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Product TypeClear Filters

Analytical Chemistry (5)
Biochemicals (38)
Small Molecule Modulators (37)

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Cancer (38)
Angiogenesis (3)
Cell Cycle (2)
Cell Death (10)
Cell Migration & Metastasis (3)
Cell Signaling (38)
Abl family & Bcr-Abl Signaling (38)
Aurora Signaling (3)
ERK/MAPK Signaling (4)
Growth Factor Receptor Signaling (16)
Hedgehog Signaling (1)
JAK/STAT Signaling (2)
PI3K/Akt/mTOR Signaling (1)
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Mass Spectrometry (5)
Displaying 1 - 25 of 38 Results
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Imatinib (mesylate)

An inhibitor of c-Abl, Bcr-Abl, PDGFR, and c-Kit

CAS No. 220127-57-1

Item No. 13139


Formulation: A crystalline solid
Purity: ≥98%
  • CGP57148B
  • STI-571

25 mg

$38

Add

50 mg

$72

Add

100 mg

$97

Add

500 mg

$449

Add

Dasatinib

An inhibitor of Abl and Src

CAS No. 302962-49-8

Item No. 11498


Formulation: A crystalline solid
Purity: ≥98%
  • BMS 354825
  • Sprycel

10 mg

$36

Add

50 mg

$53

Add

100 mg

$88

Add

250 mg

$176

Add

Nilotinib

A Bcr-Abl inhibitor

CAS No. 641571-10-0

Item No. 10010422


Formulation: A crystalline solid
Purity: ≥95%
  • AMN107

5 mg

$28

Add

10 mg

$41

Add

25 mg

$81

Add

50 mg

$130

Add

Ponatinib

An inhibitor of native and mutant Bcr-Abl

CAS No. 943319-70-8

Item No. 11494


Formulation: A crystalline solid
Purity: ≥98%
  • AP 24534

1 mg

$32

Add

5 mg

$86

Add

10 mg

$109

Add

Bosutinib

An inhibitor of Src and Abl kinases

CAS No. 380843-75-4

Item No. 12030


Formulation: A crystalline solid
Purity: ≥98%
  • SKI 606

5 mg

$49

Add

10 mg

$73

Add

50 mg

$283

Add

100 mg

$469

Add

Saracatinib

A dual inhibitor of c-Src and Abl

CAS No. 379231-04-6

Item No. 11497


Formulation: A crystalline solid
Purity: ≥90%
  • AZD 0530

5 mg

$35

Add

10 mg

$59

Add

25 mg

$119

Add

50 mg

$168

Add

PD 166326

An inhibitor of c-src and certain receptor tyrosine kinases, including c-abl

CAS No. 185039-91-2

Item No. 9000988


Formulation: A crystalline solid
Purity: ≥95%

    1 mg

    $108

    Add

    5 mg

    $481

    Add

    10 mg

    $856

    Add

    AT-9283

    A broad spectrum kinase inhibitor

    CAS No. 896466-04-9

    Item No. 11496


    Formulation: A crystalline solid
    Purity: ≥98%

      5 mg

      $98

      Add

      10 mg

      $176

      Add

      25 mg

      $318

      Add

      50 mg

      $490

      Add

      Nilotinib-d6

      An internal standard for the quantification of nilotinib

      CAS No. 1268356-17-7

      Item No. 19280


      Formulation: A solid
      Purity: ≥99% deuterated forms (d1-d6)

        1 mg

        $569

        Add

        N-desmethyl Imatinib

        A major active metabolite of imatinib

        CAS No. 404844-02-6

        Item No. 16947


        Formulation: A lyophilized solid
        Purity: ≥95%
        • N-desmethyl Gleevec
        • STI-509-00

        500 µg

        $42

        Add

        1 mg

        $79

        Add

        5 mg

        $303

        Add

        10 mg

        $561

        Add

        AST-487

        A multi-kinase inhibitor

        CAS No. 630124-46-8

        Item No. 19477


        Formulation: A crystalline solid
        Purity: ≥98%
        • NVP-AST-487

        1 mg

        $37

        Add

        5 mg

        $124

        Add

        10 mg

        $229

        Add

        25 mg

        $523

        Add

        Asciminib

        An allosteric inhibitor of Abl1

        CAS No. 1492952-76-7

        Item No. 26126


        Formulation: A crystalline solid
        Purity: ≥95%
        • ABL001

        1 mg

        $69

        Add

        5 mg

        $280

        Add

        10 mg

        $525

        Add

        ALW-II-41-27

        A multi-kinase inhibitor

        CAS No. 1186206-79-0

        Item No. 25275


        Formulation: A crystalline solid
        Purity: ≥95%

          1 mg

          $69

          Add

          5 mg

          $297

          Add

          10 mg

          $525

          Add

          Imatinib-d3

          An internal standard for the quantification of imatinib

          CAS No. 1134803-18-1

          Item No. 18257


          Formulation: A solid
          Purity: ≥99% deuterated forms (d1-d3)
          • Genfatinib-d3

