| 10007975 |
(±)11,12-DHET-d11
Exclusive |
|
- |
≥99% deuterated product
|
|
✓ |
2008-03-17
|
30.395856353591
|
-11-12-dhet-d11
|
(±)11,12-DiHETrE-d11
|
epoxides epoxygenases DHT hydrolases (+/-)11,12-DiHETrEs deuterated epoxide hydrolase deuterated deuterium |
| 10006413 |
(±)11(12)-EET-d11
Exclusive |
|
- |
≥99% deuterated product
|
|
✓ |
2008-03-25
|
41.125064456722
|
-11-12-eet-d11
|
(±)11(12)-EpETrE-d11
|
epoxides epoxygenases 11,12-EETs cytochrome P450 (+/-)11,12-EpETrEs (+/-)11(12)-EpETrEs deuterated deuterium |
| 10004549 |
11β-Hydroxysteroid Dehydrogenase (Type 2) Polyclonal Antibody
|
|
- |
|
|
|
2005-10-05
|
9.806104972376
|
11-hydroxysteroid-dehydrogenase-type-2-polyclonal-antibody
|
Corticosteroid 11β-Dehydrogenase Isozyme 2; 11β-HSD2
|
proteins diseases antibodies antisera antiserum WB western blots blotting ICC immunocytochemistry corticosteroids regulations sodium homeostasis pathophysiology hypertension converts converting cortisol inactive cortisone mutations genes encoding induction hypertension hypokalemia syndromes mineralcorticoid excess mRNA expressed placenta target tissues kidneys mouse murine tissue-specific developmentally regulated glucocorticoid-medicated maturation 11b-HSD 11beta-HSD 11.beta.-HSD 11b HSD 11b-hydroxysteroid 11beta-hydroxysteroid endocrinology immunoblotting |
| 10008040 |
(±)14,15-DHET-d11
|
|
- |
≥99% deuterated product
|
|
|
2008-03-18
|
64.776519337017
|
-14-15-dhet-d11
|
(±)14,15-DiHETrE-d11
|
epoxides epoxygenases DHT hydrolases (+/-)14,15-DiHETrEs deuterated epoxide hydrolase deuterium |
| 10004946 |
14,15-EE-5(Z)-E
Exclusive |
|
519038-92-7 |
>98%
|
|
✓ |
2007-01-15
|
70.353480662983
|
14-15-ee-5-z-e
|
14,15-Epoxyeicosa-5(Z)-enoic Acid
|
14,15-EpETrE 14,15-EETs antagonists hypertension vasodilation vasodilator vasoconstriction vasoconstrictor EDHT endothelium-derived hyperpolarizing factor U46619 bovine arteries endocrinology EEZE |
| 10010486 |
14,15-EE-8(Z)-E
Exclusive |
|
519038-93-8 |
≥98%
|
|
✓ |
2008-11-03
|
23.675408839779
|
14-15-ee-8-z-e
|
14,15-Epoxyeicosa-8(Z)-enoic Acid
|
14,15-EETs 14,15-EpETrEs vasodilation vascular disease hypertension EEZE |
| 10009286 |
(±)14(15)-EET-SI
|
|
218461-97-3 |
>95%
|
|
|
2007-05-14
|
37.276187845304
|
-14-15-eet-si
|
(±)14(15)-EET-sulfonimide; (±)14(15)-EpETrE-SI
|
arachidonic acid AA endothelium epoxytrienoic acid EETs EpETrEs cytochromes P450 acetylcholine bradykinin sulfonamide analog tyrosine phosphorylation mitogenesis renal epithelial cells hypertension EDHF |
| 10010635 |
(±)16-HETE
|
|
- |
≥98%
|
|
|
2008-06-09
|
18.474401473297
|
-16-hete
|
|
CYP450 eicosanoid metabolism kidneys ATPase ion transport vasodilation renal hypertension |
| 10004385 |
16(R)-HETE
|
|
183509-22-0 |
>98%
|
|
|
2008-07-28
|
1.724723756906
|
16-r-hete
|
|
CYP450 eicosanoid metabolism kidney ion transport vasodilation renal hypertension HETEs |
| 13076 |
16(R)-Iloprost
|
|
- |
≥98%
|
|
|
2008-10-10
|
24.321151012891
|
16-r-iloprost
|
|
prostacyclin platelet aggregation IP receptors EP vasodilation pulmonary hypertension stereoisomers inhibits inhibitors inhibition iloprosts PGI2 |
| 10004384 |
16(S)-HETE
|
|
183509-23-1 |
≥98%
|
|
|
2008-07-23
|
1.507182320442
|
16-s-hete
|
|
inhibitors inhibits inhibitions CYP450 eicosanoid metabolism kidneys ATPase ion transport renal hypertension HETEs 16SHETE 16S-HETE 16 S HETE |
| 13077 |
16(S)-Iloprost
|
|
74843-14-4 |
