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Product TypeClear Filters

Analytical Chemistry (6)
Biochemicals (48)
Antivirals (7)
Kinase Inhibitors (48)
Abl Family & Bcr-Abl (48)
Activin-like Kinases (ALKs) (1)
Aurora (5)
Dual Specificity Kinases (1)
EGFR/ErbB/HER Family (5)
FAK Family (1)
FGFR Family (5)
HGFR Family (1)
IGF-1R/InsR Family (1)
JAK Family (3)
LRRKs (1)
MAP3Ks (2)
mTOR (1)
Neurotrophin Receptor/Trk Family (3)
p38 MAPK (1)
PDGFR Family (14)
PI3K (1)
RAF (1)
RET (3)
SRC Family (20)
Syk Family (1)
Tec Family (3)
Tie Family (1)
VEGFR Family (7)
Other Non-Receptor Tyrosine Kinases (4)
Other Receptor Tyrosine Kinases (3)
Other Serine/Threonine Kinases (1)
Xenobiotic Metabolites (2)
Natural Products (1)
Small Molecule Modulators (48)

Research AreaClear Filters

Cancer (42)
Cardiovascular System (4)
Cell Biology (13)
Endocrinology & Metabolism (2)
Epigenetics, Transcription, & Translation (1)
Immunology & Inflammation (10)
Infectious Disease (7)
Neuroscience (4)
Xenobiotic Metabolism (2)

ApplicationClear Filters

Mass Spectrometry (6)
Displaying 1 - 25 of 48 Results
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Imatinib (mesylate)

An inhibitor of c-Abl, Bcr-Abl, PDGFR, and c-Kit

CAS No. 220127-57-1

Item No. 13139


Formulation: A crystalline solid
Purity: ≥98%
  • CGP57148B
  • STI-571

25 mg

$38

Add

50 mg

$72

Add

100 mg

$97

Add

500 mg

$449

Add

1-NA-PP1

Inhibitor of modified ‘analog-sensitive’ kinases

CAS No. 221243-82-9

Item No. 10954


Formulation: A crystalline solid
Purity: ≥98%
  • 1-Naphthyl-PP1
  • PP1 Analog

1 mg

$26

Add

5 mg

$115

Add

10 mg

$198

Add

50 mg

$789

Add

Dasatinib

An inhibitor of Abl and Src

CAS No. 302962-49-8

Item No. 11498


Formulation: A crystalline solid
Purity: ≥98%
  • BMS 354825
  • Sprycel

10 mg

$36

Add

50 mg

$53

Add

100 mg

$88

Add

250 mg

$176

Add

Nilotinib

A Bcr-Abl inhibitor

CAS No. 641571-10-0

Item No. 10010422


Formulation: A crystalline solid
Purity: ≥95%
  • AMN107

5 mg

$28

Add

10 mg

$41

Add

25 mg

$81

Add

50 mg

$130

Add

Ponatinib

An inhibitor of native and mutant Bcr-Abl

CAS No. 943319-70-8

Item No. 11494


Formulation: A crystalline solid
Purity: ≥98%
  • AP 24534

1 mg

$32

Add

5 mg

$86

Add

10 mg

$109

Add

Bosutinib

An inhibitor of Src and Abl kinases

CAS No. 380843-75-4

Item No. 12030


Formulation: A crystalline solid
Purity: ≥98%
  • SKI 606

5 mg

$49

Add

10 mg

$73

Add

50 mg

$283

Add

100 mg

$469

Add

Saracatinib

A dual inhibitor of c-Src and Abl

CAS No. 379231-04-6

Item No. 11497


Formulation: A crystalline solid
Purity: ≥90%
  • AZD 0530

5 mg

$35

Add

10 mg

$59

Add

25 mg

$119

Add

50 mg

$168

Add

PD 166326

An inhibitor of c-src and certain receptor tyrosine kinases, including c-abl

CAS No. 185039-91-2

Item No. 9000988


Formulation: A crystalline solid
Purity: ≥95%

    1 mg

    $108

    Add

    5 mg

    $481

    Add

    10 mg

    $856

    Add

    AT-9283

    A broad spectrum kinase inhibitor

    CAS No. 896466-04-9

    Item No. 11496


    Formulation: A crystalline solid
    Purity: ≥98%

      5 mg

      $98

      Add

      10 mg

      $176

      Add

      25 mg

      $318

      Add

      50 mg

      $490

      Add

      Nilotinib-d6

      An internal standard for the quantification of nilotinib

      CAS No. 1268356-17-7

      Item No. 19280


      Formulation: A solid
      Purity: ≥99% deuterated forms (d1-d6)

        1 mg

        $569

        Add

        Herbimycin A

        An inhibitor of tyrosine kinases and Hsp90

        CAS No. 70563-58-5

        Item No. 15504


        Formulation: A yellow lyophilisate
        Purity: ≥95%
        • Antibiotic TAN 420F
        • NSC 305978

