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Antibodies (29)
Assay & Reagent Kits (1)
Biochemicals (9)
Lipids (1)
Natural Products (4)
Proteins (3)
Small Molecule Modulators (37)

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Cancer (32)
Cardiovascular System (2)
Cell Biology (13)
Endocrinology & Metabolism (2)
Epigenetics, Transcription, & Translation (73)
Erasers (27)
Histones/Histone Peptides (27)
Readers (8)
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Displaying 1 - 25 of 73 Results
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Garcinol

A polyisoprenylated benzophenone with diverse biological activities

CAS No. 78824-30-3

Item No. 10566


Formulation: A crystalline solid
Purity: ≥95%
  • Camboginol
  • Guttiferone F

5 mg

$47

Add

10 mg

$74

Add

25 mg

$174

Add

50 mg

$301

Add

Delphinidin (chloride)

Natural vasorelaxant and inhibitor of EGFRs and HATs

CAS No. 528-53-0

Item No. 11012


Formulation: A crystalline solid
Purity: ≥97%
  • Ephdine

1 mg

$41

Add

5 mg

$167

Add

10 mg

$312

Add

HAT Inhibitor Screening Assay Kit

A fast, fluorescence-based method for evaluating PCAF HAT inhibitors

Item No. 10006515


  • Histone Acetyltransferase

96 wells

$383

Add

A-485

A p300/CBP inhibitor

CAS No. 1889279-16-6

Item No. 24119


Formulation: A crystalline solid
Purity: ≥98% (mixture of isomers)

    1 mg

    $54

    Add

    5 mg

    $209

    Add

    10 mg

    $367

    Add

    25 mg

    $783

    Add

    PCAF Histone Acetyltransferase (human, recombinant)

    Active, pure human recombinant enzyme

    Item No. 10009115


    Formulation: 50 mM HEPES, pH 8, with 150 mM NaCl, 1 mM EDTA, and 20% glycerol
    Purity: ≥80% estimated by SDS-PAGE
    • HAT
    • p300/(CREB binding protein) Associated Factor

    100 µg

    $541

    Add

    4-pentynoyl-Coenzyme A (trifluoroacetate salt)

    A protein acetylation probe

    Item No. 10547


    Formulation: A lyophilized powder
    Purity: ≥95%
    • Click Tag™ 4-pentynoyl-CoA

    500 µg

    $83

    Add

    1 mg

    $158

    Add

    5 mg

    $660

    Add

    10 mg

    $1,073

    Add

    Anacardic Acid

    A histone acetyltransferase inhibitor

    CAS No. 16611-84-0

    Item No. 13144


    Formulation: A crystalline solid
    Purity: ≥98%
    • 6-pentadecyl Salicylic Acid

    1 mg

    $29

    Add

    5 mg

    $53

    Add

    10 mg

    $94

    Add

    C646

    An inhibitor of the HAT p300

    CAS No. 328968-36-1

    Item No. 10549


    Formulation: A crystalline solid
    Purity: ≥98% (mixture of isomers)

      1 mg

      $41

      Add

      5 mg

      $116

      Add

      10 mg

      $189

      Add

      Butyrolactone 3

      A HAT inhibitor

      CAS No. 778649-18-6

      Item No. 12095


      Formulation: A crystalline solid
      Purity: ≥95%

        1 mg

        $60

        Add

        5 mg

        $171

        Add

        Gcn5 (human, recombinant)

        Active, pure human recombinant enzyme

        Item No. 10782


        Formulation: 50 mM Tris, pH 8.0, with 150 mM sodium chloride and 20% glycerol
        Purity: ≥50% estimated by SDS-PAGE
        • General control of amino acid synthesis protein 5-like 2
        • KAT2A
        • Lysine acetyltransferase 2A
        • STAF97

        100 µg

        $476

        Add

        TIP60 (human, recombinant)

        Active, human recombinant enzyme

        Item No. 10783


        Formulation: 50 mM Tris-HCl, pH 7.5, with 300 mM sodium chloride and 10% glycerol
        Purity: ≥50%
        • cPLA(2) Interacting Protein
        • Esa1
        • Histone acetyltransferase KAT5
        • HIV-1 Tat Interacting Protein 60 kDa
        • Hs.6364
        • HTATIP
        • KAT5
        • PLIP

        100 µg

        $543

        Add

        CPTH6 (hydrobromide)

