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Research Area · Drug Discovery

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Item Number Product Sizes & Pricing CAS Purity Image Exclusive Introduction Date Mojo Plain Text Name Synonyms Keywords
10008041 20S Proteasome Assay Kit - 2008-02-12 60.297624309392 20s-proteasome-assay-kit assays fluorescence fluorescent fluorometric cell-based assay cell based assay cba
10009856 7-AAD Cell Viability Assay Kit - 2008-10-29 14.545303867403 7-aad-cell-viability-assay-kit 7-Amino Actinomycin D Cell Viability Kit kits 7AAD measurement cells fixation blocking cytoxicity effects environmental toxins drug fluorescence fluorescent cell-based assays cell based assay cba
10006908 Adipogenesis Assay Kit - 2006-08-18 79.845113008538 adipogenesis-assay-kit obese obesity cells cycle differentiation inhibits inhibitors inhibition adipocytes cancers origin 3T3-L1 model drug screening adipokines endocrinology cell-based assays cell based assay cba
10009381 Adipolysis Assay Kit - 2007-07-30 41.588784530386 adipolysis-assay-kit obese obesity cells cycle differentiation inhibits inhibitors inhibition adipocytes cancers origin 3T3-L1 model drug screening adipokines lipolysis 3T3L1 kits assays FFA adipocytes endocrinology cell-based assay cell based assay cba
600140 Autophagy/Cytotoxicity Dual Staining Kit - 2009-07-14 90.794762430939 autophagy-cytotoxicity-dual-staining-kit assays kits measuring measurement MDC cell-based autophagy cells cytotoxicity staining autofluorescent autofluorescence substances multilamellar body bodies ions trapping mechanisms membranes lipids probes autophagic vacuoles cultured degradation digestion intracellular lysosomes organelles misfolded proteins microorganisms cytoplasms double membranes autophagosomes autolysosomes homeostasis dysregulation cancers infections aging degenerative diseases stress death apoptosis
600070 BACE Inhibitor Screening Assay Kit - 2009-03-26 49.041141804788 bace-inhibitor-screening-assay-kit β-Secretase Inhibitor Screening Assay Kit inhibitors inhibition inhibits assays kits β-sites .beta.-sites b-sites APP cleaving enzymes β-amyloids .beta.-amyloids b-amyloids peptides Ab A.beta. brain neurodegeneration Alzheimer's Diseases AD proteolytic cleavages precursors β-secretases b-secretases γ-secretases .gamma.-secretases g-secretases membranes aspartic C-terminal C-terminus fragments proteolysis therapeutics therapy cascade pathogenesis mice mouse murine transgenics cholinergic dysfunctions HIV humans fluorescents fluorescences fluorometer assays
10009853 CFSE Cell Division Assay Kit - 2010-01-15 64.210537139349 cfse-cell-division-assay-kit derivative carboxyfluorescein diacetate, succinimidyl ester CFDA-SE cells proliferation growth factors receptors surfaces signaling molecules transcription factors DNA deoxyribonucleases proteins divisions cascades human pathological diseases cancers cell-tracing fluorescent fluorescence dyes proliferative activity parent generations daughter acetate groups molecules cleaved background unstained staining CFSE-labeled radioactivity radioactive labeling divisions inductions inhibitors inhibits inhibitions in vitro models flow cytometry fluorochromes fluorescein
760111 Colorimetric COX (ovine) Inhibitor Screening Assay Kit - 178.933058563535 colorimetric-cox-ovine-inhibitor-screening-assay-kit cyclooxygenases cox-1 cox-2 pghs-1 pghs-2 cox1 cox2 pghs1 pghs2 prostaglandins synthases synthase-1 synthase-2 inhibition inhibitors assays screens peroxidase colorimetrically analysistools:eia
700100 COX Fluorescent Inhibitor Screening Assay Kit - 2008-07-08 131.696441988950 cox-fluorescent-inhibitor-screening-assay-kit Cyclooxygenase Fluorescent Inhibitor Screening Assay Kit cyclooxygenases synthases enzymes cox-1 cox1 cox-2 cox2 prostaglandins PGs synthase-1 synthase-2 pghs-1 pghs1 pghs-2 pghs2 assays kits peroxidase activity cellular homeostasis antiinflammatory NSAIDs nonsteroidal anti-inflammatory drugs fluorescence human recombinant ovine isozyme-specific inhibits inhibitors inhibition ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin
560131 COX Inhibitor Screening Assay Kit - 280.758003157064 cox-inhibitor-screening-assay-kit enzyme immunoassays kits measures EIAs ELISAs COX1 COX-1 COX2 COX-2 PGHS1 pghs-1 pghs2 pghs-2 prostaglandin synthases inhibitors cyclooxygenase analysistools:eia assays cox inhibitior kit
560101 COX (ovine) Inhibitor Screening Assay Kit - 89.486167127071 cox-ovine-inhibitor-screening-assay-kit enzyme immunoassays kits measures EIAs ELISAs COX1 COX-1 COX2 COX-2 PGHS1 pghs-1 pghs2 pghs-2 prostaglandin synthases inhibitors cyclooxygenases sheep screens assays cox inhibitior kit
600270 CYP3A4 Induction STEP Reporter Assay Kit (Luminescence) - 2010-03-04 95.533631500482 cyp3a4-induction-step-reporter-assay-kit-luminescence kits assays measures measurements cytochromes P450 CYP450 heme-thiolates monoxygenases metabolizes endogenous xenobiotics pollutants pollution environment drugs metabolism pharmacokinetics therapeutics CYP1A2 CYP2C9 CYP2C19 CYP2D6 inhibits inhibitors inhibition toxicity human hepatocytes cultured cells lines enzymes high-throughput Surface Transfection and Expression Protocol transient transfection technology Originus, Inc. University of Michigan US patents USPT 6897067 6902933 7056741 DNA deoxyribonucleic acids recombinant proteins plates endocytosis solution-phase plasmids Secreted Alkaline Phosphatases SEAP promoter Pregnane X Receptor PXR Hepatocyte Nuclear Factor 4α HNF4α culture mediums luminescence-based alkaline phosphatases rifampicin HNF-4α HNF-4.alpha. HNF-4alpha HNF4.alpha. HNF 4alpha HNF 4.alpha. HNF 4alpha
700390 Demethylase (Jumonji-type) Activity Assay Kit New - 2010-05-26 0E-12 demethylase-jumonji-type-activity-assay-kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC JHDM1 JHDM2 JHDM3 JARID1 UTX/UTY cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3
700210 DPP (IV) Inhibitor Screening Assay Kit - 2009-05-27 115.718314917126 dpp-iv-inhibitor-screening-assay-kit Dipeptidyl exopeptidases IV DPPIV DPP4 enzymes CD26 cluster of differentiation T-cells activation antigens adenosine deaminase complexing 2 membrane-bound glycoproteins immune regulation signal transduction apoptosis kidneys small intestines placentas humans serums seminal fluids proteolytic derivatives serines X-prolines X-alanines dipeptides N-terminus N-terminal polypeptides growth factors chemokines neuropeptides vasoactive inhibitors inhibits inhibition oral antidiabetic agents glucose homeostasis glucoregulatory hormones glucose-dependent insulinotropics GIP glucagon-like peptide-1 GLP-1 gastric therapeutics Type 2 tumors cancers markers neoplasms assays kits measures measurements fluorescences fluorescent fluorogenics substrates Gly-Pro-Aminomethylcoumarin AMC
10005196 FAAH Inhibitor Screening Assay Kit - 2008-09-05 131.968109707972 faah-inhibitor-screening-assay-kit Fatty Acid Amide Hydrolase Inhibitor Screening Assay Kit neurochemistry neuroscience endocannabinoids lipid signaling regulatory arachidonoylethanolamides AEAs 2-arachidonoyl glycerol 2-AG G Protein Coupling Receptors GPCRs CB1 motor controls cognition emotional responses homeostasis CB2 peripheral tissues modulators autonomic nervous systems immune microcirculation enzymes fatty acids amides hydrolases monoacylglycerols lipases MGL MAGL serines inhibitors pain obesity neurological diseases agonists fluorescence-based screening hydrolyzes AMC-arachidonoyl 7-amino-4-methylcoumarin fluorophores assays kits
10006515 HAT Inhibitor Screening Assay Kit - 2006-12-06 14.707366482504 hat-inhibitor-screening-assay-kit Histone Acetyltransferase Inhibitor Screening Assay Kit therapeutics histones p300/CBP-Associated Factors pCAF GNAT GCN5-related N-acetyltransferases acetylates lysines N-terminal terminus tails H3 H4 tumors suppressor genes PTEN human cancers apoptosis fluorescence fluorescent inhibitors fluorometric assays
10011564 HDAC1 Inhibitor Screening Assay Kit - 2008-04-10 27.379171270718 hdac1-inhibitor-screening-assay-kit HDAC 1 histones deacetylases lysines residues chromatin condensation transcriptional repression fluorescence deacetylation fluorescent inhibits inhibition enzymes license:cyclex fluorometric assays cancer
