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Analytical Chemistry (10)
Biochemicals (11)
Environmental Toxicology (1)
Natural Products (2)
Small Molecule Modulators (88)
Ion Channel Modulators (5)
Receptor Pharmacology (88)
Agonists (16)
Allosteric Modulators (1)
Antagonists (33)
Inverse Agonists (88)
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Mass Spectrometry (11)
Displaying 1 - 25 of 88 Results
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AM630

An inverse agonist at CB2 and partial agonist at CB1 receptors

CAS No. 164178-33-0

Item No. 10006974


Formulation: A crystalline solid
Purity: ≥98%
  • 6-Iodopravodoline

5 mg

$63

Add

10 mg

$118

Add

50 mg

$454

Add

100 mg

$842

Add

AM1241

A CB2 receptor agonist and inverse agonist

CAS No. 444912-48-5

Item No. 10010118


Formulation: A crystalline solid
Purity: ≥97%

    1 mg

    $36

    Add

    5 mg

    $86

    Add

    10 mg

    $153

    Add

    25 mg

    $336

    Add

    SR 3335

    A selective inverse agonist of RORα

    CAS No. 293753-05-6

    Item No. 12072


    Formulation: A crystalline solid
    Purity: ≥95%
    • ML 176

    1 mg

    $36

    Add

    5 mg

    $117

    Add

    10 mg

    $205

    Add

    25 mg

    $445

    Add

    BMS 493

    A pan-RAR inverse agonist

    CAS No. 215030-90-3

    Item No. 17418


    Formulation: A crystalline solid
    Purity: ≥98%
    • BMS 204493

    1 mg

    $49

    Add

    5 mg

    $120

    Add

    10 mg

    $213

    Add

    25 mg

    $469

    Add

    SR 2211

    Selective inverse agonist of RORγ

    CAS No. 1359164-11-6

    Item No. 11972


    Formulation: A crystalline solid
    Purity: ≥98%

      1 mg

      $41

      Add

      5 mg

      $148

      Add

      10 mg

      $178

      Add

      Ziprasidone-d8

      An internal standard for the quantification of ziprasidone

      CAS No. 1126745-58-1

      Item No. 30737


      Formulation: A solid
      Purity: ≥99% deuterated forms (d1-d8)
      • CP-88,059-d8

      1 mg

      $321

      Add

      N-Desmethylclozapine

      An active metabolite of clozapine

      CAS No. 6104-71-8

      Item No. 26153


      Formulation: A crystalline solid
      Purity: ≥98%
      • Norclozapine

      5 mg

      $102

      Add

      10 mg

      $172

      Add

      25 mg

      $380

      Add

      50 mg

      $557

      Add

      AM281

      A CB1 receptor antagonist/inverse agonist

      CAS No. 202463-68-1

      Item No. 10006972


      Formulation: A crystalline solid
      Purity: ≥98%

        1 mg

        $29

        Add

        5 mg

        $86

        Add

        10 mg

        $158

        Add

        11-cis Retinol

        An isomer of vitamin A

        CAS No. 22737-96-8

        Item No. 33207


        Formulation: An oil
        Purity: ≥85%
        • 11-cis Vitamin A Alcohol

        1 mg

        $334

        Add

        Paliperidone-d4

        An internal standard for the quantification of paliperidone

        CAS No. 1020719-55-4

        Item No. 28484


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d4)
        • 9-hydroxy Risperidone-d4

        500 µg

        $174

        Add

        1 mg

        $329

        Add

        Aripiprazole-d8

        An internal standard for the quantification of aripiprazole

        CAS No. 1089115-04-7

        Item No. 28487


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d8)

          1 mg

          $329

          Add

          SR9243

          An LXR inverse agonist

          CAS No. 1613028-81-1

          Item No. 18420


          Formulation: A crystalline solid
          Purity: ≥95%

            1 mg

            $36

            Add

            5 mg

            $77

            Add

            10 mg

            $120

            Add

            50 mg

            $387

            Add

            Dehydro Aripiprazole (hydrochloride)

