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Biochemicals (8)
Small Molecule Modulators (65)
Small Molecule Activators (2)
Small Molecule Inhibitors (65)
Peptidases & Proteases (2)
TNF-α/NF-κB Signaling (1)
Ubiquitin Ligase System (65)

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Cancer (47)
Cell Biology (54)
Endocrinology & Metabolism (3)
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Click Chemistry (2)
Enzyme Activity (2)
Displaying 1 - 25 of 65 Results
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MLN4924

A selective inhibitor of NEDD8-activating enzyme

CAS No. 905579-51-3

Item No. 15217


Formulation: A crystalline solid
Purity: ≥98%
  • Pevonedistat

1 mg

$58

Add

5 mg

$115

Add

10 mg

$201

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proTAME

A prodrug form of TAME

CAS No. 1362911-19-0

Item No. 25835


Formulation: A 10 mg/ml solution in methyl acetate
Purity: ≥90%
  • Pro-N-4-tosyl-L-arginine methyl ester

1 mg

$270

Add

5 mg

$809

Add

Pomalidomide

An inhibitor of cereblon

CAS No. 19171-19-8

Item No. 19877


Formulation: A crystalline solid
Purity: ≥98%
  • CC-4047
  • 3-amino Thalidomide

1 mg

$36

Add

5 mg

$75

Add

10 mg

$129

Add

25 mg

$253

Add

Eeyarestatin 1

An ERAD inhibitor

CAS No. 412960-54-4

Item No. 10012609


Formulation: A crystalline solid
Purity: ≥98%

    5 mg

    $62

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    10 mg

    $116

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    25 mg

    $222

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    MLN7243

    A UAE inhibitor

    CAS No. 1450833-55-2

    Item No. 30108


    Formulation: A crystalline solid
    Purity: ≥98%
    • TAK-243

    1 mg

    $69

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    5 mg

    $313

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    10 mg

    $493

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    PR-619

    A general inhibitor of DUBs

    CAS No. 2645-32-1

    Item No. 16276


    Formulation: A crystalline solid
    Purity: ≥98%
    • 2,6-Diamino-3,5-dithiocyanopyridine
    • DUB Inhibitor V

    5 mg

    $65

    Add

    10 mg

    $115

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    25 mg

    $172

    Add

    50 mg

    $308

    Add

    IMP-1710

    A clickable UCH-L1 inhibitor

    CAS No. 2383117-96-0

    Item No. 31391


    Formulation: A solid
    Purity: ≥98%
    • Click Tag™ IMP-1710

    500 µg

    $107

    Add

    1 mg

    $203

    Add

    5 mg

    $898

    Add

    WP1130

    A deubiquitinase inhibitor

    CAS No. 856243-80-6

    Item No. 15227


    Formulation: A crystalline solid
    Purity: ≥95%
    • Degrasyn

    5 mg

    $75

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    10 mg

    $134

    Add

    25 mg

    $315

    Add

    50 mg

    $589

    Add

    IU1

    A deubiquitinating enzyme inhibitor

    CAS No. 314245-33-5

    Item No. 10617


    Formulation: A crystalline solid
    Purity: ≥98%

      5 mg

      $42

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      10 mg

      $79

      Add

      50 mg

      $322

      Add

      100 mg

      $561

      Add

      Apcin

      An inhibitor of the APC/C

      CAS No. 300815-04-7

      Item No. 17080


      Formulation: A crystalline solid
      Purity: ≥98%

        1 mg

        $32

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        5 mg

        $96

        Add

        10 mg

        $176

        Add

        25 mg

        $319

        Add

        Spautin-1

        An autophagy inhibitor

        CAS No. 1262888-28-7

        Item No. 17769


        Formulation: A crystalline solid
        Purity: ≥95%

          1 mg

          $36

          Add

          5 mg

          $86

          Add

          10 mg

          $153

          Add

          50 mg

          $667

          Add

          b-AP15

          An inhibitor of the deubiquitinases USP14 and UCHL5

          CAS No. 1009817-63-3

          Item No. 11324


          Formulation: A crystalline solid
          Purity: ≥98%

            1 mg

            $41

            Add

            5 mg

            $80

            Add

            10 mg

            $140

            Add

            25 mg

            $293

            Add

            TG2-179-1

            A BAP1 inhibitor

            CAS No. 1135023-19-6

            Item No. 38874


            Formulation: A solid
            Purity: ≥95%

              1 mg

              $90

              Add

              5 mg

              $356

              Add

              10 mg

              $622

              Add

              ML-323

              A selective USP1-UAF1 deubiquitinase complex inhibitor

              CAS No. 1572414-83-5

              Item No. 18010


              Formulation: A crystalline solid
              Purity: ≥98%

                5 mg

                $102

                Add

                10 mg

                $192

                Add

                25 mg

                $423

                Add

                50 mg

                $791

                Add

                JNJ-26854165

                An antagonist of MDM2 action

                CAS No. 881202-45-5

                Item No. 16259


                Formulation: A crystalline solid
                Purity: ≥98%
                • Serdemetan