700230 HDAC8 Inhibitor Screening Assay Kit - 2009-05-15 11.367403314917 hdac8-inhibitor-screening-assay-kit Histone Deacetylase 8 Inhibitor Screening Assay Kit histone deacetylases inhibits inhibitors inhibition angiogenesis cycling apoptosis differentiation tumors proliferation anticancers genes epigenetic trichostatin A human class I tissues nucleus cytosolic smooth muscle neuroblastoma pathogenesis kits assays measures measurement fluorescent fluorescence-based
600150 HDAC Cell-Based Activity Assay Kit - 2009-11-09 19.212996260952 hdac-cell-based-activity-assay-kit Histone Deacetylase Cell-Based Activity Assay Kit assays kits measuring measurement histones deacetylases lysines residues chromatin condensation transcriptional repression fluorescence deacetylation fluorescent inhibits inhibition enzymes fluorometric assays cancer modulators whole cells proteins lysine-specific HDAC1 homogenous inhibitor/activator TSA
500340 Human Serum Albumin EIA Kit - 2009-07-16 84.208135359116 human-serum-albumin-eia-kit Human Serum Albumin EIA Kit; HSA ELISA Kit solid plates EIAs ELISAs enzymes immunoassays kits measures measurement renal kidneys blood proteins serums osmotic pressure buffering pH hormones fatty acids transports transportation microaluminuria macroalbuminuria disease non-diabetic nephropathy cardiovascular morbidity mortality creatinine assays
700360 JMJD2A Inhibitor Screening Assay Kit New - 2010-05-25 0E-12 jmjd2a-inhibitor-screening-assay-kit Jumonji Domain Containing 2A Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC JHDM1 JHDM2 JHDM3 JARID1 UTX/UTY cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated
700370 JMJD2D Inhibitor Screening Assay Kit New - 2010-05-25 0E-12 jmjd2d-inhibitor-screening-assay-kit Jumonji Domain Containing 2D Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation FLJ10251 replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated
10008882 LDH Cytotoxicity Assay Kit - 2006-12-15 125.354493554327 ldh-cytotoxicity-assay-kit Lactate Dehydrogenase Cytotoxicity Assay Kit cells death apoptosis necrosis measuring measurement cystolic enzymes cells membranes integrity cancer cell-based assays cell based assay cba
500001 Lipid Droplets Fluorescence Assay Kit - 2009-05-28 33.674033149171 lipid-droplets-fluorescence-assay-kit lipids droplets storage organelles cytoplasms eukaryotic cells mammalian adipocytes steroidogenic fatty acids metabolism membranes synthesis phospholipids cholesterols steroids PAT proteins Perilipin adipophilin tail-interacting TIP 47 intracellular homeostasis trafficking signaling immunopathological inflammation anti-inflammatory mediators leukocytes therapy assays kits measures measurements fluorescences fluorescent biogenesis Nile Red microscopy flow cytometry plates readers
760700 Lipoxygenase Inhibitor Screening Assay Kit - 64.737455801105 lipoxygenase-inhibitor-screening-assay-kit LO Inhibitor Screening Assay Kit 12-LOs 15-LOs 15-lipoxygenases activity hydroperoxides assays kits inhibitors 12-lipoxygenases analysistools:lis
700120 LSD1 Inhibitor Screening Assay Kit - 2008-10-16 7.456837016574 lsd1-inhibitor-screening-assay-kit Lysine-Specific Demethylase 1 lysines 4 demethylases histones residues repression transcription chromosomal DNA chromosomes inhibits inhibitors inhibition tumors suppressors activity cells cycles progression cancers fluorescent fluorescence enzymes enzymatic reactions H2O2 hydrogens peroxides peptides N-terminal tails H3 horseradish peroxidases ADHP resorufins assays
600310 Lysosome/Cytotoxicity Dual Staining Kit New - 2010-06-15 5.555555555556 lysosome-cytotoxicity-dual-staining-kit lysosomes membrane-bound acidic intracellular compartments cells waste products fats carbohydrates proteins macromolecules mobilize recycle organelles microorganisms animals leukocytes degradative enzymes hydrolases pH 5 cytoplasm homeostasis Tay-Sachs diseases arthritis neurodegeneratives Parkinson's brains cathepsin D genes therapeutics kits assays measures measurements 4-Nitro-7-(1-piperazinyl)-2,1,3-benzoxadiazole NBD-PZ membranes permeable carboxylic acids luminal cultured propidium iodides death chloroquine inhibitors positive controls fluorescence fluorescent microscopy plates reader detections flow cytometry
