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Application · Inhibitor Screening Assay

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Item Number Product Sizes & Pricing CAS Purity Image Exclusive Introduction Date Mojo Plain Text Name Synonyms Keywords Interest
700580 Autotaxin Inhibitor Screening Assay Kit - 2011-06-28 16.120036832412 autotaxin-inhibitor-screening-assay-kit ATX Inhibitor Screening Assay Kit kits assays measures measurements Ectonucleotides Pyrophosphatase-2 ENPP-2 Lysopholipases D hydrolysis lysophosphatidylcholines LPC lysophosphatidic acid LPA lipids mediators G protein-coupled receptors GPCRs neurogenesis angiogenesis smooth-muscles contraction platelets aggregations wounds healings ATX-LPA signaling tumors progression inflammation serums proteolytically peptides proteins N-glycosylation Asn53 Asn410 adipocytes cerebrospinal fluid multiple sclerosis livers fibrosis cancers genes chips analysis upregulated metastatic inhibits inhibition human 16.120036832412
600070 BACE Inhibitor Screening Assay Kit - 2009-03-26 16.731740331491 bace-inhibitor-screening-assay-kit β-Secretase Inhibitor Screening Assay Kit inhibitors inhibition inhibits assays kits β-sites .beta.-sites b-sites APP cleaving enzymes β-amyloids .beta.-amyloids b-amyloids peptides Ab A.beta. brain neurodegeneration Alzheimer's Diseases AD proteolytic cleavages precursors β-secretases b-secretases γ-secretases .gamma.-secretases g-secretases membranes aspartic C-terminal C-terminus fragments proteolysis therapeutics therapy cascade pathogenesis mice mouse murine transgenics cholinergic dysfunctions HIV humans fluorescents fluorescences fluorometer assays 16.731740331491
760111 Colorimetric COX (ovine) Inhibitor Screening Assay Kit - 185.450171561500 colorimetric-cox-ovine-inhibitor-screening-assay-kit cyclooxygenases cox-1 cox-2 pghs-1 pghs-2 cox1 cox2 pghs1 pghs2 prostaglandins synthases synthase-1 synthase-2 inhibition inhibitors assays screens peroxidase colorimetrically analysistools:eia 185.450171561500
560131 COX Inhibitor Screening Assay Kit - 239.017309632476 cox-inhibitor-screening-assay-kit enzyme immunoassays kits measures EIAs ELISAs COX1 COX-1 COX2 COX-2 PGHS1 pghs-1 pghs2 pghs-2 prostaglandin synthases inhibitors cyclooxygenase analysistools:eia assays cox inhibitior kit 239.017309632476
560101 COX (ovine) Inhibitor Screening Assay Kit - 131.589773743751 cox-ovine-inhibitor-screening-assay-kit enzyme immunoassays kits measures EIAs ELISAs COX1 COX-1 COX2 COX-2 PGHS1 pghs-1 pghs2 pghs-2 prostaglandin synthases inhibitors cyclooxygenases sheep screens assays cox inhibitior kit 131.589773743751
700210 DPP (IV) Inhibitor Screening Assay Kit - 2009-05-27 105.254259921503 dpp-iv-inhibitor-screening-assay-kit Dipeptidyl exopeptidases IV DPPIV DPP4 enzymes CD26 cluster of differentiation T-cells activation antigens adenosine deaminase complexing 2 membrane-bound glycoproteins immune regulation signal transduction apoptosis kidneys small intestines placentas humans serums seminal fluids proteolytic derivatives serines X-prolines X-alanines dipeptides N-terminus N-terminal polypeptides growth factors chemokines neuropeptides vasoactive inhibitors inhibits inhibition oral antidiabetic agents glucose homeostasis glucoregulatory hormones glucose-dependent insulinotropics GIP glucagon-like peptide-1 GLP-1 gastric therapeutics Type 2 tumors cancers markers neoplasms assays kits measures measurements fluorescences fluorescent fluorogenics substrates Gly-Pro-Aminomethylcoumarin AMC 105.254259921503
10005196 FAAH Inhibitor Screening Assay Kit - 2008-09-05 96.643796369377 faah-inhibitor-screening-assay-kit Fatty Acid Amide Hydrolase Inhibitor Screening Assay Kit neurochemistry neuroscience endocannabinoids lipid signaling regulatory arachidonoylethanolamides AEAs 2-arachidonoyl glycerol 2-AG G Protein Coupling Receptors GPCRs CB1 motor controls cognition emotional responses homeostasis CB2 peripheral tissues modulators autonomic nervous systems immune microcirculation enzymes fatty acids amides hydrolases monoacylglycerols lipases MGL MAGL serines inhibitors pain obesity neurological diseases agonists fluorescence-based screening hydrolyzes AMC-arachidonoyl 7-amino-4-methylcoumarin fluorophores assays kits 96.643796369377