        A Gcn5 and pCAF HAT inhibitor

        CAS No. 2321332-57-2

        Item No. 19828


        Formulation: A crystalline solid
        Purity: ≥98%

          1 mg

          $41

          Add

          5 mg

          $178

          Add

          10 mg

          $312

          Add

          Histone H3 Peptide Substrate (1-21) (trifluoroacetate salt)

          Target substrate for several histone modifying enzymes

          Item No. 10877


          Formulation: A lyophilized peptide
          Purity: ≥95%
          • H3 Peptide

          1 mg

          $206

          Add

          Acetyl Lysine Monoclonal Antibody (Clone 7F8)

          For immunochemical detection of acetyl lysine

          Item No. 10010567


          Immunogen: Acetylated KLH
          Host: Mouse
          Isotype: IgG1
          Applications: ELISA, ICC, WB

          1 ea (100 µg)

          $401

          Add

          CPTH2 (hydrochloride)

          A HAT inhibitor

          CAS No. 2108899-91-6

          Item No. 12086


          Formulation: A crystalline solid
          Purity: ≥95%

            5 mg

            $107

            Add

            10 mg

            $141

            Add

            CTPB

            A selective activator of p300 HAT

            CAS No. 586976-24-1

            Item No. 19570


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $54

              Add

              5 mg

              $172

              Add

              CCS-1477

              A p300 and CBP inhibitor

              CAS No. 2222941-37-7

              Item No. 34546


              Formulation: A solid
              Purity: ≥98%
              • CBP-IN-1

              1 mg

              $54

              Add

              5 mg

              $250

              Add

              10 mg

              $367

              Add

              25 mg

              $717

              Add

              Histone H3K23Ac Monoclonal Antibody (RM169)

              For immunochemical detection of H3K23Ac

              Item No. 32161


              Immunogen: Peptide corresponding to H3K23Ac
              Host: Rabbit
              Isotype: IgG
              Applications: ELISA, ICC, multiplex-based assays, WB

              100 µg

              $500

              Add

              MG149

              A HAT inhibitor

              CAS No. 1243583-85-8

              Item No. 22135


              Formulation: A crystalline solid
              Purity: ≥98%

                1 mg

                $48

                Add

                5 mg

                $184

                Add

                10 mg

                $319

                Add

                25 mg

                $627

                Add

                GSK4027

                A PCAF/GCN5 bromodomain inhibitor

                CAS No. 2079896-25-4

                Item No. 23421


                Formulation: A crystalline solid
                Purity: ≥95%

                  1 mg

                  $49

                  Add

                  5 mg

                  $154

                  Add

                  10 mg

                  $283

                  Add

                  L-Moses (hydrochloride)

                  A PCAF bromodomain inhibitor

                  CAS No. 2922480-38-2

                  Item No. 21288


                  Formulation: A crystalline solid
                  Purity: ≥98%
                  • L-45

                  1 mg

                  $41

                  Add

                  5 mg

                  $178

                  Add

                  10 mg

                  $312

                  Add

                  25 mg

                  $680

                  Add

                  CAY10669

                  An inhibitor of PCAF

                  CAS No. 1243583-88-1

                  Item No. 10974


                  Formulation: A crystalline solid
                  Purity: ≥98%

                    1 mg

                    $90

                    Add

                    5 mg

                    $392

                    Add

                    10 mg

                    $696

                    Add

                    L002

                    A p300 acetyltransferase inhibitor

                    CAS No. 321695-57-2

                    Item No. 17778


                    Formulation: A crystalline solid
                    Purity: ≥98%
                    • p300/CBP Inhibitor VI
                    • NSC 764414

                    5 mg

                    $90

                    Add

                    10 mg

                    $132

                    Add

                    25 mg

                    $306

                    Add

                    50 mg

                    $567

                    Add

                    WM-1119

                    An inhibitor of KAT6A

                    CAS No. 2055397-28-7

                    Item No. 30509


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      5 mg

                      $121

                      Add

                      10 mg

                      $215

                      Add

                      25 mg

                      $448

                      Add

                      50 mg

                      $713

                      Add

                      PF-07248144

                      A KAT6A and KAT6B inhibitor

                      CAS No. 2569008-99-5

                      Item No. 43955


                      Formulation: A solid
                      Purity: ≥98%

                        1 mg

                        $72

                        Add

                        5 mg

                        $323

                        Add

                        10 mg

                        $501

                        Add

                        25 mg

                        $984

                        Add

                        Displaying 1 - 25 of 73 Results
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