600180 Melanocortin-3 Receptor STEP Reporter Assay Kit (Luminescence) - 2010-01-05 30.470564763658 melanocortin-3-receptor-step-reporter-assay-kit-luminescence MC3R MC-3R melanocortins petides hormones proopiomelanocortins pituitary CNS central nervous systems skin placenta tissues MCR receptors G protein-coupled GPCRs cAMP Adenosine 3',5' cyclic mononucleotides messenger signal transduction pathways melanocortin-3 hypothalmus homeostasis fat lean mass hyperphagia MC4R melanocortin-4 adiposity MC3R-knockout mice mouse murine fatty acids oxidations blood pressure hypertension obesity glucose metabolisms insulin insensitivity agonists ligands Surface transfection and expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated endocytosis solution-phase co-transfection plasmids secretory alkalines phosphatases substrates SEAP proteins lipids signal transduction luminescence-based cell-based assays kits CBAs high-throughput screening a-MSH alpha-MSH α-MSH
600190 Melanocortin-4 Receptor STEP Reporter Assay Kit (Luminescence) - 2010-01-05 30.470564763658 melanocortin-4-receptor-step-reporter-assay-kit-luminescence MC4R MC-4R melanocortins petides hormones proopiomelanocortins pituitary CNS central nervous systems skin placenta tissues MCR receptors G protein-coupled GPCRs cAMP Adenosine 3',5' cyclic mononucleotides messenger signal transduction pathways melanocortin-3 hypothalmus homeostasis fat lean mass hyperphagia MC4R melanocortin-4 adiposity MC3R-knockout mice mouse murine fatty acids oxidations blood pressure hypertension obesity glucose metabolisms insulin insensitivity agonists ligands sexual function antagonists fever suppression inflammatory mediators in vivo Surface transfection and expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated endocytosis solution-phase co-transfection plasmids secretory alkalines phosphatases substrates SEAP proteins lipids signal transduction luminescence-based cell-based assays kits CBAs high-throughput screening a-MSH alpha-MSH α-MSH
700140 Methyltransferase Colorimetric Assay Kit - 2009-04-07 23.015653775321 methyltransferase-colorimetric-assay-kit MT Colorimetric Assay Kit assays kits measures measuring monitoring monitors MTs methylation signal transduction biosynthesis repair gene silencing chromatin regulation S-adenosylmethionine SAM-dependent methyltransferases enzymatic cofactors AdoMet donor modifications DNA Alzheimer's diseases depression Parkinson's multiple sclerosis liver failure cancers enzyme-coupled AdoHcy positive control S-adenosylhomocysteine
700150 Methyltransferase Fluorometric Assay Kit - 2009-04-08 22.094267955800 methyltransferase-fluorometric-assay-kit MT Fluorometric Assay Kit assays kits measures measuring monitoring monitors MTs methylation signal transduction biosynthesis proteins repair gene silencing chromatin regulation S-adenosylmethionine SAM-dependent methyltransferases enzymes enzymatic cofactors AdoMet donor proteins modifications DNA Alzheimer's diseases depression Parkinson's multiple sclerosis liver failure cancers enzyme-coupled AdoHcy positive control S-adenosylhomocysteine
705192 Monoacylglycerol Lipase Inhibitor Screening Assay Kit - 2009-10-22 70.744733326111 monoacylglycerol-lipase-inhibitor-screening-assay-kit MAGL; MGL neuroscience neurochemistry inhibitors inhibiting inhibition inhibits endocannabinoids serines hydrolases pain obesity monoglycerol
10009365 MTT Cell Proliferation Assay Kit - 2007-02-15 85.536528545120 mtt-cell-proliferation-assay-kit assays kits screen measures measurements cells cellular growth factors signaling signalling molecules transcription DNA pathological cancers aging cycles progression regulatory cytokines mitogens drugs inductions inhibitors inhibits inhibitions in vitro plasma membranes formazan intracellular NAD(P)H-oxidoreductases NADPH-oxidoreductases proteins enzymes enzymatic cleavage microtiter plates tertrazolium salts mitochondrial dehydrogenases cancer cell-based assay cell based assay cba