≥98%
|
|
|
2008-10-10
|
24.321151012891
|
16-s-iloprost
|
|
prostacyclin platelet aggregation IP receptors EP vasodilation pulmonary hypertension stereoisomers iloprosts inhibits inhibitors inhibition PGI2 |
| 10011305 |
17(S)-HETE
|
|
183509-25-3 |
>98%
|
|
|
2008-08-25
|
7.726440410418
|
17-s-hete
|
|
CYP450 Eicosanoid metabolism kidney ATPase ion transport renal hypertension |
| 10010638 |
(±)18-HETE
Exclusive |
|
- |
≥97%
|
|
✓ |
2008-06-13
|
2.100298342542
|
-18-hete
|
|
CYP450 eicosanoid metabolism kidney vasodilation CYP2E1 20-HETE 20HETE 18HETE renal hypertension |
| 10007767 |
19(R)-HETE
|
|
115461-39-7 |
>98%
|
|
|
2008-05-27
|
4.083977900552
|
19-r-hete
|
|
hypertension arterioles CYP450 kidneys angiotensin II vasodilator vasoconstricition 20-HETE 19HETE 19-HETE renal 19 HETE |
| 10007766 |
19(S)-HETE
Exclusive New |
|
115461-40-0 |
≥98%
|
|
✓ |
2010-04-06
|
2.041988950276
|
19-s-hete
|
|
cytochromes P450 CYP450 metabolites arachidonic acids kidneys angiotensin II CYP2E1 vasodilators renal preglomerular vessels ATPase hypertension arterioles vasoconstriction |
| 10007912 |
20-carboxy Arachidonic Acid
Exclusive |
|
79551-84-1 |
>98%
|
|
✓ |
2007-08-15
|
40.377605893186
|
20-carboxy-arachidonic-acid
|
20-COOH-AA
|
20-HETE metabolites PPAR.alpha. PPAR.gamma. vasorelaxation activators CYP4F3B hypertension cytochrome P450 CYP450 perioxisome proliferator activated receptor PPARs PPARalpha PPARgamma |
| 10008596 |
(±)5(6)-EET Ethanolamide
Exclusive |
|
- |
>95%
|
|
✓ |
2006-10-20
|
11.558705603788
|
-5-6-eet-ethanolamide
|
(±)5(6)-EpETrE Ethanolamide
|
epoxides epoxygenases 5,6-EETs cytochrome P450 (+/-)5(6)-EpETrEs (+/-)5,6-EpETrEs fatty acids esters ethanolamides metabolites AEA anandamides arachidonoyl neurotransmitters cannabinergic endocannabinoids CB1 CB2 receptors central peripheral FAAH hydrolases metabolism lipoxygenases inhibition (±)5(6)-Epoxy eicosatrienoyl 14,15-EET 14,15-EpETrE 14,15-EET-EA 14,15-EET-ethanolamide 14,15-epetre-ea 14,15-ethanolamide |
| 13260 |
6-keto Prostaglandin E1
|
|
67786-53-2 |
>99%
|
|
|
|
67.502872928176
|
6-keto-prostaglandin-e1
|
6-keto PGE1
|
6-keto-PGE1 metabolites prostaglandins |
| 10007210 |
6-keto Prostaglandin E1 Lipid Maps MS Standard
|
|
67786-53-2 |
>99%
|
|
|
2008-11-03
|
44.861528545119
|
6-keto-prostaglandin-e1-lipid-maps-ms-standard
|
6-keto PGE1
|
6-keto-PGE1 metabolites prostaglandins GC LC MS mass spectrometry standards GC/MS LC/MS GC-MS LC-MS |
| 10009998 |
(±)8,9-DHET-d11
Exclusive |
|
- |
≥99% deuterated product
|
|
✓ |
2008-03-17
|
9.351325966851
|
-8-9-dhet-d11
|
|
epoxides epoxygenases DHT hydrolases (+/-)14,15-DiHETrEs deuterated epoxide hydrolase deuterated deuterium |
| 18112 |
8,9-EE-14(Z)-E
Exclusive |
|
- |
≥95%
|
|
✓ |
2009-03-15
|
6.380018416206
|
8-9-ee-14-z-e
|
8,9-Epoxyeicosa-14(Z)-enoic Acid
|
14,15-EETs 14,15-EpETrEs vasodilation vascular disease hypertension EEZE |
| 10009532 |
(±)8(9)-EET-d11
Exclusive |
|
- |
≥99% deuterated product
|
|
✓ |
2008-03-25
|
9.058563535911
|
-8-9-eet-d11
|
(±)8(9)-EpETrE-d11
|
epoxides epoxygenases cytochrome P450 (±)8,9-EpETrEs (+/-)8,9-EpETrEs fatty acids (+/-)8(9)EpETrEs 8(9)EETs eicosatrienoic 8,9-EETs deuterated racemic mixture |
| 10008597 |
(±)8(9)-EET Ethanolamide
|
|
- |
>98%
|
|
|
2007-07-05
|
15.586008287292
|
-8-9-eet-ethanolamide
|
(±)8(9)-EpETrE Ethanolamide
|
