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View New Products (12)

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Analytical Chemistry (141)
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Small Molecule Modulators (1,426)
Ion Channel Modulators (71)
Receptor Pharmacology (1,426)
Agonists (124)
Allosteric Modulators (11)
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Displaying 1 - 25 of 1,426 Results
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Tamoxifen

An estrogen receptor antagonist

CAS No. 10540-29-1

Item No. 13258


Formulation: A crystalline solid
Purity: ≥95%
  • TMX

500 mg

$72

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1 g

$137

Add

5 g

$609

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10 g

$930

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Mifepristone

A glucocorticoid, progesterone, and androgen receptor antagonist

CAS No. 84371-65-3

Item No. 10006317


Formulation: A crystalline solid
Purity: ≥98%
  • RU-486

100 mg

$40

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500 mg

$109

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1 g

$198

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5 g

$693

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Ramatroban

A dual TP and DP2/CRTH2 receptor antagonist

CAS No. 116649-85-5

Item No. 10156


Formulation: A crystalline solid
Purity: ≥98%
  • Bay u3405

1 mg

$36

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5 mg

$106

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10 mg

$183

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50 mg

$820

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AL 8810

A potent, selective FP receptor antagonist

CAS No. 246246-19-5

Item No. 16735


Formulation: A crystalline solid
Purity: ≥98%

    1 mg

    $119

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    5 mg

    $505

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    10 mg

    $891

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    25 mg

    $1,782

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    GW 9662

    A PPARγ antagonist

    CAS No. 22978-25-2

    Item No. 70785


    Formulation: A crystalline solid
    Purity: ≥98%

      1 mg

      $28

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      5 mg

      $62

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      10 mg

      $97

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      25 mg

      $207

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      JTE-013

      An S1P2 and S1P4 receptor antagonist

      CAS No. 383150-41-2

      Item No. 10009458


      Formulation: A crystalline solid
      Purity: ≥98%

        1 mg

        $29

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        5 mg

        $108

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        10 mg

        $149

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        50 mg

        $602

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        AM251

        A CB1 receptor antagonist

        CAS No. 183232-66-8

        Item No. 71670


        Formulation: A crystalline solid
        Purity: ≥98%

          5 mg

          $61

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          10 mg

          $109

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          50 mg

          $363

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          100 mg

          $666

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          SQ 29,548

          A selective TP receptor antagonist

          CAS No. 98672-91-4

          Item No. 19025


          Formulation: A crystalline solid
          Purity: ≥98%

            1 mg

            $94

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            5 mg

            $422

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            10 mg

            $748

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            25 mg

            $1,403

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            (E/Z)-4-hydroxy Tamoxifen

            A mixture of (E)-4-hydroxy tamoxifen and (Z)-4-hydroxy tamoxifen

            CAS No. 68392-35-8

            Item No. 17308


            Formulation: A crystalline solid
            Purity: ≥98% (mixture of isomers)
            • Afimoxifene
            • 4-OHT

            5 mg

            $42

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            10 mg

            $80

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            25 mg

            $189

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            50 mg

            $293

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            (Z)-4-hydroxy Tamoxifen

            An active metabolite of tamoxifen

            CAS No. 68047-06-3

            Item No. 14854


            Formulation: A crystalline solid
            Purity: ≥98%
            • ICI 79280
            • trans-4-hydroxy Tamoxifen

            1 mg

            $43

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            5 mg

            $161

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            10 mg

            $215

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            25 mg

            $483

            Add

            SR 144528

            A CB2 receptor antagonist

            CAS No. 192703-06-3

            Item No. 9000491


            Formulation: A crystalline solid
            Purity: ≥98%

              5 mg

              $129

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              10 mg

              $245

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              25 mg

              $574

              Add

              50 mg

              $1,016

              Add

              Ki16425

              A selective LPA1 and LPA3 receptor antagonist

              CAS No. 355025-24-0

              Item No. 10012659


              Formulation: A crystalline solid
              Purity: ≥95%

                1 mg

                $41

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                5 mg

                $108

                Add

                10 mg

                $157

                Add

                100 mg

                $970

                Add

                Plerixafor (hydrochloride hydrate)

                An antagonist of CXCR4

                Item No. 10011332


                Formulation: A crystalline solid
                Purity: ≥98%
                • AMD 3100
                • JM 3100
                • SID 791

                1 mg

                $28

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                5 mg

                $104

                Add

                10 mg

                $193

                Add

                50 mg

                $620

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                Rimonabant

                A CB1 receptor antagonist

                CAS No. 168273-06-1

                Item No. 9000484


                Formulation: A crystalline solid
                Purity: ≥98%
                • SR141716