600330 Multi-Parameter Apoptosis Assay Kit New - 2010-08-18 5.555555555556 multi-parameter-apoptosis-assay-kit assays kits measures measurements apoptosis cells death cycles tissues homeostasis dysregulation neurodegenerative diseases ischemic damages autoimmune disorders cancers drugs discovery signaling pathways membranes phospholipids phosphatidylserines phosphatidylethanolamines leaflets bilayers externalizations residues plasma phospholipids binding proteins fluorochrome-labeled fluorochromes annexin V fluorescence microscopy flow cytometry FC plate readers TUNEL TdT-mediated dUTP Nick-End Labeling analysis ISEL in situ end labeling DNA deoxyribonucleic acids mitochondrial transmembranes tetramethylrhodamines ethyls esters TMRE lipophilics probes laddering detection fragmentation FITC-conjugated fluoresceins
700170 Myeloperoxidase Inhibitor Screening Assay Kit - 2009-04-14 24.480939226519 myeloperoxidase-inhibitor-screening-assay-kit MPO Inhibitor Screening Assay Kit heme peroxidases azurephilic granules leukocytes neutrophils monocytes tissues macrophages chlorides hydrogen peroxides H2O2 Cl- hypochlorous acids acute chronic vascular inflammatory diseases cardiac therapeutics cycles fluorescence fluorescent assays kits measures measurement crude cells lysates purified enzymes ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin 2-[6-(4-aminophenoxy)-3-oxo-3H-xanthen-9-yl]-benzoic acid APF -OCl assays
600240 Orexin 1 Receptor STEP Reporter Assay Kit (Luminescence) New - 2010-03-31 0E-12 orexin-1-receptor-step-reporter-assay-kit-luminescence OX1R hypercretins 1 orexins 2 A orexin-2 systems regulates regulator sleep wake cycles feeding cardiovascular autonomic hypothalamic neuropeptides Orexins A Orexins B gut hormones secretions hypothalamus midbrains brainstems G protein-coupled receptors GPCRs orexin-1 OX1R orexin-2 OX2R orexin-A orexin-B sleep disorders narcolepsy humans animals rodents energy homeostasis pain stress antagonists drugs addictions withdrawals therapeutics obesity Surface transfection expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated luminescent secretory alkaline phosphatases SEAP signal transduction cascades culture medium luminescence-based high throughput screening screens agonists
600250 Orexin 2 Receptor STEP Reporter Assay Kit (Luminescence) New - 2010-03-31 0E-12 orexin-2-receptor-step-reporter-assay-kit-luminescence OX2R hypercretins 1 orexin 2 systems regulates regulator sleep wake cycles feeding cardiovascular autonomic hypothalamic neuropeptides Orexins A Orexins B gut hormones secretions hypothalamus midbrains brainstems G protein-coupled receptors GPCRs orexin-1 OX1R orexin-2 OX2R orexin-A orexin-B sleep disorders narcolepsy humans animals rodents energy homeostasis pain stress antagonists drugs addictions withdrawals therapeutics obesity Surface transfection and expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated luminescent secretory alkaline phosphatases SEAP signal transduction cascades culture medium luminescence-based high throughput screening screens agonists
10004380 PAF Acetylhydrolase Inhibitor Screening Assay Kit - 2004-03-29 48.158994475137 paf-acetylhydrolase-inhibitor-screening-assay-kit PAF-AH Inhibitor Screening Assay Kit; Lp-PLA2 Inhibitor Screening Assay Kit platelet-activating factors hypotension inflammations allergys PAFAH atherosclerosis heart diseases measures kits inhibitors PAFs assays paf elisa kit
10004916 PBMC Fluorescent Titer Assay Kit - 2006-07-21 0E-12 pbmc-fluorescent-titer-assay-kit SPI-Bio spibio kits enzyme immunoassays D05003 assays fluorescence fluorescent fluorometric
789201 P-Glycoprotein Drug Interaction Assay Kit - 0E-12 p-glycoprotein-drug-interaction-assay-kit P-gp Drug Interaction Assay Kit glycoproteins pharmacokinetics cellular detoxification ATPase ADPase assays kits interactions drugs transport photodetection spi-bio spibio D5001
500290 Phagocytosis Assay Kit (IgG FITC) - 2009-04-09 95.458651933702 phagocytosis-assay-kit-igg-fitc kits assays measuring measurement ingestion killing phagocytic leukocytes defense pathogens microbe-innate immune cytoskeletal rearrangement membrane trafficking microbial mechanisms pro-inflammatory anti-inflammatory cytokines chemokines apoptosis antigen immune systems pathological Multiple Sclerosis Alzheimer's diseases atherosclerosis bacterial fungal infections in vitro fluorescently opsonizing latex beads fluorescently-labeled flow cytometry cytometric analysis quantification cell-based assay cell based assay cba