AEA endocannabinoids arachidonoyl ethanolamide CYP450 cytochrome P450 metabolism ethanolamides hypertension |
| 589451 |
AcSDKP EIA Kit
|
|
- |
|
|
|
|
183.304475138121
|
acsdkp-eia-kit
|
N-Acetyl Ser-Asp-Lys-Pro EIA Kit; AcSDKP ELISA Kit
|
N-Acetyl-Seryl-Aspartyl-Lysyl-Proline serine aspartamine lysine measures kits eias enzyme immunoassays ELISAs growth regulatory hormones plasma urine spi-bio spibio A05881 atherosclerosis hypertension endocrinology assays |
| 10004377 |
Aldosterone EIA Kit - Monoclonal
|
|
- |
|
|
|
2004-04-21
|
331.428402394107
|
aldosterone-eia-kit-monoclonal
|
Aldosterone ELISA Kit - Monoclonal
|
582041 steroids hormones mineralocorticoids salt reabsorption electrolytes renin-angiotensin system RAS enzyme immunoassays eias elisas measures kits hypertension endocrinology assays |
| 13648 |
Alfuzosin (hydrochloride)
New |
|
81403-68-1 |
≥98%
|
|
|
2010-07-19
|
0E-12
|
alfuzosin-hydrochloride
|
Uroxatral; SL 77-499-10
|
α1-adrenergic receptors antagonists lower urinary tract symptoms benign prostatic hyperplasia BPH adrenoceptors α1A α1B α1D contractions smooth muscles antihypertensives vasodilators urinary flow 133880-44-1 Urion Alfoten SL 77499-10 anti-hypertensives alpha 1 .alpha.1 |
| 10010663 |
Amlodipine-d4 (besylate)
|
|
- |
≥99% deuterated product
|
|
|
2009-08-10
|
0E-12
|
amlodipine-d4-besylate
|
|
deuterateds deuteriums standards GC/MS LC/MS GC-MS LC-MS mass spectrometry dihydropyridine pyridines calcium channel blocker angina pectoris hypertension 88150-42-9 |
| 589301 |
Angiotensin II EIA Kit
|
|
- |
|
|
|
|
141.064143646408
|
angiotensin-ii-eia-kit
|
Angiotensin II ELISA Kit
|
hypertension angiotensin measures kits eias enzyme immunoassays ELISAs spi-bio spibio A05880 atherosclerosis endocrinology assays |
| 13523 |
Apelin-13
New |
|
217082-58-1 |
≥95%
|
|
|
2010-06-29
|
0E-12
|
apelin-13
|
|
ligands APJ receptors central nervous system cardiovascular functions fluid homeostasis neurosciences hypertension diabetes metabolic syndrome insulin HIV aids |
| 583951 |
Arginine Vasopressin EIA Kit
|
|
- |
|
|
|
2007-07-19
|
150.981843294826
|
arginine-vasopressin-eia-kit
|
Vasopressin EIA Kit; AVP ELISA Kit; Antidiuretic Hormone (ADH) EIA Kit; Argipressin EIA Kit
|
enzymes immunoassays measurements arg8 measures kits eias ELISAs AChE acetylcholinesterases plasmas serums argipressin antidiuretic hormones ADH amino acids peptides regulates regulation renal water excretion cardiovascular mammals epithelial cells urinary tracts urine blood stimulates stimulation constriction capillaries aterioles pressure depressions congestive hearts failures anxious-retarded argipressins APH antidiuretics endocrinology assays |
| 10009345 |
Arginine Vasopressin EIA Kit (Solid Plate)
|
|
- |
|
|
|
2007-07-19
|
117.903943699026
|
arginine-vasopressin-eia-kit-solid-plate
|
Vasopressin EIA Kit (Solid Plate); Argipressin EIA Kit (Solid Plate); Antidiuretic Hormone (ADH) EIA Kit (Solid Plate); AVP ELISA Kit (Solid Plate)
|
AVP eias enzymes immunoassays kits measures measurements ELISAs |
| 589401 |
Atriopeptin (rat) EIA Kit
|
|
- |
|
|
|
|
24.620883977900
|
atriopeptin-rat-eia-kit
|
Atriopeptin (rat) ELISA Kit
|
naturiuretic auriculin measures kits eias enzyme immunoassays ELISAs atherosclerosis pi-bio spibio A05103 hypertension endocrinology assays |
| 10007927 |
AUDA
Exclusive |
|
479413-70-2 |
>98%
|
|
✓ |
2006-04-28
|
47.803832872928
|
auda
|
|