10010231 FABP4 Inhibitor/Ligand Screening Assay Kit - 2007-11-01 14.448967275818 fabp4-inhibitor-ligand-screening-assay-kit aP2; Adipocyte FABP; A-FABP; Fatty Acid Binding Protein 4 fabps kits atherosclerosis assays fatty acid binding protein adipocytes aP2 cytosolic lipophilic ligands uptake metabolisms cellular membranes intracellular trafficking cells growth differentiation PPARg PPARgamma PPAR.gamma. peroxisomes proliferator-activated receptors agonists insulin genes deletion mice mouse murine chronic metabolic diseases diabetes atherosclerosis fluorescence fluorescent fluorometric endocrinology 14.448967275818
700500 G9a Methyltransferase Inhibitor Screening Assay Kit - 2011-03-10 42.864293560789 g9a-methyltransferase-inhibitor-screening-assay-kit EHMT2 Methyltransferase Inhibitor Screening Assay Kit kits assays measures measurements methylations molecules proteins signals transductions biosynthesis proteins repair genes silencing chromatin regulation S-adenosylmethionine SAM methyltransferases enzymes enzymatic cofactors ATP adenosine triphosphates AdoMet donors methyls groups DNA deoxyribonucleic acids Alzheimer's diseases depression Parkinson's multiple sclerosis livers failures cancers methylations lysines transcriptional activation respression histones functions SET domain-containing mammalian monomethylates dimethylates 9 27 H3 embryogenesis genomic imprinting lymphocytes lung cells HIV-1 H3K9 viral latency GLP G9a-like EHMT1 tumors suppressors p53 373 feedback inhibition methylation reactions 42.864293560789
10011564 HDAC1 Inhibitor Screening Assay Kit - 2008-04-10 31.288852528686 hdac1-inhibitor-screening-assay-kit HDAC 1 histones deacetylases lysines residues chromatin condensation transcriptional repression fluorescence deacetylation fluorescent inhibits inhibition enzymes license:cyclex fluorometric assays cancer 31.288852528686
700230 HDAC8 Inhibitor Screening Assay Kit - 2009-05-15 21.721975138121 hdac8-inhibitor-screening-assay-kit Histone Deacetylase 8 Inhibitor Screening Assay Kit histone deacetylases inhibits inhibitors inhibition angiogenesis cycling apoptosis differentiation tumors proliferation anticancers genes epigenetic trichostatin A human class I tissues nucleus cytosolic smooth muscle neuroblastoma pathogenesis kits assays measures measurement fluorescent fluorescence-based 21.721975138121
600150 HDAC Cell-Based Activity Assay Kit - 2009-11-09 26.370505361597 hdac-cell-based-activity-assay-kit Histone Deacetylase Cell-Based Activity Assay Kit assays kits measuring measurement histones deacetylases lysines residues chromatin condensation transcriptional repression fluorescence deacetylation fluorescent inhibits inhibition enzymes fluorometric assays cancer modulators whole cells proteins lysine-specific HDAC1 homogenous inhibitor/activator TSA 26.370505361597
700360 JMJD2A Inhibitor Screening Assay Kit - 2010-05-25 19.047282813814 jmjd2a-inhibitor-screening-assay-kit Jumonji Domain Containing 2A Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC JHDM1 JHDM2 JHDM3 JARID1 UTX/UTY cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated 19.047282813814
700370 JMJD2D Inhibitor Screening Assay Kit - 2010-05-25 19.603553147282 jmjd2d-inhibitor-screening-assay-kit Jumonji Domain Containing 2D Inhibitor Screening Assay Kit kits assays measures measurements histones nucleoproteins chromatins DNA deoxynucleic acids eukaryotic nucleus nucleosomal H3 H4 H2B H2A octamers amino termini acetylation phosphorylation ubiquitination methylation FLJ10251 replication repair transcriptional activation repression dysregulation tumors suppressor genes cancers inhibitors enzymes catalyzes epigenetic marks methyls lysines arginines residues demethylases 1 JMJC cupin 2-oxoglutarate 2OG iron Fe(II) oxygenases hydroxylation JMJD2A JMJD2B JMJD2C JMJD2D JMJD2E JMJD2F fluorescence-based fluorescent cells lysates formaldehydes peptides substrates oxidation/decarboxylation acetoacetanilides ammonia H3K9(Me)3 trimethylated 19.603553147282
