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Analytical Chemistry (1)
Biochemicals (18)
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Small Molecule Modulators (18)

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Cancer (19)
Autophagy (1)
Cell Death (1)
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ALK (Activin-like Kinase) Signaling (19)
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JAK/STAT Signaling (1)
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Mass Spectrometry (1)
Displaying 1 - 19 of 19 Results
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SB-431542 (hydrate)

Inhibitor of receptors ALK4, ALK5, and ALK7

Item No. 13031


Formulation: A crystalline solid
Purity: ≥98%

    1 mg

    $45

    Add

    5 mg

    $124

    Add

    10 mg

    $180

    Add

    25 mg

    $394

    Add

    A 83-01

    A TGF-β type I receptor inhibitor

    CAS No. 909910-43-6

    Item No. 9001799


    Formulation: A crystalline solid
    Purity: ≥95%

      1 mg

      $36

      Add

      5 mg

      $71

      Add

      10 mg

      $124

      Add

      25 mg

      $264

      Add

      LY364947

      Inhibitor of TGF-β type-1 receptors

      CAS No. 396129-53-6

      Item No. 13341


      Formulation: A crystalline solid
      Purity: ≥98%
      • HTS 466284
      • TGF-β RI Kinase Inhibitor

      5 mg

      $74

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      10 mg

      $104

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      25 mg

      $240

      Add

      50 mg

      $369

      Add

      LDN-193189

      An inhibitor of BMP receptors ALK1, ALK2, ALK3, and ALK6

      CAS No. 1062368-24-4

      Item No. 11802


      Formulation: A crystalline solid
      Purity: ≥95%
      • DM-3189

      1 mg

      $33

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      5 mg

      $92

      Add

      10 mg

      $116

      Add

      25 mg

      $207

      Add

      DMH1

      A potent ALK2 inhibitor

      CAS No. 1206711-16-1

      Item No. 16679


      Formulation: A crystalline solid
      Purity: ≥98%
      • BMP Inhibitor II
      • DorsoMorphin Homolog 1
      • VU036482

      1 mg

      $44

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      5 mg

      $121

      Add

      10 mg

      $220

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      50 mg

      $660

      Add

      LDN-193189 (hydrochloride)

      An inhibitor of BMP receptors ALK1, ALK2, ALK3, and ALK6

      CAS No. 1435934-00-1

      Item No. 19396


      Formulation: A crystalline solid
      Purity: ≥98%
      • DM-3189

      1 mg

      $30

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      5 mg

      $68

      Add

      10 mg

      $119

      Add

      25 mg

      $224

      Add

      Dorsomorphin (hydrochloride)

      A potent, reversible AMPK inhibitor

      CAS No. 1219168-18-9

      Item No. 21207


      Formulation: A crystalline solid
      Purity: ≥98%
      • BML-275
      • Compound C
      • CpdC

      1 mg

      $36

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      5 mg

      $128

      Add

      10 mg

      $169

      Add

      25 mg

      $378

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      BLU-782

      An ALK2R206H inhibitor

      CAS No. 2141955-96-4

      Item No. 35490


      Formulation: A solid
      Purity: ≥95%
      • Activin Receptor-like Kinase 2 Inhibitor 1
      • ALK2-IN-1
      • Fidrisertib

      1 mg

      $62

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      5 mg

      $244

      Add

      10 mg

      $395

      Add

      25 mg

      $909

      Add

      EW-7197

      A potent inhibitor of ALK5

      CAS No. 1352608-82-2

      Item No. 19231


      Formulation: A crystalline solid
      Purity: ≥98%
      • Vactosertib

      1 mg

      $134

      Add

      5 mg

      $253

      Add

      10 mg

      $399

      Add

      K02288

      A BMP signaling inhibitor

      CAS No. 1431985-92-0

      Item No. 16678


      Formulation: A crystalline solid
      Purity: ≥98%

        1 mg

        $41

        Add

        5 mg

        $148

        Add

        10 mg

        $255

        Add

        50 mg

        $873

        Add

        Ceritinib-d7

        An internal standard for the quantification of ceritinib

        CAS No. 1632484-77-5

        Item No. 28768


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d7)
        • LDK 378-d7

        1 mg

        $468

        Add

        LY3200882

        An inhibitor of TGF-βRI

        CAS No. 1898283-02-7

        Item No. 25276


        Formulation: A crystalline solid
        Purity: ≥95%

          1 mg

          $41

          Add

          5 mg

          $178

          Add

          10 mg

          $312

          Add

          25 mg

          $680

          Add

          SM-16

          An inhibitor of ALK5

          CAS No. 614749-78-9

          Item No. 34061


          Formulation: A solid
          Purity: ≥98%

            1 mg

            $41

            Add

            5 mg

            $186

            Add

            10 mg

            $351

            Add

            25 mg

            $728

            Add

            TPX-0005

            A multi-kinase inhibitor

            CAS No. 1802220-02-5

            Item No. 23397


            Formulation: A crystalline solid
            Purity: ≥98%
            • Repotrectinib

            1 mg

            $36

            Add

            5 mg

            $153

            Add

            10 mg

            $268

            Add

            25 mg

            $587

            Add

            SB-505124 (hydrochloride)

            An ALK5 and ALK4 inhibitor

            CAS No. 356559-13-2

            Item No. 42056


            Formulation: A solid
            Purity: ≥98%
            • TGF-β Receptor Type I Kinase Inhibitor III
            • TGF-β RI Kinase Inhibitor III

            1 mg

            $28

            Add

            5 mg

            $104

            Add

            10 mg

            $165

            Add

            25 mg

            $379

            Add

            RIPK2 Inhibitor OD36 (hydrochloride)

            A RIPK2 inhibitor

            CAS No. 2387510-88-3

            Item No. 42171


            Formulation: A solid
            Purity: ≥98%
            • OD36
            • Receptor-interacting Serine/Threonine Kinase 2 Inhibitor OD36

            1 mg

            $43

            Add

            5 mg

            $183

            Add

            10 mg

            $323

            Add

            25 mg

            $537

            Add

            BMS 986260

            An ALK5 inhibitor

            CAS No. 2001559-19-7

            Item No. 42042


            Formulation: A solid
            Purity: ≥98%

              5 mg

              $102

              Add

              10 mg

              $193

              Add

              50 mg

              $557

              Add

              100 mg

              $1,012

              Add

              M4K2234

              An ALK1 and ALK2 inhibitor

              CAS No. 2421141-51-5

              Item No. 41169


              Formulation: A solid
              Purity: ≥98%

                1 mg

                $50

                Add

                5 mg

                $161

                Add

                10 mg

                $248

                Add

                25 mg

                $495

                Add

                ALK2 Extracellular Domain (human, recombinant)

                Host: Insect cells • AA: 21-124 • Tag: C-terminal His • MW: 12.8 kDa

                Item No. 44183


                Formulation: Sterile 20 mM Tris, pH 7.4, with 500 mM sodium chloride and 10% glycerol
                Purity: ≥93% estimated by SDS-PAGE
                • Activin Receptor-like Kinase 2
                • Activin Receptor Type I
                • ACTR-I
                • ACVR1
                • Serine/threonine-protein Kinase Receptor R1
                • TGF-β Superfamily Receptor Type I
                • TSR-I

                100 µg

                $298

                Add

                1 mg

                $1,937

                Add

                Displaying 1 - 19 of 19 Results
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