epoxides hydrolases hypertension dihydroxy-eicosatrienoic acids DHETs 11(12)-EETs 14(15)-EETs blood pressure soluble sEH inhibits inhibitors inhibition peroxisome proliferator-activated receptors PPARalpha PPAR.alpha. DiHETrEs EpETrEs endocrinology |
| 10005186 |
CAY10441
Exclusive |
|
221529-58-4 |
>98%
|
|
✓ |
2004-09-16
|
112.584337016574
|
cay10441
|
RO1138452
|
receptors antagonists IPs prostaglandins carbaprostacyclins inhibits inhibitors inhibition analgesics high-affinity ligands neuroblastoma cyclic AMP cAMP adenylate cyclase 4,5-dihydro-1H-imidazol-2-yl-4-4-isopropoxy benzyl phenylamine atherosclerosis |
| 10005913 |
CAY10449
Exclusive |
|
- |
>98%
|
|
✓ |
2004-10-26
|
202.691795580110
|
cay10449
|
|
receptors antagonists IPs prostaglandins carbaprostacyclins inhibits inhibitors inhibition analgesics high-affinity ligands neuroblastoma adenylate cyclase cyclic AMP cAMP iloprost athersclerosis CAY 10449 |
| 10012447 |
CG 4305
New |
|
- |
≥95%
|
|
|
2010-05-12
|
0E-12
|
cg-4305
|
|
antithrombotic PGI2 epoprostenol prostacyclins platelets aggregation 89955-40-8 PGs prostaglandins I2 cartoid artery thrombosis inhibits inhibited inhibition inhibitory |
| 30001 |
cGMP Alprostadil
New GMP API |
|
745-65-3 |
|
|
|
2010-08-17
|
0E-12
|
cgmp-alprostadil
|
Prostaglandin E1
|
|
| 30024 |
cGMP Alprostadil-Alfadex
New GMP API |
|
93591-00-5 |
|
|
|
2010-08-17
|
0E-12
|
cgmp-alprostadil-alfadex
|
Prostaglandin E1 with α-cyclodextrin
|
|
| 30010 |
cGMP Epoprostenol (sodium salt)
New GMP API |
|
61849-14-7 |
|
|
|
2010-08-17
|
0E-12
|
cgmp-epoprostenol-sodium-salt
|
Prostaglandin I2 (sodium salt); Prostacyclin (sodium salt)
|
|
| 589101 |
CGRP (human) EIA Kit
|
|
- |
|
|
|
|
171.001381215470
|
cgrp-human-eia-kit
|
Calcitonin Gene-related Peptide (human) EIA Kit; CGRP (human) ELISA Kit
|
calcitonin peptides measures kits eias enzyme immunoassays ELISAs spi-bio neurochemistry neuroscience spibio A05481 endocrinology assays |
| 10007923 |
CUDA
Exclusive |
|
479413-68-8 |
>98%
|
|
✓ |
2006-04-28
|
42.116700868192
|
cuda
|
|
epoxides hydrolases hypertension dihydroxy eicosatrienoic acids DiHETrEs DHETs 11(12)-EETs 14(15)-EETs EpETrEs blood pressure soluble sEH inhibits inhibitors inhibition peroxisome proliferator-activated receptors PPARalpha PPAR.alpha. activates activation endocrinology |
| 10018 |
DDMS
|
|
206052-03-1 |
>98%
|
|
|
2005-02-22
|
5.549723756906
|
ddms
|
Dibromo-dodecenyl-methylsulfimide
|
20-HETEs inhibits inhibitors inhibition synthesis CYP450-4A2 renal hypotension vascular homeostasis circulation kidneys vasodilation vasodilators NONOates CYP4A2 donors cytochrome |
| 10010588 |
Desmethylsildenafil-d8 Citrate
|
|
- |
>98% deuterated product
|
|
|
2008-04-14
|
0E-12
|
desmethylsildenafil-d8-citrate
|
|
drugs PAH pulmonary arterial hypertension erectile dysfunction impotence |
| 10006865 |
Docosahexaenoic Acid methyl ester
|
|
2566-90-7 |
>98%
|
|
|
2005-09-06
|
33.374751381215
|
docosahexaenoic-acid-methyl-ester
|
Cervonic Acid methyl ester; DHA methyl ester
|
polyunsaturated fatty acids PUFAs omega-3 brain .omega.-3 w-3 esters diets dietary supplements hypertension neonatal photoreceptor degeneration retinitis pigmentosa depiration neural tissues retina |
| 10008610 |
Epoxy Fluor 7
|
|
863223-43-2 |
>98%
|
|
|
2006-08-30
|
21.267289364641
|
epoxy-fluor-7
|
|
epoxides hydrolases fluorescence enzymes activity inhibition screening hypertension inflammation sepsis EETs DHETs EpETrEs DiHETrEs fluorescent SEH soluble endocrinology |