760700 Lipoxygenase Inhibitor Screening Assay Kit - 59.859187056037 lipoxygenase-inhibitor-screening-assay-kit LO Inhibitor Screening Assay Kit 12-LOs 15-LOs 15-lipoxygenases activity hydroperoxides assays kits inhibitors 12-lipoxygenases analysistools:lis 59.859187056037
700120 LSD1 Inhibitor Screening Assay Kit - 2008-10-16 24.063191420214 lsd1-inhibitor-screening-assay-kit Lysine-Specific Demethylase 1 lysines 4 demethylases histones residues repression transcription chromosomal DNA chromosomes inhibits inhibitors inhibition tumors suppressors activity cells cycles progression cancers fluorescent fluorescence enzymes enzymatic reactions H2O2 hydrogens peroxides peptides N-terminal tails H3 horseradish peroxidases ADHP resorufins assays 24.063191420214
705192 Monoacylglycerol Lipase Inhibitor Screening Assay Kit - 2009-10-22 102.257324388319 monoacylglycerol-lipase-inhibitor-screening-assay-kit MAGL; MGL neuroscience neurochemistry inhibitors inhibiting inhibition inhibits endocannabinoids serines hydrolases pain obesity monoglycerol 102.257324388319
700170 Myeloperoxidase Inhibitor Screening Assay Kit - 2009-04-14 99.838640883977 myeloperoxidase-inhibitor-screening-assay-kit MPO Inhibitor Screening Assay Kit heme peroxidases azurephilic granules leukocytes neutrophils monocytes tissues macrophages chlorides hydrogen peroxides H2O2 Cl- hypochlorous acids acute chronic vascular inflammatory diseases cardiac therapeutics cycles fluorescence fluorescent assays kits measures measurement crude cells lysates purified enzymes ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin 2-[6-(4-aminophenoxy)-3-oxo-3H-xanthen-9-yl]-benzoic acid APF -OCl assays 99.838640883977
700560 PAD4 Inhibitor Screening Assay Kit - 2011-05-04 49.092011970534 pad4-inhibitor-screening-assay-kit Protein Arginine Deiminase 4; Peptidylarginine Deiminase 4 kits assays measures measurements proteins arginines deiminases PADs guanidine-modifying enzymes peptidylarginine deiminase amidinotransferases nucleus homodimers transcriptional coregulator catalyzes residues citrulline calcium-dependent substrates histones H2A H3 H4 post-translational modifications genes regulations autocitrullination inhibits enzymatic activity cells rheumatoid arthritis citrulline-containing immune response autoantibodies tissues multiple sclerosis Alzheimer's diseases glaucoma cancers human deiminates N-α-benzoyl-L-arginine ethyl esters BAEE kinetic ammonia detectors fluorescent fluorescence 49.092011970534
10004380 PAF Acetylhydrolase Inhibitor Screening Assay Kit - 2004-03-29 47.752897483117 paf-acetylhydrolase-inhibitor-screening-assay-kit PAF-AH Inhibitor Screening Assay Kit; Lp-PLA2 Inhibitor Screening Assay Kit platelet-activating factors hypotension inflammations allergys PAFAH atherosclerosis heart diseases measures kits inhibitors PAFs assays paf elisa kit 47.752897483117
10007685 PPARγ Ligand Screening Assay Kit - 2009-07-16 45.958161727774 ppar-ligand-screening-assay-kit Peroxisome Proliferator-activated Receptor γ FP-Based Ligand Screening Assay Kit - Green FP-based peroxisomes proliferator-activated receptors PPARs proliferator activated PPARgamma PPAR.gamma. PPARg PPARγ PPAR-γ PPAR-gamma gamma g γ .gamma. PPAR-.gamma. PPAR-g kits assys atherosclerosis TF diabetes drugs discovery discover endocrinology high throughput screens screening inflammations inhibitors inhibits inhibition metabolic syndromes metabolism nuclear receptors fluorescence FP-based FP based base ligands probes proteins isoforms γ1 γ2 γ-1 γ-2 1 2 adipose tissues colon immune systems retinas adipogenesis cells cellular differentiation insulin sensitization cancers fatty acids FAAH arachdionic 15-deoxy-DELTA12,14-prostaglandin 15-deoxy-DELTA12,14-PGs 15-deoxy-DELTA12,14-PGJ2 15 deoxy DELTA 12,14 PGs prostaglandins PGJ2 15-deoxy-Δ12,14-PGs 15-deoxy-Δ12,14-prostaglandins 15-deoxy-Δ12,14-PGJ2 15-deoxy-D12,14-prostaglandins 15-deoxy-D12,14-PGs 15-deoxy-D12,14-PGJ2 15-deoxy-.DELTA.12,14-prostaglandins 15-deoxy-.DELTA.12,14-PGs 15-deoxy-.DELTA.12,14-PGJ2 J2 thiazolidinediones TZD pioglitazone rosiglitazone agonists hyperglycemia hyperinsulinemia hypertriglyceridemia types 2 antidiabetics diabetes oral antagonists 45.958161727774
