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Biochemicals (7)
Small Molecule Modulators (80)
Small Molecule Inhibitors (80)
Acetyltransferases (5)
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Chromatin Reader Interactions (80)
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Displaying 1 - 25 of 80 Results
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(+)-JQ1

An inhibitor of BRD bromodomains

CAS No. 1268524-70-4

Item No. 11187


Formulation: A crystalline solid
Purity: ≥98%

    1 mg

    $31

    Add

    5 mg

    $108

    Add

    10 mg

    $154

    Add

    25 mg

    $270

    Add

    I-BET151

    A BRD2, BRD3, and BRD4 inhibitor

    CAS No. 1300031-49-5

    Item No. 11181


    Formulation: A crystalline solid
    Purity: ≥98%
    • GSK1210151A

    1 mg

    $40

    Add

    5 mg

    $108

    Add

    10 mg

    $197

    Add

    25 mg

    $443

    Add

    I-BET762

    Inhibitor of BET proteins

    CAS No. 1260907-17-2

    Item No. 10676


    Formulation: A crystalline solid
    Purity: ≥98%
    • GSK525762A

    1 mg

    $36

    Add

    5 mg

    $120

    Add

    10 mg

    $219

    Add

    25 mg

    $502

    Add

    OTX015

    A BRD2, BRD3, and BRD4 inhibitor

    CAS No. 202590-98-5

    Item No. 15947


    Formulation: A crystalline solid
    Purity: ≥95%
    • HY-15743
    • (−)-OTX015

    1 mg

    $54

    Add

    5 mg

    $172

    Add

    10 mg

    $238

    Add

    AZD 5153

    A BRD4 inhibitor

    CAS No. 1869912-39-9

    Item No. 20864


    Formulation: A crystalline solid
    Purity: ≥95%

      1 mg

      $42

      Add

      5 mg

      $194

      Add

      10 mg

      $322

      Add

      25 mg

      $653

      Add

      SGC-CBP30

      A potent inhibitor of CREBBP/EP300 bromodomains

      CAS No. 1613695-14-9

      Item No. 14469


      Formulation: A crystalline solid
      Purity: ≥98%

        5 mg

        $121

        Add

        10 mg

        $229

        Add

        50 mg

        $894

        Add

        I-CBP112 (hydrochloride)

        A p300 and CBP inhibitor

        CAS No. 2147701-33-3

        Item No. 14468


        Formulation: A crystalline solid
        Purity: ≥90%

          1 mg

          $49

          Add

          5 mg

          $190

          Add

          10 mg

          $283

          Add

          RVX-208

          A selective BET bromodomain antagonist

          CAS No. 1044870-39-4

          Item No. 16424


          Formulation: A crystalline solid
          Purity: ≥98%
          • Apabetalone
          • RVX-000222

          1 mg

          $49

          Add

          5 mg

          $120

          Add

          10 mg

          $213

          Add

          25 mg

          $445

          Add

          SGC Epigenetic Probe Set

          A library of epigenetic probes from the Structural Genomics Consortium

          Item No. 17748



            1 ea

            $3,003

            Add

            CPI-203

            A bioavailable inhibitor of BET bromodomains

            CAS No. 1446144-04-2

            Item No. 15479


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $63

              Add

              5 mg

              $274

              Add

              10 mg

              $454

              Add

              25 mg

              $678

              Add

              OICR-9429

              A probe for WDR5

              CAS No. 1801787-56-3

              Item No. 16095


              Formulation: A crystalline solid
              Purity: ≥98%

                1 mg

                $63

                Add

                5 mg

                $168

                Add

                10 mg

                $242

                Add

                25 mg

                $527

                Add

                I-BRD9

                A BRD9 bromodomain inhibitor

                CAS No. 1714146-59-4

                Item No. 17749


                Formulation: A crystalline solid
                Purity: ≥98%

                  1 mg

                  $81

                  Add

                  5 mg

                  $159

                  Add

                  10 mg

                  $255

                  Add

                  50 mg

                  $1,064

                  Add

                  UNC3866

                  An inhibitor of CBX7

                  CAS No. 1872382-47-2

                  Item No. 19237


                  Formulation: A crystalline solid
                  Purity: ≥95%

                    1 mg

                    $53

                    Add

                    5 mg

                    $168

                    Add

                    10 mg

                    $306

                    Add

                    25 mg

                    $636

                    Add

                    (+)-JQ1 (free acid)