| 10010559 |
HA-1077 (hydrochloride)
|
|
203911-27-7 |
≥98%
|
|
|
2008-09-03
|
30.874281767956
|
ha-1077-hydrochloride
|
Eril; Fasudil (hydrochloride)
|
protein kinase inhibitors inhibits inhibition ROCK-II ROCKII PRK2 MSK1 MAPKAP-K1b vasodilation hypertension diabetes renal nephropathy cancers |
| 10011038 |
Hemopressin
|
|
- |
|
|
|
2009-08-13
|
58.529090909091
|
hemopressin
|
|
peptides antagonist inhibitors inhibits inhibition hypertension binding asoactive vasoactive |
| 10005518 |
IP Receptor (human) Polyclonal Antibody
|
|
- |
|
|
|
2004-10-21
|
21.225132305903
|
ip-receptor-human-polyclonal-antibody
|
Prostaglandin I2 Receptor; Prostacyclin Receptor; PGI2 Receptor
|
antibodies antisera antiserum western blots blotting wb prostacyclins rat PGI2 prostaglandins receptors immunoblotting atherosclerosis |
| 10010572 |
Lercanidipine-d3 (hydrochloride)
|
|
- |
>99% deuterated product
|
|
|
2008-04-14
|
0E-12
|
lercanidipine-d3-hydrochloride
|
|
SPI blocker calcium dihydropyrine neurochemistry |
| 16833 |
Lisinopril
|
|
76547-98-3 |
≥98%
|
|
|
2009-03-09
|
2.077348066299
|
lisinopril
|
MK 522; MK 521
|
inhibitors inhibits inhibition angiotensin I II ACE endothelin 1 nitric oxide renin hypertension diabetes |
| 10010971 |
Luminex® 11-dehydro Thromboxane B2 Kit
|
|
- |
|
|
|
2008-01-24
|
52.225662983425
|
luminex-11-dehydro-thromboxane-b2-kit
|
Luminex® 11-dehydro TXB2 Kit
|
thromboxanes thromboxane A2 TXA2 metabolites urine in vivo measures kits luminex xMAP beads assays |
| 10009835 |
MK 0524
|
|
571170-77-9 |
>98%
|
|
|
2008-05-06
|
62.451239147592
|
mk-0524
|
Laropiprant
|
antagonist PGD2 allergy asthma DP1 niacin vasodilations flushing dyslipidemia receptors atherosclerosis hypertension inflammation mk0524 |
| 10010412 |
MRE-269
Exclusive |
|
475085-57-5 |
≥98%
|
|
✓ |
2008-11-06
|
64.450011049724
|
mre-269
|
|
MRE269 prostaglandins PGI2 IP receptors inflammation NS-304 NS304 agonists vasodilator hypotensive vascular diseases atherosclerosis hypertension analogs potent selective PGs prodrugs |
| 10010653 |
Nisoldipine-d3
|
|
- |
≥99% deuterated product
|
|
|
2009-04-15
|
0E-12
|
nisoldipine-d3
|
|
63675-72-9 86189-67-5 calcium channel dihydropyridine cardiac failure angina deuterateds deuteriums standards GC/MS LC/MS GC-MS LC-MS mass spectrometry |
| 10010411 |
NS-304
|
|
475086-01-2 |
>98%
|
|
|
2008-04-09
|
56.267127071823
|
ns-304
|
ACT-293987; Selexipag
|
prostaglandins PGI2 IP receptors inflammation MRE-269 agonists vasodilator hypotensive vascular diseases atherosclerosis hypertension analogs potent selective PGs |
| 10006803 |
O-1602
|
|
317321-41-8 |
>98%
|
|
|
2005-09-12
|
17.105911602209
|
o-1602
|
|
abnormal cannabidiols CB1 CB2 receptors vasorelaxation neurochemistry neuroscience central cannabinoids peripheral selective antagonists nonendothelium-dependant vasodilation nitric oxides NOs inhibits inhibitors inhibition vasorelaxant |
| 10006804 |
O-1821
|
|
35482-50-9 |
>97%
|
|
|
2005-09-12
|
0.884493554327
|
o-1821
|
|
abnormal cannabidiol central cannabinoids peripheral CB1 CB2 receptors vasorelaxation neurochemistry neuroscience antagonists synthetic regioisomer endothelium dependent vasodilation |
| 10004914 |
O-1918
|
|
536697-79-7 |
>98%
|
|
|
2005-09-09
|
3.982550644567
|
o-1918
|
|