10007685 PPARγ FP-Based Ligand Screening Assay Kit - Green - 2009-07-16 60.499944751381 ppar-fp-based-ligand-screening-assay-kit-green Peroxisome Proliferator-activated Receptor γ FP-Based Ligand Screening Assay Kit - Green peroxisomes proliferator-activated receptors PPARs proliferator activated PPARgamma PPAR.gamma. PPARg PPARγ PPAR-γ PPAR-gamma gamma g γ .gamma. PPAR-.gamma. PPAR-g kits assys atherosclerosis TF diabetes drugs discovery discover endocrinology high throughput screens screening inflammations inhibitors inhibits inhibition metabolic syndromes metabolism nuclear receptors fluorescence FP-based FP based base ligands probes proteins isoforms γ1 γ2 γ-1 γ-2 1 2 adipose tissues colon immune systems retinas adipogenesis cells cellular differentiation insulin sensitization cancers fatty acids FAAH arachdionic 15-deoxy-DELTA12,14-prostaglandin 15-deoxy-DELTA12,14-PGs 15-deoxy-DELTA12,14-PGJ2 15 deoxy DELTA 12,14 PGs prostaglandins PGJ2 15-deoxy-Δ12,14-PGs 15-deoxy-Δ12,14-prostaglandins 15-deoxy-Δ12,14-PGJ2 15-deoxy-D12,14-prostaglandins 15-deoxy-D12,14-PGs 15-deoxy-D12,14-PGJ2 15-deoxy-.DELTA.12,14-prostaglandins 15-deoxy-.DELTA.12,14-PGs 15-deoxy-.DELTA.12,14-PGJ2 J2 thiazolidinediones TZD pioglitazone rosiglitazone agonists hyperglycemia hyperinsulinemia hypertriglyceridemia types 2 antidiabetics diabetes oral antagonists
500581 Prostaglandin D2 FPIA Kit - Green - 2004-11-16 61.908493219487 prostaglandin-d2-fpia-kit-green PGD2 Fluorescence Polarization Immunoassay - Green PGD2 metabolites prostaglandins immunoassays HTS high-throughput kits screenings rapid measurements assays
10007835 Prostaglandin D2 FPIA Kit - Red - 2007-09-07 101.043268876611 prostaglandin-d2-fpia-kit-red PGD2 Fluorescence Polarization Immunoassay - Red PGD2 metabolites prostaglandins immunoassays HTS high-throughput kits screenings rapid measurements assays
600007 Prostaglandin D Synthase (hematopoietic-type) FP-Based Inhibitor Screening Assay Kit - Green - 2009-01-21 82.026804788213 prostaglandin-d-synthase-hematopoietic-type-fp-based-inhibitor-screening-assay-kit-green H-PGDS FP-Based Inhibitor Screening Assay Kit - Green; Prostaglandin D Synthase (hematopoietic-type) Fluorescence Polarization-Based Inhibitor Screening Assay Kit - Green assays kits measures measurements FPs fluorescent fluorescences polarizations polarization-based inhibitors inhibits inhibition prostaglandins synthases pgs H-PGDS PGD2 lipocalin-types L-PGDS allergies allergy allergic inflammatory inflammations reactions mast Th2 microglia necrotic muscles fibers apoptotic smooth HQL-79 tranilast guinea pigs lungs tissues pyrimidines amides amide-based single step fluoresceins probes Z' dynamic ranges mP units BSPTfluorescently-labeled HPGDS H-PGDS assays
10006593 Prostaglandin D Synthase (hematopoietic-type; human recombinant) - >95% 2005-02-16 29.085078926597 prostaglandin-d-synthase-hematopoietic-type-human-recombinant Hematopoietic-PGDS; H-PGDS; PGD Synthase (hematopoietic-type; human recombinant) prostaglandins synthases PGDs PGD2 HPGDS H-PGDS enzymes peripheral tissues antigen-presenting cells mast megakaryocytes glutathiones glutathione-S-transferases allergen allergy allergic mediators
10006595 Prostaglandin D Synthase Inhibitor Screening Assay Kit - 2005-08-31 54.944638253091 prostaglandin-d-synthase-inhibitor-screening-assay-kit PGDS Inhibitor Screening Assay Kit prostaglandins synthases inhibitors PGDS assays hematopoietic-types lipocalin-types pro-inflammatory mediators allergic allergy allergies allergens activity inhibitors inhibition inhibits H-PGDS L-PGDS
10006270 Renin Inhibitor Screening Assay Kit - 2005-05-04 64.085943172849 renin-inhibitor-screening-assay-kit Protease measurement assays aspartyl renal juxtaglomerular cells sodium depletion blood volume pressure .beta.-adrenergic stimulation angiotensinogens angiotensins I II converting ACE monomeric zinc metalloenzymes vascular endothelium messengers RAS vasoconstrictor peripheral hypertension receptors blockers fluorescence fluorescent fluorometric atherosclerosis endocrinology
