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Product TypeClear Filters

Analytical Chemistry (3)
Biochemicals (56)
Kinase Inhibitors (56)
Abl Family & Bcr-Abl (1)
ATM (1)
ATR (2)
DNA-PK (6)
MAP3Ks (1)
mTOR (56)
PI3K (26)
SRC Family (1)
VEGFR Family (1)
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Small Molecule Modulators (56)

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Cancer (53)
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Mass Spectrometry (2)
Displaying 1 - 25 of 56 Results
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Rapamycin

An allosteric inhibitor of mTORC1

CAS No. 53123-88-9

Item No. 13346


Formulation: A crystalline solid
Purity: ≥95%
  • AY 22989
  • NSC 226080
  • Sirolimus
  • Wy 090217

1 mg

$43

Add

5 mg

$108

Add

10 mg

$194

Add

25 mg

$429

Add

Torin 1

Selective inhibitor of mTOR

CAS No. 1222998-36-8

Item No. 10997


Formulation: A crystalline solid
Purity: ≥95%

    10 mg

    $161

    Add

    25 mg

    $363

    Add

    50 mg

    $591

    Add

    PI-103

    A potent, cell-permeable PI3-kinase inhibitor

    CAS No. 371935-74-9

    Item No. 10009209


    Formulation: A crystalline solid
    Purity: ≥98%

      1 mg

      $33

      Add

      5 mg

      $125

      Add

      10 mg

      $186

      Add

      25 mg

      $347

      Add

      NVP-BEZ235

      A dual inhibitor of class I PI3Ks and mTOR

      CAS No. 915019-65-7

      Item No. 10565


      Formulation: A crystalline solid
      Purity: ≥98%
      • Dactolisib

      25 mg

      $49

      Add

      50 mg

      $86

      Add

      100 mg

      $152

      Add

      250 mg

      $259

      Add

      INK128

      Inhibitor of TORC1/2

      CAS No. 1224844-38-5

      Item No. 11811


      Formulation: A crystalline solid
      Purity: ≥98%
      • MLN0128

      1 mg

      $28

      Add

      5 mg

      $49

      Add

      10 mg

      $83

      Add

      50 mg

      $275

      Add

      Torin 2

      Selective inhibitor of mTOR

      CAS No. 1223001-51-1

      Item No. 14185


      Formulation: A crystalline solid
      Purity: ≥98%

        5 mg

        $95

        Add

        10 mg

        $178

        Add

        25 mg

        $370

        Add

        Rapamycin-d3

        An internal standard for the quantification of rapamycin

        CAS No. 392711-19-2

        Item No. 22093


        Formulation: A 1 mg/ml solution in ethanol
        Purity: ≥98% deuterated forms (d1-d3)
        • Sirolimus-d3

        500 µg

        $134

        Add

        1 mg

        $202

        Add

        AZD 8055

        A potent mTOR inhibitor

        CAS No. 1009298-09-2

        Item No. 16978


        Formulation: A crystalline solid
        Purity: ≥98%
        • CCG-168

        1 mg

        $49

        Add

        5 mg

        $96

        Add

        10 mg

        $143

        Add

        50 mg

        $423

        Add

        PP242

        Potent inhibitor of mTOR kinase in both mTORC1 and mTORC2

        CAS No. 1092351-67-1

        Item No. 13643


        Formulation: A crystalline solid
        Purity: ≥95%

          1 mg

          $36

          Add

          5 mg

          $91

          Add

          10 mg

          $147

          Add

          25 mg

          $319

          Add

          Everolimus-d4

          An internal standard for the quantification of everolimus

          CAS No. 1338452-54-2

          Item No. 22559


          Formulation: A solid
          Purity: ≥99% deuterated forms (d1-d4); ≤1% d0

            500 µg

            $160

            Add

            1 mg

            $289

            Add

            CAY10626

            A dual PI3Kα/mTOR kinase inhibitor

            CAS No. 1202884-94-3

            Item No. 13838


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $116

              Add

              5 mg

              $521

              Add

              10 mg

              $924

              Add

              25 mg

              $1,877

              Add

              GSK2126458

              A potent pan-PI3K and mTOR inhibitor

              CAS No. 1086062-66-9

              Item No. 17377


              Formulation: A crystalline solid
              Purity: ≥98%
              • GSK458
              • Omipalisib

