| 10976 |
10-HDA
|
|
14113-05-4 |
≥98%
|
|
|
2011-10-13
|
79.840110497237
|
10-hda
|
|
fatty acids royal jelly lifespan MMP RA, rheumatoid arthritis VEGF angiogenesis antitumor neurogenesis collagen |
79.840110497237
|
| 13021 |
2-Methoxyestradiol
|
|
362-07-2 |
≥98%
|
|
|
2009-01-06
|
80.715256511444
|
2-methoxyestradiol
|
Panzem; NSC 659853; 2-ME2; 2-Hydroxyestradiol 2-methyl ether
|
estradiol steroids catechol-O-methyltransferase COMT pre-eclampsia preeclampsia angiogenesis cancers anticaner HIF-1α HIF1α 2-methoxyestradiol |
80.715256511444
|
| 582261 |
2-Methoxyestradiol EIA Kit
|
|
- |
|
|
|
2010-12-09
|
176.477409453652
|
2-methoxyestradiol-eia-kit
|
2-Hydroxyestradiol 2-methyl ester; 2-ME2
|
metabolites estradiols antitumors antiangiogenics breast prostate cancers cardioprotective cytochromes P450 CYP450 P450-dependent hydroxylation 17β-estradiols 2-position O-methylation catechol-O-methyltransferases pre-eclampsia plasma urine urinary markers therapeutics supplements estrogen receptors pregnancy ELISAs EIAs enzymes immunoassays kits competitive quantification measures measurements sample matrices |
176.477409453652
|
| 10397 |
3-amino Benzamide
|
|
3544-24-9 |
≥98%
|
|
|
2011-10-07
|
2.107037223058
|
3-amino-benzamide
|
3-(Aminocarbonyl) Aniline; 3-Carboxamidoaniline
|
poly(ADP-ribose) polymerases PARPs DNA repairs DNA strands breaks apoptosis inflammation atherosclerosis neruogenesis cancers angiogenesis signaling cellular responses inhibits inhibitor inhibition telomere shortening shortens stimulates mediated mediates PARP-mediated |
2.107037223058
|
| 580170 |
ANGPTL3 (human) EIA Kit
New
|
|
- |
|
|
|
2012-01-10
|
53.539463299131
|
angptl3-human-eia-kit
|
Angiopoietin-like protein 3
|
kits assays measures measurements angiopoietin-like proteins ANGPTLs angiopoietin-related growth factors AGF ligands regulated regulation angiogenesis glucose lipids energy metabolisms ANGPTL1 ANGPTL2 ANGPTL4 ANGPTL5 ANGPTL6 ANGPTL7 N-terminal N-terminus coiled-coil domains C-terminal C-terminus fibrinogen-like angiopoietins receptors Tie2 proteins Tie1 livers pro-angiogenic integrins αvβ3 endothelial cells migration adhesion inhibits inhibitors inhibition catalytic lipoproteins lipases catalyzes hydrolysis triglycerides HDL high density phospholipids hypolipidemic obese ob KK/Snk mice mouse expression hyperlipidemia atherosclerosis plasma human cholesterols immunometrics sandwich serums cultures supernatants |
53.539463299131
|
| 580190 |
ANGPTL6 (human) EIA Kit
New
|
|
- |
|
|
|
2012-01-10
|
48.569067273318
|
angptl6-human-eia-kit
|
Angiopoietin-like protein 6
|
kits assays measures measurements angiopoietin-like proteins ANGPTLs angiopoietin-related growth factors AGF ligands regulated regulation angiogenesis glucose lipids energy metabolisms ANGPTL1 ANGPTL2 ANGPTL4 ANGPTL5 ANGPTL3 ANGPTL7 N-terminal N-terminus coiled-coil domains C-terminal C-terminus fibrinogen-like angiopoietins receptors Tie2 proteins Tie1 hepatocytes angiogenesis arteriogenesis ERK1/2-eNOS pathways transgenic mice mouse systemic expenditure high-fat diet-induced obesity ob insulin resistance null diabetic fasting serums levels immunometric sandwich plasma cells cultures supernatants |