            A metabolite of aripiprazole

            CAS No. 1008531-60-9

            Item No. 19539


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $107

              Add

              5 mg

              $371

              Add

              10 mg

              $688

              Add

              Paliperidone

              An atypical antipsychotic

              CAS No. 144598-75-4

              Item No. 15556


              Formulation: A crystalline solid
              Purity: ≥98%
              • 9-hydroxy Risperidone
              • RO76477

              25 mg

              $81

              Add

              50 mg

              $152

              Add

              100 mg

              $255

              Add

              500 mg

              $946

              Add

              8-hydroxy Amoxapine

              A metabolite of amoxapine

              CAS No. 61443-78-5

              Item No. 29192


              Formulation: A solid
              Purity: ≥95%

                1 mg

                $336

                Add

                IMMA

                A CB2 receptor inverse agonist

                CAS No. 2854-32-2

                Item No. 70275


                Formulation: A crystalline solid
                Purity: ≥98%
                • BML-190
                • Indomethacin Morpholinylamide
                • LM-4131

                5 mg

                $29

                Add

                10 mg

                $53

                Add

                50 mg

                $215

                Add

                100 mg

                $376

                Add

                CID-16020046

                A selective GPR55 inverse agonist

                CAS No. 834903-43-4

                Item No. 15247


                Formulation: A crystalline solid
                Purity: ≥98%

                  1 mg

                  $40

                  Add

                  5 mg

                  $124

                  Add

                  10 mg

                  $190

                  Add

                  25 mg

                  $376

                  Add

                  Loratadine

                  A histamine H1 receptor inverse agonist

                  CAS No. 79794-75-5

                  Item No. 15625


                  Formulation: A crystalline solid
                  Purity: ≥98%
                  • SCH 29851

                  5 mg

                  $49

                  Add

                  10 mg

                  $86

                  Add

                  25 mg

                  $143

                  Add

                  50 mg

                  $213

                  Add

                  SB-224289

                  A 5-HT1B receptor inverse agonist

                  CAS No. 180083-23-2

                  Item No. 17036


                  Formulation: A crystalline solid
                  Purity: ≥98%

                    5 mg

                    $63

                    Add

                    10 mg

                    $110

                    Add

                    25 mg

                    $229

                    Add

                    50 mg

                    $332

                    Add

                    SR 1555 (hydrochloride)

                    An inverse agonist of RORγ

                    CAS No. 2309312-90-9

                    Item No. 12071


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      1 mg

                      $36

                      Add

                      5 mg

                      $117

                      Add

                      10 mg

                      $205

                      Add

                      25 mg

                      $445

                      Add

                      Cimetidine-d3

                      An internal standard for the quantification of cimetidine

                      CAS No. 1185237-29-9

                      Item No. 29050


                      Formulation: A solid
                      Purity: ≥99% deuterated forms (d1-d3)

                        1 mg

                        $343

                        Add

                        CB-25

                        A stable analog of Δ9-THC

                        CAS No. 869376-63-6

                        Item No. 10010116


                        Formulation: A crystalline solid
                        Purity: ≥98%

                          1 mg

                          $36

                          Add

                          5 mg

                          $132

                          Add

                          10 mg

                          $253

                          Add

                          GSK2981278

                          An inverse agonist of RORγ

                          CAS No. 1474110-21-8

                          Item No. 20974


                          Formulation: A crystalline solid
                          Purity: ≥98%

                            1 mg

                            $41

                            Add

                            5 mg

                            $178

                            Add

                            10 mg

                            $312

                            Add

                            25 mg

                            $680

                            Add

                            N-Desmethylclozapine-d8

                            An internal standard for the quantification of N-desmethylclozapine

                            CAS No. 1189888-77-4

                            Item No. 26027


                            Formulation: A solid
                            Purity: ≥99% deuterated forms (d1-d8)
                            • Norclozapine-d8

                            500 µg

                            $119

                            Add

                            1 mg

                            $189

                            Add

                            cis-Flupenthixol (hydrochloride)

                            A typical antipsychotic

                            CAS No. 51529-01-2

                            Item No. 17634


                            Formulation: A crystalline solid
                            Purity: ≥95%
                            • cis-Flupentixol

                            1 mg

                            $36

                            Add

                            5 mg

                            $103

                            Add

                            10 mg

                            $186

                            Add

                            50 mg

                            $336

                            Add

                            Displaying 1 - 25 of 88 Results
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