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Product TypeClear Filters

Biochemicals (34)
Antivirals (4)
Kinase Inhibitors (34)
CaMKs (1)
CDKs (2)
Checkpoint Kinases (1)
ERK (1)
GSK3 (1)
MEK (1)
PDGFR Family (1)
PDPK1/PDK1 (3)
PKA (8)
PKB/Akt (34)
PKC (3)
PKD & PKG (2)
ROCK (1)
S6K (5)
SRC Family (1)
TAM Family (1)
VEGFR Family (2)
Other Serine/Threonine Kinases (1)
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Phosphoinositides (2)
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Natural Products (2)
Small Molecule Modulators (34)

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Cancer (31)
Cell Biology (13)
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Displaying 1 - 25 of 34 Results
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D-myo-Inositol-1,3,4,5,6-pentaphosphate (sodium salt)

An anticancer inositol phosphate

Item No. 10007784


Formulation: A lyophilized powder
Purity: ≥98%
  • Ins(1,3,4,5,6)P5
  • 1,3,4,5,6-IP5

100 µg

$69

Add

500 µg

$297

Add

1 mg

$525

Add

KT 5720

A potent inhibitor of PKA

CAS No. 108068-98-0

Item No. 10011011


Formulation: A clear film
Purity: ≥98%

    50 µg

    $90

    Add

    100 µg

    $142

    Add

    250 µg

    $328

    Add

    500 µg

    $479

    Add

    Triciribine

    An Akt activation inhibitor and a prodrug form of triciribine phosphate

    CAS No. 35943-35-2

    Item No. 10010237


    Formulation: A crystalline solid
    Purity: ≥98%
    • API 2
    • NSC 154020
    • TCN
    • Tricyclic Nucleoside

    1 mg

    $52

    Add

    5 mg

    $118

    Add

    10 mg

    $182

    Add

    Akt Inhibitor VIII

    A potent inhibitor of Akt1 and Akt2

    CAS No. 612847-09-3

    Item No. 14870


    Formulation: A crystalline solid
    Purity: ≥98%

      500 µg

      $32

      Add

      1 mg

      $61

      Add

      5 mg

      $141

      Add

      10 mg

      $217

      Add

      PKC 412

      Kinase inhibitor with potential use in cancer treatment

      CAS No. 120685-11-2

      Item No. 10459


      Formulation: A crystalline solid
      Purity: ≥98%
      • N-Benzoylstaurosporine
      • CGP 41231
      • CGP 41251
      • Midostaurin

      1 mg

      $31

      Add

      5 mg

      $93

      Add

      10 mg

      $154

      Add

      25 mg

      $270

      Add

      D-myo-Inositol-1,3,4,5,6-pentaphosphate (ammonium salt)

      An anticancer inositol phosphate

      Item No. 10009851


      Formulation: A lyophilized powder
      Purity: ≥98%
      • Ins(1,3,4,5,6)P5
      • 1,3,4,5,6-IP5 (sodium salt)

      100 µg

      $69

      Add

      500 µg

      $297

      Add

      1 mg

      $525

      Add

      AZD 5363

      A pan-Akt inhibitor

      CAS No. 1143532-39-1

      Item No. 15406


      Formulation: A crystalline solid
      Purity: ≥98%
      • Capivasertib

      1 mg

      $54

      Add

      5 mg

      $149

      Add

      10 mg

      $270

      Add

      25 mg

      $472

      Add

      GDC-0068

      A pan-Akt inhibitor

      CAS No. 1001264-89-6

      Item No. 18412


      Formulation: A crystalline solid
      Purity: ≥98%
      • Ipatasertib
      • RG-7440

      1 mg

      $63

      Add

      5 mg

      $274

      Add

      10 mg

      $481

      Add

      25 mg

      $1,053

      Add

      TIC10

      A TRAIL-inducing compound

      CAS No. 1616632-77-9

      Item No. 16109


      Formulation: A crystalline solid
      Purity: ≥98%
      • Dordaviprone
      • ONC201

      1 mg

      $36

      Add

      5 mg

      $120

      Add

      10 mg

      $219

      Add

      25 mg

      $462

      Add

      Arctigenin

      A plant lignan with antioxidant, anti-inflammatory, antiproliferative, and antiviral activity

      CAS No. 7770-78-7

      Item No. 14913


      Formulation: A crystalline solid
      Purity: ≥95%

        10 mg

        $69

        Add

        25 mg

        $102

        Add

        50 mg

        $183

        Add

        100 mg

        $329

        Add

        ML-9

        A PKB/Akt inhibitor

        CAS No. 105637-50-1

        Item No. 10010236


        Formulation: A crystalline solid
        Purity: ≥98%

          10 mg

          $63

          Add

          50 mg

          $242

          Add

          100 mg

          $363

          Add

          250 mg

          $678

          Add

          UCN-01

          A nonspecific protein kinase inhibitor

          CAS No. 112953-11-4

          Item No. 18130


          Formulation: A 1 mg/ml solution in ethanol
          Purity: ≥95%
          • NSC 638850
          • ​7-hydroxy Staurosporine