48.569067273318
|
| 10808 |
ANGPTL6 (human) Monoclonal Antibody (Clone Kairos-60)
|
|
- |
|
|
|
2011-06-27
|
0.395948434622
|
angptl6-human-monoclonal-antibody-clone-kairos-60
|
Angiopoietin-Related Growth Factor; AGF; Angiopoietin-Like Protein 6
|
antibodies antiserum serum western blot WB immunoblotting ELISA enzyme-linked immunosorbent assay ANGPTL-6 ANGPTL energy metabolism glucose lipids |
0.395948434622
|
| 13321 |
ARP 100
|
|
704888-90-4 |
≥98%
|
|
|
2009-10-07
|
2.175690607734
|
arp-100
|
MMP-2 Inhibitor III; CAY10609
|
matrix metalloproteinases MMP-2 MMP2 MMP 2 ECM cancers cells migration inhibitors gelatinase A MMPs proteases HT1080 tumors invasive |
2.175690607734
|
| 10009644 |
BAY-43-9006
|
|
284461-73-0 |
≥98%
|
|
|
2011-09-13
|
25.839792817680
|
bay-43-9006
|
Sorafenib; Nexovar®
|
inhibitors raf-1 b-raf receptors tyrosine kinases VEGF VEGFR PDGF PDGFR cancers angiogenesis apoptosis tumors cells cellular proliferation Flt-3 c-KIT carcinoma growth factor tosylate |
25.839792817680
|
| 11022 |
BIBF 1120
|
|
928326-83-4 |
≥95%
|
|
|
2011-11-10
|
6.088397790055
|
bibf-1120
|
Vargatef™
|
receptors tyrosine kinases inhibitors vascular endothelial growth factor VEGFR platelet-derived growth PDGFR fibroblasts FGFR angiogenesis cancers pulmonary fibrosis diseases |
6.088397790055
|
| 13187 |
Cardiogenol C (hydrochloride)
|
|
671225-39-1 |
≥97%
|
|
|
2009-02-06
|
3.462044198895
|
cardiogenol-c-hydrochloride
|
|
Embryonic stem cells Differentiation Cardiomyocytes Cardiac muscle GATA-4 MEF2 Nkx2.5 |
3.462044198895
|
| 10012682 |
CAY10585
|
|
934593-90-5 |
≥97%
|
|
|
2008-11-06
|
48.964775059194
|
cay10585
|
Hypoxia Inducible Factor-1α Inhibitor
|
HIF-1α HIF1α hypoxia cancers transcriptions factors VEGFs erythropoietin inhibitors inhibits inhibition |
48.964775059194
|
| 10208 |
CD34 Monoclonal FITC Antibody (Clone ICO-115)
|
|
- |
|
|
|
2008-07-23
|
34.607099447513
|
cd34-monoclonal-fitc-antibody-clone-ico-115
|
|
antibodies antiserum antisera flow cytometry immunofluorescence FC IF transmembranes glycoproteins leukemias stem cell lines |
34.607099447513
|
| 13199 |
cis-trismethoxy Resveratrol
|
|
94608-23-8 |
≥98%
|
|
|
2009-03-25
|
15.301954419889
|
cis-trismethoxy-resveratrol
|
cis-Trimethoxy Stilbene
|
resveratrol anti-mitotic growth inhibitors colon cancers tubulin polymerization polyamines putrescine spermidine cis-Trimethoxy resveratrol 3,5,4'-trimethoxystilbene 3,5,4'-trimethoxy-cis-stilbene trismethoxy inhibitor inhibition caco-2 caco 2 cells AHR antagonists aryl hydrocarbon receptors |
15.301954419889
|
| 580200 |
CTRP3 (human) EIA Kit
New
|
|
- |
|
|
|
2012-01-20
|
7.725669358266
|
ctrp3-human-eia-kit
|
Complement C1q TNF-related Protein 3
|