600260 Secreted Alkaline Phosphatase Reporter Gene Assay Kit (Luminescence) New - 2010-04-27 0E-12 secreted-alkaline-phosphatase-reporter-gene-assay-kit-luminescence SEAP Reporter Gene kits assays measuring measurement phosphatases genes expression transfected cells culture mediums intracellular mRNA messenger ribonucleic acids proteins kinetics chromogenic substrates p-nitrophenyl para-nitrophenyl phosphates pNPP chemiluminescence chemiluminescent detections AP
700270 SET7/9 Methyltransferase Inhibitor Screening Assay Kit - 2009-12-04 8.851754409264 set7-9-methyltransferase-inhibitor-screening-assay-kit methyltransferases SET Domain-containing Protein 7/9 lysines 7 KMT7 methylation signal transduction biosynthesis proteins repair genes silencing chromatins S-adenosylmethionine SAM AdoMet methyl donors Alzheimer's depression Parkinson's Diseases multiple sclerosis liver cancers substrates histones histone 3 lysine residue 4 H3K4 p53 transcription factors TAF10 mono-methylated mono-methylase DNA damage acetylation human tumorigenesis inhibitors acceptor peptides S-adenosylhomocysteine S-ribosylhomocysteine adenine nucleosidase hypoxanthine deaminase urate hydrogen peroxide H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin fluorescence measures measurement assays kits
700350 SET8 Methyltransferase Inhibitor Screening Assay Kit New - 2010-03-09 128.769140822226 set8-methyltransferase-inhibitor-screening-assay-kit SET domain-containing (lysine methyltransferase) 8; PR-Set7; SETD8 assays kits measures measurement methyltransferases MTs inhibits inhibitors inhibition methylation signal transduction biosynthesis protein repair genes silencing chromatins regulation S-adenosylmethionine (SAM)-dependent AdoMet DNA deoxyribonucleic acids Alzheimer's diseases depression Parkinson's multiple sclerosis livers cancers KMT5A lysines PR-Set 7 methylates histones H4 residues 20 H4K20 transcriptional p53 tumors suppressors tumorigenesis inhibits inhibition inhibitors peptides S-adenosylhomocysteines S-ribosylhomocysteines adenines nucleosidases hypoxanthines deaminases hydrogen peroxides H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazines fluorescent fluorescence resorufin
700280 SIRT2 Direct Fluorescent Screening Assay Kit - 2009-12-10 12.508674010897 sirt2-direct-fluorescent-screening-assay-kit Nucleosomes chromosomal deoxyribonucleases DNA histones H2A H2B H3 H4 octameric cores transcription amino termini acetylation phosphorylation methylation ε-amino lysines acetyltransferases HATs chromatins genes activation deacetylases HDACs catalyzes hydrolytic acetyls sirtuins trichostatins A-insensitive lysyl-deacetylases class III catalyzes deacetylation nicotinamides O-acetyl-ADP-ribose NAD+ human SIRT1 SIRT2 SIRT3 SIRT4 SIRT5 SIRT6 SIRT7 cytoplasmic proteins H4 lysine-16 lysine-40 α-tubulin a-tubulin alpha-tubulin HDAC6 microtubules mitotic chromosomal hyperpolid cells tissues skeletal muscle heart oligodendroglia brain tumor suppressor gliomas Down-regulation gene chromosomal region diagnostic marker fluorescence-based inhibitors activators p53 Gln-Pro-Lys-Lys(ε-acetyl)-AMC recombinant NAD+ fluorescent fluorescence kits assays measures measurement
10011566 SIRT3 Direct Fluorescent Screening Assay Kit - 2008-08-21 16.213853591160 sirt3-direct-fluorescent-screening-assay-kit SIRT 3 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human mitochondrial proteins mitochondrias localization matrix-processing peptidase translocated nucleus cells cellular stress overexpression mice mouse murine caloric restriction up-regulates expression levels white brown adipose tissue BAT cold exposure PGC-1a PGC-1alpha PGC-1.alpha. UCP1 modulates adaptive thermogenesis deacetylation activation acetyl coenzymes A synthetase 2 AceCS2 catalyzes acetate CoA ketogenesis ATP direct genetic link longevity mutations genes enhancers marker life extension cellular metabolic control whole-body metabolism chronic diseases dysfunction neuronal pathogenesis neurodegenerative cancers aging apoptosis screening fluorescence activators fluorescent fluorometric