antagonists abnormal cannabinoids cannabidiols cannabidiol-mediated synthetic regioisomers CB1 CB2 responsiveness psychotropics activity induces endothelium-dependent vasodilations NO-independent nitric oxides mechanisms analogs endothelial receptors inhibits inhibition inhibitors vasorelexants in vitro blocks induced activations PI3-kinases Akt pathway umbilical vein cells neuroscience neurochemistry O1918 0-1918 |
| 600240 |
Orexin 1 Receptor STEP Reporter Assay Kit (Luminescence)
New |
|
- |
|
|
|
2010-03-31
|
0E-12
|
orexin-1-receptor-step-reporter-assay-kit-luminescence
|
OX1R
|
hypercretins 1 orexins 2 A orexin-2 systems regulates regulator sleep wake cycles feeding cardiovascular autonomic hypothalamic neuropeptides Orexins A Orexins B gut hormones secretions hypothalamus midbrains brainstems G protein-coupled receptors GPCRs orexin-1 OX1R orexin-2 OX2R orexin-A orexin-B sleep disorders narcolepsy humans animals rodents energy homeostasis pain stress antagonists drugs addictions withdrawals therapeutics obesity Surface transfection expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated luminescent secretory alkaline phosphatases SEAP signal transduction cascades culture medium luminescence-based high throughput screening screens agonists |
| 600250 |
Orexin 2 Receptor STEP Reporter Assay Kit (Luminescence)
New |
|
- |
|
|
|
2010-03-31
|
0E-12
|
orexin-2-receptor-step-reporter-assay-kit-luminescence
|
OX2R
|
hypercretins 1 orexin 2 systems regulates regulator sleep wake cycles feeding cardiovascular autonomic hypothalamic neuropeptides Orexins A Orexins B gut hormones secretions hypothalamus midbrains brainstems G protein-coupled receptors GPCRs orexin-1 OX1R orexin-2 OX2R orexin-A orexin-B sleep disorders narcolepsy humans animals rodents energy homeostasis pain stress antagonists drugs addictions withdrawals therapeutics obesity Surface transfection and expression protocols solid phase transient transfection technology originus patents USPT US6897067 US6902933 US7056741 US 6897067 6902933 7056741 DNA deoxyribonucleases adherent cells receptor-mediated luminescent secretory alkaline phosphatases SEAP signal transduction cascades culture medium luminescence-based high throughput screening screens agonists |
| 70515 |
Ozagrel
|
|
82571-53-7 |
>98%
|
|
|
|
3.896095764272
|
ozagrel
|
OKY-046
|
thromboxanes synthases inhibitors inhibits imidizoles TXAs antihypertensive inhibition atherosclerosis |
| 10007852 |
Pargyline (hydrochloride)
|
|
306-07-0 |
>98%
|
|
|
2006-08-30
|
48.184551104972
|
pargyline-hydrochloride
|
|
MAO inhibitors inhibits inhibition ROS-mediated Hypertension 3 blood pressures systolic brains monocytes hypertrophy reactive oxygen species endocrinology |
| 10009567 |
PCSK9 Western Ready Control
|
|
- |
|
|
|
2007-01-31
|
10.271860036832
|
pcsk9-western-ready-control
|
Proprotein Convertase Subtilisin Kexin 9; NARC-1
|
PSEC0052 subtilisin serine proteases LDLs low density lipoproteins cholesterol receptors golgi atherosclerosis |
| 10009134 |
PHOME
Exclusive |
|
- |
>98%
|
|
✓ |
2007-01-16
|
43.239459791283
|
phome
|
|
sEH epoxides hydrolase inhibitors inhibition inhibits substrates HTS fluorogenic high throughput screening fluorescent fluorescence hypertension endocrinology |
| 10011724 |
Propenyl-L-NIO (hydrochloride)
Exclusive |
|
- |
>90%
|
|
✓ |
2008-08-19
|
9.454972375691
|
propenyl-l-nio-hydrochloride
|
ENIPO
|