          1 mg

          $197

          Add

          A-443654

          A pan Akt inhibitor

          CAS No. 552325-16-3

          Item No. 16499


          Formulation: A crystalline solid
          Purity: ≥98%

            500 µg

            $75

            Add

            1 mg

            $120

            Add

            5 mg

            $442

            Add

            GSK690693

            An Akt inhibitor

            CAS No. 937174-76-0

            Item No. 16891


            Formulation: A crystalline solid
            Purity: ≥95%

              1 mg

              $54

              Add

              5 mg

              $132

              Add

              10 mg

              $209

              Add

              25 mg

              $458

              Add

              Akt Inhibitor XI

              A cell-permeable Akt inhibitor

              CAS No. 902779-59-3

              Item No. 18604


              Formulation: A crystalline solid
              Purity: ≥95%
              • FPA-124

              1 mg

              $32

              Add

              5 mg

              $88

              Add

              10 mg

              $160

              Add

              25 mg

              $359

              Add

              Oridonin

              A diterpenoid with diverse biological activities

              CAS No. 28957-04-2

              Item No. 25665


              Formulation: A crystalline solid
              Purity: ≥98%
              • NSC 250682

              5 mg

              $52

              Add

              10 mg

              $86

              Add

              50 mg

              $227

              Add

              100 mg

              $396

              Add

              Akt Inhibitor IV

              An inhibitor of Akt activation

              CAS No. 681281-88-9

              Item No. 15569


              Formulation: A crystalline solid
              Purity: ≥95%

                1 mg

                $79

                Add

                5 mg

                $176

                Add

                10 mg

                $313

                Add

                25 mg

                $684

                Add

                KP372-1

                An Akt inhibitor

                CAS No. 1374996-60-7

                Item No. 17808


                Formulation: A crystalline solid
                Purity: ≥95% (sum of isomers)

                  1 mg

                  $81

                  Add

                  5 mg

                  $297

                  Add

                  10 mg

                  $553

                  Add

                  ARQ 092

                  An orally bioavailable pan-Akt inhibitor

                  CAS No. 1313881-70-7

                  Item No. 21388


                  Formulation: A crystalline solid
                  Purity: ≥98%

                    1 mg

                    $49

                    Add

                    5 mg

                    $190

                    Add

                    10 mg

                    $354

                    Add

                    25 mg

                    $762

                    Add

                    Afuresertib (hydrochloride)

                    A pan-Akt inhibitor

                    CAS No. 1047645-82-8

                    Item No. 17988


                    Formulation: A crystalline solid
                    Purity: ≥98%
                    • GSK2110183B

                    1 mg

                    $44

                    Add

                    5 mg

                    $152

                    Add

                    10 mg

                    $280

                    Add

                    25 mg

                    $642

                    Add

                    AT-13148

                    A multi-AGC kinase inhibitor

                    CAS No. 1056901-62-2

                    Item No. 21597


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      1 mg

                      $41

                      Add

                      5 mg

                      $148

                      Add

                      10 mg

                      $235

                      Add

                      25 mg

                      $341

                      Add

                      SC-66

                      A dual inhibitor of Akt

                      CAS No. 871361-88-5

                      Item No. 10876


                      Formulation: A crystalline solid
                      Purity: ≥98%

                        5 mg

                        $42

                        Add

                        10 mg

                        $79

                        Add

                        25 mg

                        $183

                        Add

                        100 mg

                        $561

                        Add

                        A-674563

                        An Akt inhibitor

                        CAS No. 552325-73-2

                        Item No. 18715


                        Formulation: A crystalline solid
                        Purity: ≥95%

                          500 µg

                          $54

                          Add

                          1 mg

                          $102

                          Add

                          5 mg

                          $367

                          Add

                          10 mg

                          $627

                          Add

                          CCT128930

                          An inhibitor of Akt2

                          CAS No. 885499-61-6

                          Item No. 18194


                          Formulation: A crystalline solid
                          Purity: ≥95%

                            1 mg

                            $28

                            Add

                            5 mg

                            $104

                            Add

                            10 mg

                            $193

                            Add

                            25 mg

                            $275

                            Add

                            Triciribine Phosphate

                            An Akt activation inhibitor and active metabolite of triciribine

                            CAS No. 61966-08-3

                            Item No. 37985


                            Formulation: A crystalline solid
                            Purity: ≥95%
                            • TCN-P
                            • Triciribine-5'-monophosphate
                            • NSC 280594

                            1 mg

                            $40

                            Add

                            5 mg

                            $187

                            Add

                            10 mg

                            $355

                            Add

                            Displaying 1 - 25 of 34 Results
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