              1 mg

              $54

              Add

              5 mg

              $238

              Add

              10 mg

              $418

              Add

              50 mg

              $1,303

              Add

              Ku-0063794

              An inhibitor of mTORC1 and mTORC2

              CAS No. 938440-64-3

              Item No. 13597


              Formulation: A crystalline solid
              Purity: ≥98%

                5 mg

                $81

                Add

                10 mg

                $152

                Add

                50 mg

                $436

                Add

                100 mg

                $633

                Add

                OSI-027

                Dual mTORC1/mTORC2 inhibitor

                CAS No. 936890-98-1

                Item No. 17379


                Formulation: A crystalline solid
                Purity: ≥98%

                  1 mg

                  $41

                  Add

                  5 mg

                  $148

                  Add

                  10 mg

                  $274

                  Add

                  50 mg

                  $737

                  Add

                  Wortmannin-Rapamycin Conjugate

                  Separate PI3K and mTORC1 inhibitors joined by prodrug linker

                  CAS No. 1067892-47-0

                  Item No. 13671


                  Formulation: A crystalline solid
                  Purity: ≥98%

                    500 µg

                    $168

                    Add

                    1 mg

                    $317

                    Add

                    5 mg

                    $1,325

                    Add

                    AZD 2014

                    A potent dual mTORC1/2 inhibitor

                    CAS No. 1009298-59-2

                    Item No. 17378


                    Formulation: A crystalline solid
                    Purity: ≥98%
                    • Vistusertib

                    1 mg

                    $36

                    Add

                    5 mg

                    $103

                    Add

                    10 mg

                    $161

                    Add

                    25 mg

                    $336

                    Add

                    WYE-125132

                    Dual mTORC1/mTORC2 inhibitor

                    CAS No. 1144068-46-1

                    Item No. 18372


                    Formulation: A crystalline solid
                    Purity: ≥98%
                    • WYE-132

                    500 µg

                    $41

                    Add

                    1 mg

                    $69

                    Add

                    5 mg

                    $106

                    Add

                    10 mg

                    $196

                    Add

                    17β-hydroxy Wortmannin

                    Inhibitor of phosphoinoside 3-kinase

                    CAS No. 58053-83-1

                    Item No. 13812


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      500 µg

                      $65

                      Add

                      1 mg

                      $119

                      Add

                      5 mg

                      $493

                      Add

                      10 mg

                      $862

                      Add

                      PF-05212384

                      A potent, dual PI3K/mTOR inhibitor

                      CAS No. 1197160-78-3

                      Item No. 14567


                      Formulation: A crystalline solid
                      Purity: ≥95%
                      • PK-1587
                      • PKI-587

                      1 mg

                      $41

                      Add

                      5 mg

                      $178

                      Add

                      10 mg

                      $312

                      Add

                      AZD 3147

                      A dual mTORC1/mTORC2 inhibitor

                      CAS No. 1101810-02-9

                      Item No. 22474


                      Formulation: A solid
                      Purity: ≥95%

                        500 µg

                        $36

                        Add

                        1 mg

                        $61

                        Add

                        5 mg

                        $219

                        Add

                        10 mg

                        $303

                        Add

                        MK-8669

                        A rapamycin analog that selectively inhibits mTOR in mTORC1

                        CAS No. 572924-54-0

                        Item No. 10543


                        Formulation: A crystalline solid
                        Purity: ≥95%
                        • AP23573
                        • Deforolimus
                        • Ridaforolimus

                        1 mg

                        $46

                        Add

                        5 mg

                        $202

                        Add

                        10 mg

                        $290

                        Add

                        WYE-28

                        An inhibitor of mTOR

                        CAS No. 1062172-60-4

                        Item No. 21200


                        Formulation: A crystalline solid
                        Purity: ≥98%

                          500 µg

                          $49

                          Add

                          1 mg

                          $93

                          Add

                          5 mg

                          $376

                          Add

                          10 mg

                          $655

                          Add

                          GDC-0980

                          A dual inhibitor of PI3K and mTOR

                          CAS No. 1032754-93-0

                          Item No. 18303


                          Formulation: A crystalline solid
                          Purity: ≥98%
                          • Apitolisib
                          • RG7422

                          1 mg

                          $69

                          Add

                          5 mg

                          $198

                          Add

                          10 mg

                          $329

                          Add

                          25 mg

                          $655

                          Add

                          WYE-354

                          Potent inhibitor of mTOR in both mTORC1 and mTORC2

                          CAS No. 1062169-56-5

                          Item No. 13604


                          Formulation: A crystalline solid
                          Purity: ≥98%

                            5 mg

                            $103

                            Add

                            10 mg

                            $194

                            Add

                            25 mg

                            $454

                            Add

                            50 mg

                            $801

                            Add

                            PF-04691502

                            A PI3Kα, -β, -δ, -γ, and mTOR inhibitor

                            CAS No. 1013101-36-4

                            Item No. 15017


                            Formulation: A crystalline solid
                            Purity: ≥95%
                            • HNC-VP-L
                            • PF-502

                            5 mg

                            $98

                            Add

                            10 mg

                            $157

                            Add

                            25 mg

                            $367

                            Add

                            50 mg

                            $636

                            Add

                            Displaying 1 - 25 of 56 Results
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