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Holiday Notification: Cayman Chemical will be closed Monday, May 28, 2012, in observance of the Memorial Day holiday. More…
Please feel free to continue placing orders via our website or via fax at 734-971-3640. You may send an email to customer service at custserv@caymanchem.com , or to technical support at techserv@caymanchem.com which we will respond to the next business day. Cayman will resume regular business hours and shipping schedules on Tuesday, May 29, 2012. Thank you for your patience and understanding.

Chemical Class · Kinases

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Item Number Product Sizes & Pricing CAS Purity Image Exclusive Introduction Date Mojo Plain Text Name Synonyms Keywords Interest
10010079 Akt (human recombinant) Western Ready Control Exclusive - 2008-08-26 3.961519337016 akt-human-recombinant-western-ready-control Protein Kinase B; PKB; AKT1 western blots proteins antibodies antiserum antisera WB kinases serine threonine hexahistidine his-tag his-tagged N-terminal immunoblotting blotting 3.961519337016
11226 AS-703026 New 1236699-92-5 ≥98% 2012-03-08 27.541067090939 as-703026 MSC1936369B AS 703026 AS703026 1204531-26-9 MEKs MEK1/2 MEK-1/2 MEK1 MEK2 ERKs Ras Raf inhibitors inhibits inhibitions cancers multiple myeloma EGFR signals transductions kinases cells biology 27.541067090939
11020 Bisindolylmaleimide II New 137592-45-1 ≥97% (isomer mixture) 2012-03-13 33.836712196878 bisindolylmaleimide-ii PKC staurosporines inhibitors inhibits inhibition PDK1 PKA kinases C PKCα signaling insulin ligands binding protein kinase C 33.836712196878
11073 Bisindolylmaleimide XI (hydrochloride) New 145333-02-4 ≥98% 2012-03-21 37.214390955495 bisindolylmaleimide-xi-hydrochloride Ro 32-0432 131848-98-1 Ro32-0432 Ro-32-0432 Ro-320432 Ro 320432 Ro320432 PKC isozymes Staurosporine inhibitors inhibits inhibition proteins kinases C PKCα PKCβI PKCε hydrochloride HCl cells hearts T-cell T cell inflammatory inflammation 37.214390955495
10990 Glucokinase (human liver recombinant) - ≥85% 2011-09-08 72.112744014733 glucokinase-human-liver-recombinant Human Hexokinase IV isoform 2; Hexokinase D; ATP:D-Hexose 6-Phosphotransferase GCK metabolism insulin non-insulin-dependent (type 2) diabetes mellitus glucose kinases GCK ATP-dependent phosphorylation glycolytic liver tissues neurons pancreatic cells pituitary endocrine hexokinases mutations active 72.112744014733
10989 Glucokinase (human pancreatic recombinant) - ≥90% 2011-09-08 72.873333333333 glucokinase-human-pancreatic-recombinant Human Hexokinase IV isoform 1; Hexokinase D; ATP:D-Hexose 6-Phosphotransferase GCK metabolism insulin non-insulin-dependent (type 2) diabetes mellitus glucose kinases GCK ATP-dependent phosphorylation glycolytic liver tissues neurons pancreatic cells pituitary endocrine hexokinases mutations active 72.873333333333
11569 GSK 1059615 New 958852-01-2 ≥98% 2012-03-15 30.959325890116 gsk-1059615 Phosphatidylinositols PI 3-kinases α PI3Ks PI3Kα PI3Ka PI3K.alpha. inhibits inhibitors inhibition thiazolidinediones cells growth human cancers ATP-competitive p110α p110.alpha. p110a E542K E545K H1047R BT474 tumors xenografts MAPKs signaling biology signals transductions 30.959325890116
10505 Kinase Screening Library (96-Well) - 2010-08-09 15.102751381215 kinase-screening-library-96-well screening kinases inhibitors 15.102751381215
10348 Sphingosine Kinase 1 (human recombinant) - ≥90% by SDS-PAGE 2011-04-12 43.316690105475 sphingosine-kinase-1-human-recombinant SPHK1; SK1 sphingosines phosphates ceramides apoptosis acids cells death kinases sphingomyelin growth calcium active 43.316690105475
10009237 Sphingosine Kinase 2 (human recombinant) - >80% by SDS-PAGE 2007-01-18 34.970201262825 sphingosine-kinase-2-human-recombinant SPHK 2; SK2 signalling inflammatory enzymes proteins GenBank Accession No AF245447 SK2 SPK2 kinases sphingolipids SPHKs D-erythro-sphingosines phosphorylates sphingosine-1-phosphates S1Ps isoforms mammalian cells signals signaling pathways cancers inflammation proliferation apoptosis calcium homeostasis angiogenesis vascular maturation diseases active 34.970201262825
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