kits assays EIAs ELISAs enzymes immunoassays measures measurements complements C1q TNF-related tumors necrosis factor-relateds proteins 3 secreted glycoproteins morphogenesis metabolisms cells functions cellular paralog adiponectins adipocytes leukocytes blood chondrogenic differentiations bone cartilage angiogenesis ERF1/2 signaling signalling adipokines mice mouse humans recombinants suppresses suppression hepatic livers glucose sugar C6H12O6 output inhibition inhibits inhibitors gluconeogenesis levels normal ob/ob obese/obese antagonizes lipopolysaccharides LPS toll-like receptors 4 TLR4 competitive serums plasmas cultures supernatants |
7.725669358266
|
| 63500 |
Cytotrienin A
|
|
189010-85-3 |
≥95%
|
|
|
2009-07-06
|
22.799469613259
|
cytotrienin-a
|
|
anti-tumor anti-cancer apoptosis ROS caspace-3 p36 MBP kinase JNK |
22.799469613259
|
| 10009851 |
D-myo-Inositol-1,3,4,5,6-pentaphosphate (ammonium salt)
|
|
- |
>98%
|
|
|
2007-06-04
|
6.835635359115
|
d-myo-inositol-1-3-4-5-6-pentaphosphate-ammonium-salt
|
1,3,4,5,6-IP5 (sodium salt); Ins(1,3,4,5,6)P5
|
inositols phosphate IP5 signal transduction InsP phosphitidylinositol phospholipase C PLC phosphioinositide 3-kinase PI3-K Akt cancer angiogenesis PKB protein kinase B |
6.835635359115
|
| 11049 |
Echinomycin
New
|
|
512-64-1 |
≥98%
|
|
|
2012-03-21
|
41.796717171717
|
echinomycin
|
NSC 13502; SK 302B; NSC 526417; Antibiotic A 654I; Quinomycin A
|
11016-61-8 NSC13502 NSC526417 NSC-13502 NSC-526417 SK302B SK-302B hypoxia HIF-1 cancers neuroscience VEGF inhibitors inhibits inhibition genes expression glycolysis angiogenesis migration invasion cells DNA HIF-1α HIF-1β U215 hippocampal neurons myeloma melphalan |
41.796717171717
|
| 11332 |
Fumagillin
New
|
|
23110-15-8 |
≥95%
|
|
|
2012-02-22
|
0E-12
|
fumagillin
|
NSC 9168; Amebacilin
|
297-95-0 47721-00-6 47721-01-7 106215-84-3 746540-00-1 fugillin fumadil B fumagillin fumagillin DCH fumidil microsporidia inhibitors angiogenesis cancers cells growth proliferation genes expression fungus infection infectious diseases adipose tissues obesity Aspergillus fumigatus MetAP2 antibiotics |
0E-12
|
| 10010622 |
Genipin
|
|
6902-77-8 |
≥98%
|
|
|
2008-05-09
|
144.961325966851
|
genipin
|
(+)-Genipin
|
obesity diabeties glucose insulin mitochondria UCP2 pancreatic .beta. cells anti-inflammatory antiinflammatory angiogenesis inhibitors inhibits inhibition uncoupling proteins 2 un-coupling angiogenesis apotosis diabetes inflammation metabolism obesity |
144.961325966851
|
| 10009880 |
GW 590735
Exclusive
|
|
622402-22-6 |
≥98%
|
|
✓ |
2007-06-18
|
9.053149171270
|
gw-590735
|
|
PPAR PPAR.alpha. PPAR.BETA. PPAR.gamma. PPAR.delta. receptor transcription factors lipidtriglyceride TG lipoprotein VLDL ApoCIII ApoA1 HDL atherosclerosis endocrinology |
9.053149171270
|
| 10010559 |
HA-1077 (hydrochloride)
|
|
203911-27-7 |
≥98%
|
|
|
2008-09-03
|
53.702559852670
|
ha-1077-hydrochloride
|
Eril; Fasudil; AT-877
|
protein kinase inhibitors inhibits inhibition ROCK-II ROCKII PRK2 MSK1 MAPKAP-K1b vasodilation hypertension diabetes renal nephropathy cancers 105628-07-7 AT877 AT 877 hydrochloride dihydrochloride monohydrochloride HCl HA1077 HA 1077 |