nitric oxide synthase NOS iNOS selective inhibitors inhibits inhibition |
| 10007599 |
Prorenin (human recombinant)
|
|
- |
>99% by SDS-PAGE
|
|
|
2005-10-19
|
83.509309392265
|
prorenin-human-recombinant
|
|
enzymes aspartyl proteases angiotensins II glycoproteins angiotensinogen salt balance hypertension angiotensinogens kidney renal preprorenin endocrinology |
| 10010 |
Prostaglandin A1
|
|
14152-28-4 |
>98%
|
|
|
|
111.669352801894
|
prostaglandin-a1
|
PGA1
|
prostaglandins renal vasodilation pge1 dehydration semen antimitotic antiproliferative |
| 10020 |
Prostaglandin A1 ethyl ester
|
|
93464-24-5 |
>98%
|
|
|
|
101.926077348067
|
prostaglandin-a1-ethyl-ester
|
PGA1 ethyl ester
|
PGA1 renal vasodilation prostaglandins esters prodrugs lipid-soluble |
| 12990 |
Prostaglandin D3
|
|
71902-47-1 |
>98%
|
|
|
|
97.405607734806
|
prostaglandin-d3
|
PGD3
|
PGD3 omega-3 w-3 .omega.-3 metabolites EPA eicoaspentaenoic acid prostaglandins |
| 13010 |
Prostaglandin E1
|
|
745-65-3 |
>98%
|
|
|
|
69.748572259377
|
prostaglandin-e1
|
Alprostadil; PGE1
|
PGE1 vasodilation atherosclerosis erectile dysfunction prostaglandins pharma:1 |
| 13010.1 |
Prostaglandin E1 Analytical Reference Standard
|
|
745-65-3 |
>99%
|
|
|
|
27.062348066298
|
prostaglandin-e1-analytical-reference-standard
|
Alprostadil; PGE1
|
PGE1 vasodilation USP erectile dysfunction prostaglandins |
| 10006906 |
Renin Fluorogenic Substrate
|
|
- |
>95%
|
|
|
2006-12-12
|
108.399092344120
|
renin-fluorogenic-substrate
|
|
substrates aspartyl proteases angiotensinogens peptides peptide-EDANS non-fluorescent quenching molecules Dabcyl fluorescent excitation emission hypertension endocrinology |
| 10006217 |
Renin (human recombinant)
|
|
- |
>99% by SDS-PAGE
|
|
|
2004-12-13
|
75.871298342541
|
renin-human-recombinant
|
|
enzymes aspartyl proteases angiotensins II glycoproteins angiotensinogen salt balance hypertension angiotensinogens kidney renal preprorenin atherosclerosis endocrinology |
| 10006270 |
Renin Inhibitor Screening Assay Kit
|
|
- |
|
|
|
2005-05-04
|
64.085943172849
|
renin-inhibitor-screening-assay-kit
|
|
Protease measurement assays aspartyl renal juxtaglomerular cells sodium depletion blood volume pressure .beta.-adrenergic stimulation angiotensinogens angiotensins I II converting ACE monomeric zinc metalloenzymes vascular endothelium messengers RAS vasoconstrictor peripheral hypertension receptors blockers fluorescence fluorescent fluorometric atherosclerosis endocrinology |
| 13082 |
Resorcinolnaphthalein
|
|
41307-63-5 |
≥98%
|
|
|
2009-02-24
|
66.719907918969
|
resorcinolnaphthalein
|
NSC 354317
|
angiotensin converting enzyme 2 ACE2 hypertension blood pressure activators fibrosis |
| 10010662 |
Rilmenidine-d4
|
|
85047-14-9 |
≥99% deuterated product
|
|
|
2009-04-17
|
0E-12
|
rilmenidine-d4
|
|
adrenergic agonist agents antihypertensive deuterateds deuteriums standards GC/MS LC/MS GC-MS LC-MS mass spectrometry |
| 10010586 |
Sildenafil-d8 Citrate
|
|
- |
>98% deuterated product
|
|
|
2008-04-14
|
11.933701657459
|
sildenafil-d8-citrate
|
|
SPI PAH drugs males pulmonary inpotance ER erectile dysfunction arterial hypertension |
| 10008609 |
S-NEPC
Exclusive |
|
- |
>98%
|
|
✓ |
2007-05-01
|
23.396330570901
|
s-nepc
|
|
Cytochrome P450 CYP450 subtrates glutathione s-transferase hydrolases procine liver carboxylesterase hydrolysis spectrophotometry (+)-NEPC (-)-NEPC hypertension sEH epoxides sEH inhibitor substrate GST endocrinology |