        500 µg

        $418

        Add

        2.5 mg

        $1,355

        Add

        N-desmethyl Imatinib

        A major active metabolite of imatinib

        CAS No. 404844-02-6

        Item No. 16947


        Formulation: A lyophilized solid
        Purity: ≥95%
        • N-desmethyl Gleevec
        • STI-509-00

        500 µg

        $42

        Add

        1 mg

        $79

        Add

        5 mg

        $303

        Add

        10 mg

        $561

        Add

        Dasatinib-d8

        An internal standard for the quantification of GC- or LC-MS

        CAS No. 1132093-70-9

        Item No. 22368


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1d8); ≤1% d0
        • Sprycel-d8

        500 µg

        $125

        Add

        1 mg

        $236

        Add

        AST-487

        A multi-kinase inhibitor

        CAS No. 630124-46-8

        Item No. 19477


        Formulation: A crystalline solid
        Purity: ≥98%
        • NVP-AST-487

        1 mg

        $37

        Add

        5 mg

        $124

        Add

        10 mg

        $229

        Add

        25 mg

        $523

        Add

        Asciminib

        An allosteric inhibitor of Abl1

        CAS No. 1492952-76-7

        Item No. 26126


        Formulation: A crystalline solid
        Purity: ≥95%
        • ABL001

        1 mg

        $69

        Add

        5 mg

        $280

        Add

        10 mg

        $525

        Add

        Danusertib

        A pan-Aurora kinase and Abl inhibitor

        CAS No. 827318-97-8

        Item No. 18387


        Formulation: A crystalline solid
        Purity: ≥95%
        • PHA-739358

        1 mg

        $42

        Add

        5 mg

        $147

        Add

        10 mg

        $230

        Add

        50 mg

        $627

        Add

        ALW-II-41-27

        A multi-kinase inhibitor

        CAS No. 1186206-79-0

        Item No. 25275


        Formulation: A crystalline solid
        Purity: ≥95%

          1 mg

          $69

          Add

          5 mg

          $297

          Add

          10 mg

          $525

          Add

          Imatinib-d3

          An internal standard for the quantification of imatinib

          CAS No. 1134803-18-1

          Item No. 18257


          Formulation: A solid
          Purity: ≥99% deuterated forms (d1-d3)
          • Genfatinib-d3

          500 µg

          $112

          Add

          1 mg

          $202

          Add

          CZC-8004

          A tyrosine kinase inhibitor

          CAS No. 916603-07-1

          Item No. 16718


          Formulation: A crystalline solid
          Purity: ≥98%
          • Dianilinopyrimidine-01

          500 µg

          $90

          Add

          1 mg

          $158

          Add

          5 mg

          $436

          Add

          10 mg

          $696

          Add

          GZD-824

          A Bcr/Abl inhibitor

          CAS No. 1257628-77-5

          Item No. 21508


          Formulation: A crystalline solid
          Purity: ≥98%
          • HQP1351
          • Olverembatinib

          1 mg

          $36

          Add

          5 mg

          $153

          Add

          10 mg

          $268

          Add

          25 mg

          $502

          Add

          Ponatinib-d8

          An internal standard for the quantification of ponatinib

          CAS No. 1562993-37-6

          Item No. 28905


          Formulation: A solid
          Purity: ≥99% deuterated forms (d1-d8)

            1 mg

            $390

            Add

            Radotinib

            A selective Bcr-Abl tyrosine kinase inhibitor

            CAS No. 926037-48-1

            Item No. 19923


            Formulation: A crystalline solid
            Purity: ≥98%
            • IY-5511

            1 mg

            $36

            Add

            5 mg

            $120

            Add

            10 mg

            $203

            Add

            25 mg

            $378

            Add

            MGCD-265

            A c-Met and VEGFR2 inhibitor

            CAS No. 875337-44-3

            Item No. 20097


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $48

              Add

              5 mg

              $190

              Add

              10 mg

              $355

              Add

              25 mg

              $708

              Add

              Bafetinib

              A Bcr-Abl inhibitor

              CAS No. 859212-16-1

              Item No. 19169


              Formulation: A crystalline solid
              Purity: ≥95%
              • INNO-406
              • NS-187

              1 mg

              $49

              Add

              5 mg

              $130

              Add

              10 mg

              $236

              Add

              KW 2449

              A multi-kinase inhibitor

              CAS No. 1000669-72-6

              Item No. 22207


              Formulation: A crystalline solid
              Purity: ≥98%

                5 mg

                $36

                Add

                10 mg

                $64

                Add

                25 mg

                $150

                Add

                50 mg

                $264

                Add

                Displaying 1 - 25 of 48 Results
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