53.702559852670
|
| 10347 |
HIF-1α Monoclonal Antibody (Clone H1α67)
|
|
- |
|
|
|
2011-05-09
|
40.105239410681
|
hif-1-monoclonal-antibody-clone-h1-67
|
Hypoxia Inducible Factor-1α
|
WBs western blots IHC immunohistochemistry antibodies HIF-1alpha HIF1a HIF-1a antisera serum cancers H1α67 transcription factors oxidative tumors EPAS-1 EPAS1 EPAS 1 DMOG 2,4-DPD desferrioxamine CoCl2 |
40.105239410681
|
| 13295 |
HNHA
|
|
926908-04-5 |
≥98%
|
|
|
2009-09-03
|
23.011531893520
|
hnha
|
Histone Deacetylase Inhibitor VI
|
inhibitors inhibits inhibition histones deacetylase HDACs cancers fibrosarcoma HT1080 cells hyperacetylation p21 genes expressions transcription cycles arrest tumor growth murine xenograph human umbilical vein endothelial HUVECs tubes formation migration vascular endothelial factors VEGF retinal neovascularization angiogenesis |
23.011531893520
|
| 10007502 |
Luminex® Thromboxane B2 Kit
|
|
- |
|
|
|
2009-07-13
|
37.424419889502
|
luminex-thromboxane-b2-kit
|
Luminex® TXB2 Kit
|
thromboxanes thromboxane A2 TXA2 metabolites urine in vivo measures kits luminex xMAP beads assays |
37.424419889502
|
| 13196 |
NSC 23766 (hydrochloride)
|
|
1177865-17-6 |
≥98%
|
|
|
2010-07-20
|
18.908674033149
|
nsc-23766-hydrochloride
|
|
733767-34-5 GTPases cells cycles growth proliferations cell-cell adhesions motility differentiation guanine nucleotides exchange factors GEFs inhibitors inhibits inhibition cell migration Aminoquinolines angiogenesis leukemia cancers gene expression Rac1 Inhibitor |
18.908674033149
|
| 13641 |
NVP-AEW541 (hydrochloride)
|
|
- |
≥98%
|
|
|
2010-07-28
|
41.979834254143
|
nvp-aew541-hydrochloride
|
|
475488-34-7 IGF-1R Insulin-like growth factor I receptors tyrosine kinases angiogenesis cells proliferation cancers inhibitors inhibition inhibits 701294-63-5 Ins-R NWT-21 Pyrroles |
41.979834254143
|
| 10565 |
NVP-BEZ235
|
|
915019-65-7 |
≥98%
|
|
|
2010-10-12
|
48.377927007512
|
nvp-bez235
|
|
phosphatidylinositols 3-kinases PI3Ks Akt/PKB mTORs cancers inhibitors inhibits inhibition angiogenesis genes expressions apoptosis differentiation rapamycin phosphatidyls inositols phosphatidylinositols-3-kinase Imidazoles BEZ235 |
48.377927007512
|
| 10011619 |
Terbinafine (hydrochloride)
|
|
78628-80-5 |
≥98%
|
|
|
2010-02-16
|
4.223204419890
|
terbinafine-hydrochloride
|
|
antifungals squalene epoxidase antitumor tumors antiangiogenic anticancer cancers inhibitors inhibits inhibition Naphthalenes |
4.223204419890
|
| 13044 |
Tranilast
|
|
53902-12-8 |
≥98%
|
|
|
2008-08-29
|
71.116731123388
|
tranilast
|
SB 252218; Rizaben; MK 341; Tranpro; N-(3',4'-Dimethyoxycinnamoyl)Anthranilic Acid
|
anti-inflammatory antiinflammatory angiogenesis PGDF TGF-.beta.1 TGF.beta.1 IL-8 IL8 PGE2 TXB2 antiallergenic anti-allergenic atherosclerosis vascular disease VEGF |
71.116731123388
|
| 71800 |
(Z)-Guggulsterone
|
|
39025-23-5 |
≥98%
|
|
|
2009-12-01
|
1.169042357274
|
-z-guggulsterone
|
|
anti flammatory cancers FXR bile acids LDL cholesterol tumors IL-6 STAT3 VEGF Akt |
1.169042357274
|