                    A selective inhibitor of BET bromodomains

                    CAS No. 202592-23-2

                    Item No. 9002910


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      1 mg

                      $60

                      Add

                      5 mg

                      $213

                      Add

                      10 mg

                      $310

                      Add

                      25 mg

                      $702

                      Add

                      PFI-1

                      A BET bromodomain inhibitor

                      CAS No. 1403764-72-6

                      Item No. 11155


                      Formulation: A crystalline solid
                      Purity: ≥98%
                      • PF-06405761

                      1 mg

                      $42

                      Add

                      5 mg

                      $115

                      Add

                      10 mg

                      $183

                      Add

                      25 mg

                      $402

                      Add

                      Bromosporine

                      A non-specific bromodomain inhibitor

                      CAS No. 1619994-69-2

                      Item No. 14119


                      Formulation: A crystalline solid
                      Purity: ≥98%

                        1 mg

                        $41

                        Add

                        5 mg

                        $119

                        Add

                        10 mg

                        $215

                        Add

                        25 mg

                        $389

                        Add

                        ABBV-075

                        A BRD2, BRD4, and BRDT inhibitor

                        CAS No. 1445993-26-9

                        Item No. 21033


                        Formulation: A crystalline solid
                        Purity: ≥98%
                        • Mivebresib

                        500 µg

                        $36

                        Add

                        1 mg

                        $68

                        Add

                        5 mg

                        $186

                        Add

                        10 mg

                        $336

                        Add

                        TP-472

                        A BRD9 inhibitor

                        CAS No. 2079895-62-6

                        Item No. 20030


                        Formulation: A solid
                        Purity: ≥98%

                          1 mg

                          $36

                          Add

                          5 mg

                          $153

                          Add

                          Trotabresib

                          A BRD4 inhibitor

                          CAS No. 1706738-98-8

                          Item No. 36292


                          Formulation: A solid
                          Purity: ≥98%
                          • BMS-986378
                          • CC-90010

                          1 mg

                          $49

                          Add

                          5 mg

                          $182

                          Add

                          10 mg

                          $339

                          Add

                          25 mg

                          $723

                          Add

                          NVS-CECR2-1

                          A potent and selective CECR2 inhibitor

                          CAS No. 1992047-61-6

                          Item No. 18316


                          Formulation: A crystalline solid
                          Purity: ≥95%
                          • NVS-1

                          1 mg

                          $90

                          Add

                          5 mg

                          $241

                          Add

                          10 mg

                          $436

                          Add

                          25 mg

                          $869

                          Add

                          I-BET726

                          A selective inhibitor of BET family proteins

                          CAS No. 1300031-52-0

                          Item No. 16872


                          Formulation: A crystalline solid
                          Purity: ≥98%
                          • GSK1324726A

                          1 mg

                          $46

                          Add

                          5 mg

                          $157

                          Add

                          10 mg

                          $290

                          Add

                          25 mg

                          $662

                          Add

                          BAZ2-ICR

                          A BAZ2A/B bromodomain inhibitor

                          CAS No. 1665195-94-7

                          Item No. 17448


                          Formulation: A crystalline solid
                          Purity: ≥98%

                            1 mg

                            $50

                            Add

                            5 mg

                            $171

                            Add

                            10 mg

                            $266

                            Add

                            25 mg

                            $602

                            Add

                            BI-9564

                            A selective BRD9/7 bromodomain inhibitor

                            CAS No. 1883429-22-8

                            Item No. 17897


                            Formulation: A crystalline solid
                            Purity: ≥98%

                              500 µg

                              $36

                              Add

                              1 mg

                              $61

                              Add

                              10 mg

                              $236

                              Add

                              BI-7273

                              A potent BRD9 bromodomain inhibitor

                              CAS No. 1883429-21-7

                              Item No. 20311


                              Formulation: A crystalline solid
                              Purity: ≥98%

                                1 mg

                                $41

                                Add

                                5 mg

                                $178

                                Add

                                10 mg

                                $312

                                Add

                                25 mg

                                $631

                                Add

                                BMS 986158

                                A BET bromodomain inhibitor

                                CAS No. 1800340-40-2

                                Item No. 27789


                                Formulation: A solid
                                Purity: ≥98%

                                  1 mg

                                  $105

                                  Add

                                  5 mg

                                  $262

                                  Add

                                  10 mg

                                  $418

                                  Add

                                  25 mg

                                  $654

                                  Add

                                  Displaying 1 - 25 of 80 Results
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