10006595 Prostaglandin D Synthase Inhibitor Screening Assay Kit - 2005-08-31 33.210460405156 prostaglandin-d-synthase-inhibitor-screening-assay-kit PGDS Inhibitor Screening Assay Kit prostaglandins synthases inhibitors PGDS assays hematopoietic-types lipocalin-types pro-inflammatory mediators allergic allergy allergies allergens activity inhibitors inhibition inhibits H-PGDS L-PGDS 33.210460405156
10006270 Renin Inhibitor Screening Assay Kit - 2005-05-04 55.100208717004 renin-inhibitor-screening-assay-kit Protease measurement assays aspartyl renal juxtaglomerular cells sodium depletion blood volume pressure .beta.-adrenergic stimulation angiotensinogens angiotensins I II converting ACE monomeric zinc metalloenzymes vascular endothelium messengers RAS vasoconstrictor peripheral hypertension receptors blockers fluorescence fluorescent fluorometric atherosclerosis endocrinology 55.100208717004
700270 SET7/9 Methyltransferase Inhibitor Screening Assay Kit - 2009-12-04 24.872556970425 set7-9-methyltransferase-inhibitor-screening-assay-kit methyltransferases SET Domain-containing Protein 7/9 lysines 7 KMT7 methylation signal transduction biosynthesis proteins repair genes silencing chromatins S-adenosylmethionine SAM AdoMet methyl donors Alzheimer's depression Parkinson's Diseases multiple sclerosis liver cancers substrates histones histone 3 lysine residue 4 H3K4 p53 transcription factors TAF10 mono-methylated mono-methylase DNA damage acetylation human tumorigenesis inhibitors acceptor peptides S-adenosylhomocysteine S-ribosylhomocysteine adenine nucleosidase hypoxanthine deaminase urate hydrogen peroxide H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazine resorufin fluorescence measures measurement assays kits 24.872556970425
700350 SET8 Methyltransferase Inhibitor Screening Assay Kit - 2010-03-09 21.155178831055 set8-methyltransferase-inhibitor-screening-assay-kit SET domain-containing (lysine methyltransferase) 8; PR-Set7; SETD8 assays kits measures measurement methyltransferases MTs inhibits inhibitors inhibition methylation signal transduction biosynthesis protein repair genes silencing chromatins regulation S-adenosylmethionine (SAM)-dependent AdoMet DNA deoxyribonucleic acids Alzheimer's diseases depression Parkinson's multiple sclerosis livers cancers KMT5A lysines PR-Set 7 methylates histones H4 residues 20 H4K20 transcriptional p53 tumors suppressors tumorigenesis inhibits inhibition inhibitors peptides S-adenosylhomocysteines S-ribosylhomocysteines adenines nucleosidases hypoxanthines deaminases hydrogen peroxides H2O2 ADHP 10-acetyl-3,7-dihydroxyphenoxazines fluorescent fluorescence resorufin 21.155178831055
10010401 SIRT1 Direct Fluorescent Screening Assay Kit - 2008-02-26 51.236933701657 sirt1-direct-fluorescent-screening-assay-kit SIRT 1 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human homologs yeast SIR2 silent information regulators 2 tumors cancers suppressors inhibits inhitors inhibition apoptosis screening fluorescence activators fluorescent fluorometric 51.236933701657
10010991 SIRT1 FRET-Based Screening Assay Kit - 2008-02-19 20.010414364640 sirt1-fret-based-screening-assay-kit SIRT 1 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human homologs yeast SIR2 silent information regulators 2 tumors cancers suppressors inhibits inhitors inhibition apoptosis screening fluorescence activators fluorescent fluorometric 20.010414364640