600090 Soluble Epoxide Hydrolase Cell-Based Assay Kit - 2009-05-14 58.766314127860 soluble-epoxide-hydrolase-cell-based-assay-kit sEH Cell-Based Assay Kit kits assays measuring measurement mammalian epoxides α/β-hydrolases enzymes catalyzes hydrolysis exogenous endogenous vicinal diols homodimers C-terminal N-terminal domains vasodilatory vasodilation anti-inflammatory hypertension vascular inflammation inhibitors therapeutics fluorescence-based fluorescent whole cells Epoxy Fluor 7 6-methoxy-2-naphthaldehyde AUDA
10011671 Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit - 2009-02-24 73.638447513812 soluble-epoxide-hydrolase-inhibitor-screening-assay-kit sEH Inhibitor Screening Assay Kit epoxides hydrolases sEHs inhibits inhibition assays kits fluorescence-based catalyzes hydrolysis exogenous endogenous vicinal diols substrates EETs epoxyeicosatrienoic acids vasodilatory vasodilation anti-inflammatory molecules therapy therapeutics hypertension vascular diseases PHOME (3-phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester 6-methoxy-2-naphthaldehyde excitation emission wavelengths a/b-hydrolases alpha/beta-hydrolases .alpha./.beta.-hydrolases enzymes homodimers C-terminal C-terminus animals models cyanohydrins cyanide ions
700330 Sphingomyelinase Inhibitor Screening Assay Kit - 2010-02-09 90.860927587085 sphingomyelinase-inhibitor-screening-assay-kit assays kits measures measuring measurementsphingomyelinases SMases hydrolases enzymes sphingolipids metabolisms DNase I superfamily phosphocholines ceramides cellular cells stress pathophysiological lysosomal digestion ceramide-mediated signal transductions cytokine-induced apoptosis differentiation immune inflammatory lipoproteins aggregation vessels atherogenesis intracellular cholesterols trafficking acidic neutral proliferation depressive disorders neurodegenerative disorders strokes Alzheimer's dementia diseases therapeutics cleavage conjugates free thiols
10004883 sPLA2 (Type V) Inhibitor Screening Assay Kit - 2004-05-07 49.962603591160 spla2-type-v-inhibitor-screening-assay-kit Secretory Phospholipase A2 (Type V) assays measures kits inhibition inhibitors phospholipases inflammation eicosanoids colorimetric sPLA2s enzymes diheptanoyl thio-pc
10012643 Steatosis Colorimetric Assay Kit Exclusive - 2008-07-01 18.161988950276 steatosis-colorimetric-assay-kit kits fatty liver lipids cells obesity assy kits measuring measurement cell-based assays cell based assay cba
10008883 WST-1 Cell Proliferation Assay Kit - 2006-09-07 33.206016837673 wst-1-cell-proliferation-assay-kit assays cells proliferation induction inhibitors inhibition inhibits growth factors signaling signalling molecules cycles regulatory factors cytokines mitogens drugs microtiter plates in vitro enzymes enzymatic cleavage tertrazolium salts formazan cellular mitochondrial dehydrogenases screen kits measures measurements cancers cell-based assay cell based assay cba
10010199 WST-8 Cell Proliferation Assay Kit - 2007-09-11 60.442836095763 wst-8-cell-proliferation-assay-kit assays cells proliferation induction inhibitors inhibition inhibits growth factors signaling signalling molecules cycles regulatory factors cytokines mitogens drugs microwell plates in vitro enzymes enzymatic cleavage tertrazolium salts formazan cellular mitochondrial dehydrogenases screen kits measures measurements special:quarterly specialdiscount:50 specialstart:2007-12-01 specialend:2008-02-29 cell-based assay cell based assay cba
10010200 XTT Cell Proliferation Assay Kit - 2007-09-11 41.906003683241 xtt-cell-proliferation-assay-kit assays cells proliferation induction inhibitors inhibition inhibits growth factors signaling signalling molecules cycles regulatory factors cytokines mitogens drugs microtiter plates in vitro enzymes enzymatic cleavage tertrazolium salts formazan cellular mitochondrial dehydrogenases screen kits measures measurements special:quarterly specialdiscount:50 specialstart:2007-12-01 specialend:2008-02-29 cell-based assay cell based assay cba
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