                1 mg

                $41

                Add

                5 mg

                $134

                Add

                10 mg

                $235

                Add

                25 mg

                $487

                Add

                PRT4165

                An inhibitor of PRC1 ubiquitin ligases

                CAS No. 31083-55-3

                Item No. 19093


                Formulation: A crystalline solid
                Purity: ≥98%
                • NSC 600157

                5 mg

                $63

                Add

                10 mg

                $94

                Add

                25 mg

                $195

                Add

                SMER3

                A selective inhibitor of SCFMET30 ubiquitin E3 ligase

                CAS No. 67200-34-4

                Item No. 15324


                Formulation: A crystalline solid
                Purity: ≥95%
                • SCFMET30 Inhibitor
                • MET30 Antagonist

                5 mg

                $90

                Add

                10 mg

                $132

                Add

                25 mg

                $219

                Add

                50 mg

                $470

                Add

                PYR41

                An irreversible inhibitor of ubiquitin-activating enzyme

                CAS No. 418805-02-4

                Item No. 15226


                Formulation: A crystalline solid
                Purity: ≥95% (mixture of cis and trans isomers)

                  1 mg

                  $29

                  Add

                  5 mg

                  $57

                  Add

                  10 mg

                  $99

                  Add

                  RG-7112

                  An inhibitor of the MDM2-p53 interaction

                  CAS No. 939981-39-2

                  Item No. 25673


                  Formulation: A crystalline solid
                  Purity: ≥98%
                  • RO5045337

                  1 mg

                  $63

                  Add

                  5 mg

                  $257

                  Add

                  10 mg

                  $481

                  Add

                  25 mg

                  $976

                  Add

                  FT709

                  A USP9X inhibitor

                  CAS No. 2413991-74-7

                  Item No. 39971


                  Formulation: A solid
                  Purity: ≥98%

                    1 mg

                    $92

                    Add

                    5 mg

                    $412

                    Add

                    10 mg

                    $731

                    Add

                    ML-364

                    An inhibitor of USP2

                    CAS No. 1991986-30-1

                    Item No. 21774


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      1 mg

                      $37

                      Add

                      5 mg

                      $106

                      Add

                      10 mg

                      $194

                      Add

                      25 mg

                      $436

                      Add

                      SP-141

                      An inhibitor of MDM2

                      CAS No. 1253491-42-7

                      Item No. 17003


                      Formulation: A crystalline solid
                      Purity: ≥98%
                      • AGN-PC-0D106I

                      1 mg

                      $49

                      Add

                      5 mg

                      $130

                      Add

                      10 mg

                      $213

                      Add

                      50 mg

                      $934

                      Add

                      NSC 697923

                      A selective inhibitor of Ubc13

                      CAS No. 343351-67-7

                      Item No. 15346


                      Formulation: A solid
                      Purity: ≥98%

                        1 mg

                        $26

                        Add

                        5 mg

                        $63

                        Add

                        25 mg

                        $183

                        Add

                        LDN-57444

                        An inhibitor of UCH-L1

                        CAS No. 668467-91-2

                        Item No. 15396


                        Formulation: A crystalline solid
                        Purity: ≥95%
                        • Ubiquitin C-terminal Hydrolase L1 Inhibitor
                        • UCH-L1 Inhibitor

                        1 mg

                        $36

                        Add

                        5 mg

                        $86

                        Add

                        10 mg

                        $120

                        Add

                        25 mg

                        $253

                        Add

                        NSC 632839

                        A deubiquitylase and deSUMOylase inhibitor

                        CAS No. 157654-67-6

                        Item No. 16893


                        Formulation: A crystalline solid
                        Purity: ≥98%
                        • F6
                        • Ubiquitin Isopeptidase Inhibitor II

                        1 mg

                        $36

                        Add

                        5 mg

                        $103

                        Add

                        25 mg

                        $253

                        Add

                        50 mg

                        $336

                        Add

                        Displaying 1 - 25 of 65 Results
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