700280 SIRT2 Direct Fluorescent Screening Assay Kit - 2009-12-10 40.755135213724 sirt2-direct-fluorescent-screening-assay-kit Nucleosomes chromosomal deoxyribonucleases DNA histones H2A H2B H3 H4 octameric cores transcription amino termini acetylation phosphorylation methylation ε-amino lysines acetyltransferases HATs chromatins genes activation deacetylases HDACs catalyzes hydrolytic acetyls sirtuins trichostatins A-insensitive lysyl-deacetylases class III catalyzes deacetylation nicotinamides O-acetyl-ADP-ribose NAD+ human SIRT1 SIRT2 SIRT3 SIRT4 SIRT5 SIRT6 SIRT7 cytoplasmic proteins H4 lysine-16 lysine-40 α-tubulin a-tubulin alpha-tubulin HDAC6 microtubules mitotic chromosomal hyperpolid cells tissues skeletal muscle heart oligodendroglia brain tumor suppressor gliomas Down-regulation gene chromosomal region diagnostic marker fluorescence-based inhibitors activators p53 Gln-Pro-Lys-Lys(ε-acetyl)-AMC recombinant NAD+ fluorescent fluorescence kits assays measures measurement 40.755135213724
700290 SIRT6 Direct Fluorescent Screening Assay Kit - 2010-02-18 37.424678867403 sirt6-direct-fluorescent-screening-assay-kit SIRT 6 SIRT-6 assays kits measures sirtuins trichostatins A-intensive lysyl-deacetylases class III HDACs human mitochondrial nuclear proteins mitochondrias translocated nucleus cells cellular stress lysine deacetylation nicotinamides O-acetyl-ADP-ribose NAD+ abstracted ADP-ribosyl transferases deacetylases telomeres chromatins NF-κB NF-kappaB NF-.kappa.B signaling signalling mammalian cells Werner Syndromes aging disorders anti-cancers anti-inflammatory drugs apoptosis screening fluorescence activators Arg-His-Lys-Lys(ε-acetyl)-AMC fluorescent fluorometric 37.424678867403
10011671 Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit - 2009-02-24 8.720009208103 soluble-epoxide-hydrolase-inhibitor-screening-assay-kit sEH Inhibitor Screening Assay Kit epoxides hydrolases sEHs inhibits inhibition assays kits fluorescence-based catalyzes hydrolysis exogenous endogenous vicinal diols substrates EETs epoxyeicosatrienoic acids vasodilatory vasodilation anti-inflammatory molecules therapy therapeutics hypertension vascular diseases PHOME (3-phenyl-oxiranyl)-acetic acid cyano-(6-methoxy-naphthalen-2-yl)-methyl ester 6-methoxy-2-naphthaldehyde excitation emission wavelengths a/b-hydrolases alpha/beta-hydrolases .alpha./.beta.-hydrolases enzymes homodimers C-terminal C-terminus animals models cyanohydrins cyanide ions 8.720009208103
700330 Sphingomyelinase Inhibitor Screening Assay Kit - 2010-02-09 42.857868184608 sphingomyelinase-inhibitor-screening-assay-kit SMase assays kits measures measuring measurementsphingomyelinases SMases hydrolases enzymes sphingolipids metabolisms DNase I superfamily phosphocholines ceramides cellular cells stress pathophysiological lysosomal digestion ceramide-mediated signal transductions cytokine-induced apoptosis differentiation immune inflammatory lipoproteins aggregation vessels atherogenesis intracellular trafficking acidic neutral proliferation depressive disorders neurodegenerative disorders strokes Alzheimer's dementia diseases therapeutics cleavage conjugates free thiols 42.857868184608
700430 Sphingosine Kinase 1 Inhibitor Screening Assay Kit - 2010-09-16 46.168646408839 sphingosine-kinase-1-inhibitor-screening-assay-kit SPHK 1 kits assays measures measurements SK1 SPHK1 sphingolipids metabolic pathways phosphorylates D-erythro-sphingosines sphingosine-1-phosphates S1P cells proliferations migrations cytoskeletal morphogenesis SPHK2 2 mammalian signalling signaling masts TNF-a TNFa TNF-alpha TNFalpha TNF-α TNFα-triggered Tumors Necrosis Factor-α fibroblasts epithelial mRNA messenger ribonucleic acids levels brains oncogenics erythroleukemias therapy therapeutics cancers inflammation up-regulated phagocytes peritoneal sepsis mice murine mouse inhibition inhibitors inhibits septic shock fluorescence-based fluorescent ATP adenosine triphosphates phosphorylates phosphorylation C-18 ADP diphosphates hydrogen peroxides H2O2 resorufin 46.168646408839
10004883 sPLA2 (Type V) Inhibitor Screening Assay Kit - 2004-05-07 52.717553275453 spla2-type-v-inhibitor-screening-assay-kit Secretory Phospholipase A2 (Type V) assays measures kits inhibition inhibitors phospholipases inflammation eicosanoids colorimetric sPLA2s enzymes diheptanoyl thio-pc 52.717553275453
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