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Product TypeClear Filters

Biochemicals (6)
Small Molecule Modulators (70)
Small Molecule Inhibitors (70)
Acetyltransferases (5)
ATPases (2)
Chromatin Reader Interactions (70)
Deacetylases (2)
DNA Repair Enzymes (1)
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Cancer (34)
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Epigenetics, Transcription, & Translation (70)
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Readers (70)
Bromodomains (70)
PHD Domains (1)
RNA, DNA, & Protein Synthesis (1)
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Click Chemistry (1)
Displaying 1 - 25 of 70 Results
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(+)-JQ1

An inhibitor of BRD bromodomains

CAS No. 1268524-70-4

Item No. 11187


Formulation: A crystalline solid
Purity: ≥98%

    1 mg

    $31

    Add

    5 mg

    $108

    Add

    10 mg

    $154

    Add

    25 mg

    $270

    Add

    I-BET151

    A BRD2, BRD3, and BRD4 inhibitor

    CAS No. 1300031-49-5

    Item No. 11181


    Formulation: A crystalline solid
    Purity: ≥98%
    • GSK1210151A

    1 mg

    $40

    Add

    5 mg

    $108

    Add

    10 mg

    $197

    Add

    25 mg

    $443

    Add

    I-BET762

    Inhibitor of BET proteins

    CAS No. 1260907-17-2

    Item No. 10676


    Formulation: A crystalline solid
    Purity: ≥98%
    • GSK525762A

    1 mg

    $36

    Add

    5 mg

    $120

    Add

    10 mg

    $219

    Add

    25 mg

    $502

    Add

    OTX015

    A BRD2, BRD3, and BRD4 inhibitor

    CAS No. 202590-98-5

    Item No. 15947


    Formulation: A crystalline solid
    Purity: ≥95%
    • HY-15743
    • (−)-OTX015

    1 mg

    $54

    Add

    5 mg

    $172

    Add

    10 mg

    $238

    Add

    AZD 5153

    A BRD4 inhibitor

    CAS No. 1869912-39-9

    Item No. 20864


    Formulation: A crystalline solid
    Purity: ≥95%

      1 mg

      $42

      Add

      5 mg

      $194

      Add

      10 mg

      $322

      Add

      25 mg

      $653

      Add

      SGC-CBP30

      A potent inhibitor of CREBBP/EP300 bromodomains

      CAS No. 1613695-14-9

      Item No. 14469


      Formulation: A crystalline solid
      Purity: ≥98%

        5 mg

        $121

        Add

        10 mg

        $229

        Add

        50 mg

        $894

        Add

        I-CBP112 (hydrochloride)

        A p300 and CBP inhibitor

        CAS No. 2147701-33-3

        Item No. 14468


        Formulation: A crystalline solid
        Purity: ≥90%

          1 mg

          $49

          Add

          5 mg

          $190

          Add

          10 mg

          $283

          Add

          RVX-208

          A selective BET bromodomain antagonist

          CAS No. 1044870-39-4

          Item No. 16424


          Formulation: A crystalline solid
          Purity: ≥98%
          • Apabetalone
          • RVX-000222

          1 mg

          $49

          Add

          5 mg

          $120

          Add

          10 mg

          $213

          Add

          25 mg

          $445

          Add

          CPI-203

          A bioavailable inhibitor of BET bromodomains

          CAS No. 1446144-04-2

          Item No. 15479


          Formulation: A crystalline solid
          Purity: ≥98%

            1 mg

            $63

            Add

            5 mg

            $274

            Add

            10 mg

            $454

            Add

            25 mg

            $678

            Add

            I-BRD9

            A BRD9 bromodomain inhibitor

            CAS No. 1714146-59-4

            Item No. 17749


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $81

              Add

              5 mg

              $159

              Add

              10 mg

              $255

              Add

              50 mg

              $1,064

              Add

              (+)-JQ1 (free acid)

              A selective inhibitor of BET bromodomains

              CAS No. 202592-23-2

              Item No. 9002910


              Formulation: A crystalline solid
              Purity: ≥98%

                1 mg

                $60

                Add

                5 mg

                $213

                Add

                10 mg

                $310

                Add

                25 mg

                $702

                Add

                PFI-1

                A BET bromodomain inhibitor

                CAS No. 1403764-72-6

                Item No. 11155


                Formulation: A crystalline solid
                Purity: ≥98%
                • PF-06405761