          500 µg

          $112

          Add

          1 mg

          $202

          Add

          GZD-824

          A Bcr/Abl inhibitor

          CAS No. 1257628-77-5

          Item No. 21508


          Formulation: A crystalline solid
          Purity: ≥98%
          • HQP1351
          • Olverembatinib

          1 mg

          $36

          Add

          5 mg

          $153

          Add

          10 mg

          $268

          Add

          25 mg

          $502

          Add

          Ponatinib-d8

          An internal standard for the quantification of ponatinib

          CAS No. 1562993-37-6

          Item No. 28905


          Formulation: A solid
          Purity: ≥99% deuterated forms (d1-d8)

            1 mg

            $390

            Add

            Radotinib

            A selective Bcr-Abl tyrosine kinase inhibitor

            CAS No. 926037-48-1

            Item No. 19923


            Formulation: A crystalline solid
            Purity: ≥98%
            • IY-5511

            1 mg

            $36

            Add

            5 mg

            $120

            Add

            10 mg

            $203

            Add

            25 mg

            $378

            Add

            MGCD-265

            A c-Met and VEGFR2 inhibitor

            CAS No. 875337-44-3

            Item No. 20097


            Formulation: A crystalline solid
            Purity: ≥98%

              1 mg

              $48

              Add

              5 mg

              $190

              Add

              10 mg

              $355

              Add

              25 mg

              $708

              Add

              Bafetinib

              A Bcr-Abl inhibitor

              CAS No. 859212-16-1

              Item No. 19169


              Formulation: A crystalline solid
              Purity: ≥95%
              • INNO-406
              • NS-187

              1 mg

              $49

              Add

              5 mg

              $130

              Add

              10 mg

              $236

              Add

              KW 2449

              A multi-kinase inhibitor

              CAS No. 1000669-72-6

              Item No. 22207


              Formulation: A crystalline solid
              Purity: ≥98%

                5 mg

                $36

                Add

                10 mg

                $64

                Add

                25 mg

                $150

                Add

                50 mg

                $264

                Add

                Rebastinib

                An orally bioavailable tyrosine kinase inhibitor

                CAS No. 1020172-07-9

                Item No. 21465


                Formulation: A crystalline solid
                Purity: ≥98%
                • DCC-2036

                1 mg

                $52

                Add

                5 mg

                $227

                Add

                10 mg

                $396

                Add

                25 mg

                $867

                Add

                NG 25 (hydrochloride hydrate)

                An inhibitor of MAP4K2 and TAK1

                Item No. 27579


                Formulation: A solid
                Purity: ≥98%

                  1 mg

                  $60

                  Add

                  5 mg

                  $185

                  Add

                  10 mg

                  $339

                  Add

                  XL228

                  A tyrosine kinase inhibitor

                  CAS No. 898280-07-4

                  Item No. 21506


                  Formulation: A crystalline solid
                  Purity: ≥98%

                    5 mg

                    $90

                    Add

                    10 mg

                    $158

                    Add

                    25 mg

                    $354

                    Add

                    50 mg

                    $634

                    Add

                    Ponatinib (hydrochloride)

                    An inhibitor of native and mutant Bcr-Abl

                    CAS No. 1114544-31-8

                    Item No. 35778


                    Formulation: A solid
                    Purity: ≥98%
                    • AP 24534

                    50 mg

                    $46

                    Add

                    100 mg

                    $85

                    Add

                    500 mg

                    $357

                    Add

                    1 g

                    $579

                    Add

                    Bosutinib-d8

                    An internal standard for the quantification of bosutinib

                    CAS No. 2733145-45-2

                    Item No. 25460


                    Formulation: A solid
                    Purity: ≥99% deuterated forms (d1-d8)

                      500 µg

                      $160

                      Add

                      1 mg

                      $304

                      Add

                      Displaying 1 - 25 of 38 Results
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