                5 mg

                $29

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                10 mg

                $52

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                25 mg

                $108

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                50 mg

                $172

                Add

                BW A868C

                A DP receptor antagonist

                CAS No. 118675-50-6

                Item No. 12060


                Formulation: A 10 mg/ml solution in ethanol
                Purity: ≥98%

                  1 mg

                  $96

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                  5 mg

                  $423

                  Add

                  10 mg

                  $748

                  Add

                  CV-6209 (chloride)

                  A potent PAF receptor antagonist

                  CAS No. 100488-87-7

                  Item No. 15955


                  Formulation: A crystalline solid
                  Purity: ≥95%

                    500 µg

                    $107

                    Add

                    1 mg

                    $182

                    Add

                    5 mg

                    $794

                    Add

                    AH 6809

                    An EP and DP receptor antagonist

                    CAS No. 33458-93-4

                    Item No. 14050


                    Formulation: A crystalline solid
                    Purity: ≥97%

                      1 mg

                      $21

                      Add

                      5 mg

                      $86

                      Add

                      10 mg

                      $152

                      Add

                      50 mg

                      $655

                      Add

                      CAY10471

                      A potent, highly selective CRTH2/DP2 receptor antagonist

                      CAS No. 627865-18-3

                      Item No. 10006735


                      Formulation: A crystalline solid
                      Purity: ≥95%
                      • TM30089

                      1 mg

                      $74

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                      5 mg

                      $327

                      Add

                      10 mg

                      $578

                      Add

                      50 mg

                      $2,522

                      Add

                      Losartan (potassium salt)

                      An AT1b antagonist

                      CAS No. 124750-99-8

                      Item No. 10006594


                      Formulation: A crystalline solid
                      Purity: ≥98%
                      • DuP-753
                      • MK 954

                      10 mg

                      $19

                      Add

                      50 mg

                      $74

                      Add

                      100 mg

                      $130

                      Add

                      500 mg

                      $561

                      Add

                      TAK-242

                      A TLR4 antagonist

                      CAS No. 243984-11-4

                      Item No. 13871


                      Formulation: A crystalline solid
                      Purity: ≥98%
                      • Resatorvid

                      1 mg

                      $81

                      Add

                      5 mg

                      $239

                      Add

                      10 mg

                      $436

                      Add

                      25 mg

                      $887

                      Add

                      MK-571 (sodium salt)

                      A CysLT1 receptor antagonist

                      CAS No. 115103-85-0

                      Item No. 70720


                      Formulation: A crystalline solid
                      Purity: ≥95%
                      • L-660,711

                      1 mg

                      $36

                      Add

                      5 mg

                      $70

                      Add

                      10 mg

                      $120

                      Add

                      50 mg

                      $502

                      Add

                      U-75302

                      A BLT1 receptor antagonist

                      CAS No. 119477-85-9

                      Item No. 70705


                      Formulation: A 500 µg/ml solution in ethanol
                      Purity: ≥95%

                        50 µg

                        $96

                        Add

                        100 µg

                        $183

                        Add

                        500 µg

                        $764

                        Add

                        1 mg

                        $1,050

                        Add

                        Tauro-β-muricholic Acid (sodium salt)

                        An FXR receptor antagonist

                        CAS No. 145022-92-0

                        Item No. 20289


                        Formulation: A crystalline solid
                        Purity: ≥95%
                        • Tauro-β-muricholate
                        • TβMCA

                        500 µg

                        $86

                        Add

                        1 mg

                        $154

                        Add

                        5 mg

                        $472

                        Add

                        CAY10441

                        An IP receptor antagonist

                        CAS No. 221529-58-4

                        Item No. 10005186


                        Formulation: A crystalline solid
                        Purity: ≥98%
                        • Ro 1138452

                        5 mg

                        $165

                        Add

                        10 mg

                        $253

                        Add

                        25 mg

                        $614

                        Add

                        50 mg

                        $1,008

                        Add

                        GANT 61

                        Antagonist of Gli transcription factors, involved in Hedgehog signaling

                        CAS No. 500579-04-4

                        Item No. 13841


                        Formulation: A crystalline solid
                        Purity: ≥98%
                        • NSC 136476

                        5 mg

                        $65

                        Add

                        10 mg

                        $117

                        Add

                        25 mg

                        $260

                        Add

                        50 mg

                        $455

                        Add

                        Displaying 1 - 25 of 1,426 Results
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