                1 mg

                $42

                Add

                5 mg

                $115

                Add

                10 mg

                $183

                Add

                25 mg

                $402

                Add

                Bromosporine

                A non-specific bromodomain inhibitor

                CAS No. 1619994-69-2

                Item No. 14119


                Formulation: A crystalline solid
                Purity: ≥98%

                  1 mg

                  $41

                  Add

                  5 mg

                  $119

                  Add

                  10 mg

                  $215

                  Add

                  25 mg

                  $389

                  Add

                  ABBV-075

                  A BRD2, BRD4, and BRDT inhibitor

                  CAS No. 1445993-26-9

                  Item No. 21033


                  Formulation: A crystalline solid
                  Purity: ≥98%
                  • Mivebresib

                  500 µg

                  $36

                  Add

                  1 mg

                  $68

                  Add

                  5 mg

                  $186

                  Add

                  10 mg

                  $336

                  Add

                  TP-472

                  A BRD9 inhibitor

                  CAS No. 2079895-62-6

                  Item No. 20030


                  Formulation: A solid
                  Purity: ≥98%

                    1 mg

                    $36

                    Add

                    5 mg

                    $153

                    Add

                    Trotabresib

                    A BRD4 inhibitor

                    CAS No. 1706738-98-8

                    Item No. 36292


                    Formulation: A solid
                    Purity: ≥98%
                    • BMS-986378
                    • CC-90010

                    1 mg

                    $49

                    Add

                    5 mg

                    $182

                    Add

                    10 mg

                    $339

                    Add

                    25 mg

                    $723

                    Add

                    NVS-CECR2-1

                    A potent and selective CECR2 inhibitor

                    CAS No. 1992047-61-6

                    Item No. 18316


                    Formulation: A crystalline solid
                    Purity: ≥95%
                    • NVS-1

                    1 mg

                    $90

                    Add

                    5 mg

                    $241

                    Add

                    10 mg

                    $436

                    Add

                    25 mg

                    $869

                    Add

                    I-BET726

                    A selective inhibitor of BET family proteins

                    CAS No. 1300031-52-0

                    Item No. 16872


                    Formulation: A crystalline solid
                    Purity: ≥98%
                    • GSK1324726A

                    1 mg

                    $46

                    Add

                    5 mg

                    $157

                    Add

                    10 mg

                    $290

                    Add

                    25 mg

                    $662

                    Add

                    BAZ2-ICR

                    A BAZ2A/B bromodomain inhibitor

                    CAS No. 1665195-94-7

                    Item No. 17448


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      1 mg

                      $50

                      Add

                      5 mg

                      $171

                      Add

                      10 mg

                      $266

                      Add

                      25 mg

                      $602

                      Add

                      BI-9564

                      A selective BRD9/7 bromodomain inhibitor

                      CAS No. 1883429-22-8

                      Item No. 17897


                      Formulation: A crystalline solid
                      Purity: ≥98%

                        500 µg

                        $36

                        Add

                        1 mg

                        $61

                        Add

                        10 mg

                        $236

                        Add

                        BI-7273

                        A potent BRD9 bromodomain inhibitor

                        CAS No. 1883429-21-7

                        Item No. 20311


                        Formulation: A crystalline solid
                        Purity: ≥98%

                          1 mg

                          $41

                          Add

                          5 mg

                          $178

                          Add

                          10 mg

                          $312

                          Add

                          25 mg

                          $631

                          Add

                          BMS 986158

                          A BET bromodomain inhibitor

                          CAS No. 1800340-40-2

                          Item No. 27789


                          Formulation: A solid
                          Purity: ≥98%

                            1 mg

                            $105

                            Add

                            5 mg

                            $262

                            Add

                            10 mg

                            $418

                            Add

                            25 mg

                            $654

                            Add

                            LP99

                            A selective inhibitor of BRD7/9

                            CAS No. 1808951-93-0

                            Item No. 17661


                            Formulation: A crystalline solid
                            Purity: ≥98%

                              500 µg

                              $54

                              Add

                              1 mg

                              $96

                              Add

                              5 mg

                              $315

                              Add

                              GSK4027

                              A PCAF/GCN5 bromodomain inhibitor

                              CAS No. 2079896-25-4

                              Item No. 23421


                              Formulation: A crystalline solid
                              Purity: ≥95%

                                1 mg

                                $49

                                Add

                                5 mg

                                $154

                                Add

                                10 mg

                                $283

                                Add

                                L-Moses (hydrochloride)

                                A PCAF bromodomain inhibitor

                                CAS No. 2922480-38-2

                                Item No. 21288


                                Formulation: A crystalline solid
                                Purity: ≥98%
                                • L-45

                                1 mg

                                $41

                                Add

                                5 mg

                                $178

                                Add

                                10 mg

                                $312

                                Add

                                25 mg

                                $680

                                Add

                                Displaying 1 - 25 of 70 Results
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