-tubulin HDAC6 microtubules mitotic chromosomal hyperpolid cells tissues skeletal muscle heart oligodendroglia brain tumor suppressor gliomas Down-regulation gene chromosomal region diagnostic marker fluorescence-based inhibitors activators p53 Gln-Pro-Lys-Lys(ε-acetyl)-AMC recombinant NAD+ fluorescent fluorescence kits assays measures measurement 40.755135213724
10011566 SIRT3 Direct Fluorescent Screening Assay Kit - 2008-08-21 48.920476519337 sirt3-direct-fluorescent-screening-assay-kit SIRT 3 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human mitochondrial proteins mitochondrias localization matrix-processing peptidase translocated nucleus cells cellular stress overexpression mice mouse murine caloric restriction up-regulates expression levels white brown adipose tissue BAT cold exposure PGC-1a PGC-1alpha PGC-1.alpha. UCP1 modulates adaptive thermogenesis deacetylation activation acetyl coenzymes A synthetase 2 AceCS2 catalyzes acetate CoA ketogenesis ATP direct genetic link longevity mutations genes enhancers marker life extension cellular metabolic control whole-body metabolism chronic diseases dysfunction neuronal pathogenesis neurodegenerative cancers aging apoptosis screening fluorescence activators fluorescent fluorometric 48.920476519337
700290 SIRT6 Direct Fluorescent Screening Assay Kit - 2010-02-18 37.424678867403 sirt6-direct-fluorescent-screening-assay-kit SIRT 6 SIRT-6 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human mitochondrial nuclear proteins mitochondrias translocated nucleus cells cellular stress lysine deacetylation nicotinamides O-acetyl-ADP-ribose NAD+ abstracted ADP-ribosyl transferases deacetylases telomeres chromatins NF-κB NF-kappaB NF-.kappa.B signaling signalling mammalian cells Werner Syndromes aging disorders anti-cancers anti-inflammatory drugs apoptosis screening fluorescence activators Arg-His-Lys-Lys(ε-acetyl)-AMC fluorescent fluorometric 37.424678867403
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