| 600090 |
Soluble Epoxide Hydrolase Cell-Based Assay Kit
|
|
- |
|
|
|
2009-05-14
|
58.766314127860
|
soluble-epoxide-hydrolase-cell-based-assay-kit
|
sEH Cell-Based Assay Kit
|
kits assays measuring measurement mammalian epoxides α/β-hydrolases enzymes catalyzes hydrolysis exogenous endogenous vicinal diols homodimers C-terminal N-terminal domains vasodilatory vasodilation anti-inflammatory hypertension vascular inflammation inhibitors therapeutics fluorescence-based fluorescent whole cells Epoxy Fluor 7 6-methoxy-2-naphthaldehyde AUDA |
| 10011669 |
Soluble Epoxide Hydrolase (human recombinant)
|
|
- |
≥95%
|
|
|
2008-07-02
|
312.558116022099
|
soluble-epoxide-hydrolase-human-recombinant
|
CEH; Cytosolic Epoxide Hydrolase; sEH; Epoxide Hydrolase 2; EPHX2
|
recombinant proteins mammalian hydrolases enzymes exogenous endogenous his-tags hexahistindes His-tagged anti-inflammatory inflammation sehs hydrolases hydrolysis |
| 10011671 |
Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit
|
|
- |
|
|
|
2009-02-24
|
73.638447513812
|
soluble-epoxide-hydrolase-inhibitor-screening-assay-kit
|
sEH Inhibitor Screening Assay Kit
|
epoxides hydrolases sEHs inhibits inhibition assays kits fluorescence-based catalyzes hydrolysis exogenous endogenous vicinal diols substrates EETs epoxyeicosatrienoic acids vasodilatory vasodilation anti-inflammatory molecules therapy therapeutics hypertension vascular diseases PHOME (3-phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester 6-methoxy-2-naphthaldehyde excitation emission wavelengths a/b-hydrolases alpha/beta-hydrolases .alpha./.beta.-hydrolases enzymes homodimers C-terminal C-terminus animals models cyanohydrins cyanide ions |
| 10011670 |
Soluble Epoxide Hydrolase (murine recombinant from Sf21 cells)
Exclusive |
|
- |
≥95%
|
|
✓ |
2008-07-01
|
44.923475138121
|
soluble-epoxide-hydrolase-murine-recombinant-from-sf21-cells
|
sEH; Epoxide Hydrolase 2; EPHX2; Cytosolic Epoxide Hydrolase; CEH
|
recombinant proteins mammalian hydrolases enzymes exogenous endogenous hexahistidine His-tag His-tagged N-terminal anti-inflammatory inflammation 10278 |
| 10010146 |
Soluble Epoxide Hydrolase Polyclonal Antibody
|
|
- |
|
|
|
2008-03-03
|
15.367648480662
|
soluble-epoxide-hydrolase-polyclonal-antibody
|
Epoxide Hydrolase 2; EPHX2; sEH; Cytosolic Epoxide Hydrolase (CEH)
|
metabolism hypertension inflammation EpETrEs EETs DiHETrEs DHET inhibitors inhibit inhibitions epoxyeicosatrienoic acids eicosatrienoic WB western blots blotting immunoblotting |
| 10162 |
Treprostinil
|
|
81846-19-7 |
>98%
|
|
|
2005-08-30
|
107.833449969306
|
treprostinil
|
|
primary pulmonary hypertension PPH arterial vascular resistance stable analogs prostacyclins increase plasma half-life vasodilatory inhibits inflammatory cytokines inhibition inhibitors GM-CF human alveolar macrophages NF-KB NF-.kappa. translocations nucleus NF-kappaB nfkb nf-kb NF-.kappa.B atherosclerosis |
| 700320 |
Uric Acid Assay Kit
New |
|
- |
|
|
|
2010-08-30
|
0E-12
|
uric-acid-assay-kit
|
Urate Assay Kit
|
kits assays measures measurement acids human purines metabolisms urine serum renal excretion excreted allantoin enzymes urate oxidases uricase genes obesity alcohol consumption hyperuricemia gout kidney stones metabolic syndromes hypertension cardiovascular diseases exercise-induced acute failure hypouricemia |