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Environmental Toxicology (1)
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Small Molecule Modulators (24)

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Displaying 1 - 25 of 28 Results
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Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate)

A metabolite of estrogen

Item No. 16156


Formulation: A crystalline solid
Purity: ≥95%
  • E217G
  • β-Estradiol 17-(β-D-Glucuronide)
  • 17β-Estradiol 17-(β-D-Glucuronide)
  • 17β-Oestradiol 17-(β-D-Glucuronide)

5 mg

$81

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10 mg

$152

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25 mg

$279

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50 mg

$436

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Estradiol 3-(β-D-Glucuronide) (sodium salt)

An isomer of estradiol-(β-D-glucuronide)

CAS No. 14982-12-8

Item No. 16155


Formulation: A crystalline solid
Purity: ≥95%
  • E23G
  • β-Estradiol 3-(β-D-Glucuronide)
  • 17β-Estradiol 3-(β-D-Glucuronide)
  • 17β-Oestradiol 3-(β-D-Glucuronide)

1 mg

$75

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5 mg

$300

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10 mg

$524

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25 mg

$1,029

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Multidrug Resistance Assay Kit (Calcein AM)

A convenient tool for studying MDR protein modulators

Item No. 600370


  • MDR

1,000 tests

$290

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Elacridar

An inhibitor of MRP-1 and BCRP

CAS No. 143664-11-3

Item No. 18128


Formulation: A crystalline solid
Purity: ≥98%
  • GF120918
  • GG918
  • GW0918

1 mg

$36

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5 mg

$77

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10 mg

$120

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50 mg

$387

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Fumitremorgin C

Inhibitor of BCRP multidrug transporter

CAS No. 118974-02-0

Item No. 11030


Formulation: A crystalline solid
Purity: ≥98%
  • Tryptoquivaline

250 µg

$234

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1 mg

$602

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Roquefortine C

A mycotoxin

CAS No. 58735-64-1

Item No. 15376


Formulation: A solid
Purity: ≥98%
  • NSC 292134

500 µg

$189

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1 mg

$336

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Silychristin

A flavonolignan with diverse biological activities

CAS No. 33889-69-9

Item No. 34658


Formulation: A solid
Purity: ≥98%
  • Silychristin A
  • (+)-Silychristin

5 mg

$196

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10 mg

$351

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25 mg

$680

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Oroxylin A

A flavonoid with diverse biological activities

CAS No. 480-11-5

Item No. 27363


Formulation: A solid
Purity: ≥98%
  • 6-Methoxybaicalein

1 mg

$61

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5 mg

$213

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10 mg

$303

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25 mg

$605

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Etonogestrel

A progesterone and androgen receptor antagonist and an active metabolite of desogestrel

CAS No. 54048-10-1

Item No. 21062


Formulation: A crystalline solid
Purity: ≥98%
  • ORG 3236
  • 3-keto Desogestrel
  • 3-oxo Desogestrel

1 mg

$36

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5 mg

$103

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10 mg

$153

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25 mg

$336

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Atorvastatin lactone

An active metabolite of atorvastatin

CAS No. 125995-03-1

Item No. 20951


Formulation: A crystalline solid
Purity: ≥95%

    1 mg

    $36

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    5 mg

    $128

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    10 mg

    $186

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    25 mg

    $294

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    BMS 986020

    An LPA1 receptor antagonist

    CAS No. 1257213-50-5

    Item No. 22049


    Formulation: A crystalline solid
    Purity: ≥95%
    • AM-000152

    500 µg

    $36

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    1 mg

    $68

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    5 mg

    $169

    Add

    1-Palmitoleoyl glycerol

    A monoacylglycerol

    CAS No. 37515-61-0

    Item No. 25697


    Formulation: A low melting solid
    Purity: ≥98%
    • 1-Monopalmitoleoyl-rac-glycerol

    25 mg

    $75

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    50 mg

    $134

    Add

    100 mg

    $252

    Add

    250 mg

    $589

    Add

    6’,7’-Epoxybergamottin

    A potent CYP3A4 inhibitor from grapefruit

    CAS No. 206978-14-5

    Item No. 19760


    Formulation: A crystalline solid
    Purity: ≥95%
    • Epoxybergamottin

    1 mg

    $51

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    5 mg

    $191

    Add

    10 mg

    $355

    Add

    25 mg

    $758

    Add

    ONT-093

    A P-glycoprotein inhibitor

    CAS No. 216227-54-2

    Item No. 28758


    Formulation: A crystalline solid
    Purity: ≥98%
    • OC 144093

    1 mg

    $103

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    5 mg

    $454

    Add

    10 mg

    $753

    Add

    S-(2,4-Dinitrophenyl)-Glutathione

    A substrate for glutathione-S-transferase

    CAS No. 26289-39-4

    Item No. 24660


    Formulation: A solid
    Purity: ≥98%
    • Dinitrophenyl-S-Glutathione
    • GS-DNP
    • NSC 131112
    • NSC 638615

    1 mg

    $54

    Add

    5 mg

    $238

    Add

    10 mg

    $392

    Add

    Hypophyllanthin

    A P-glycoprotein inhibitor

    CAS No. 33676-00-5

    Item No. 11715


    Formulation: A crystalline solid
    Purity: ≥98%
    • NSC 619044

    1 mg

    $69

    Add

    5 mg

    $297

    Add

    10 mg

    $493

    Add

    25 mg

    $1,062

    Add

    Bromosulfalein

    An OATP and MDR2 substrate and inhibitor

    CAS No. 71-67-0

    Item No. 21058


    Formulation: A crystalline solid
    Purity: ≥95%
    • Bromosulfophthalein
    • Bromosulphalein
    • Sulfobromophthalein
    • Sulphobromophthalein

    1 g

    $35

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    5 g

    $94

    Add

    10 g

    $169

    Add

    Chrysin 7-Glucuronide

    A flavonoid glucuronide with diverse biological activities and an active metabolite of chrysin

    CAS No. 35775-49-6

    Item No. 35034


    Formulation: A solid
    Purity: ≥98%
    • Chrysin 7-O-Glucuronide
    • Chrysin 7-O-β-D-Glucuronide

    1 mg

    $69

    Add

    5 mg

    $248

    Add

    10 mg

    $461

    Add

    25 mg

    $1,062

    Add

    CP 100,356 (hydrochloride)

    A P-glycoprotein inhibitor

    CAS No. 142715-48-8

    Item No. 32853


    Formulation: A solid
    Purity: ≥98%

      1 mg

      $69

      Add

      5 mg

      $149

      Add

      10 mg

      $256

      Add

      Bacoside A3

      An antioxidant and P-gp inhibitor

      CAS No. 157408-08-7

      Item No. 11824


      Formulation: A solid
      Purity: ≥98%
      • Bacopa Pgp

      5 mg

      $636

      Add

      Sciadopitysin

      A biflavonoid with diverse biological activities

      CAS No. 521-34-6

      Item No. 27900


      Formulation: A solid
      Purity: ≥98%
      • NSC 45108

      5 mg

      $134

      Add

      10 mg

      $253

      Add

      25 mg

      $565

      Add

      50 mg

      $926

      Add

      Desogestrel

      A synthetic progestogen

      CAS No. 54024-22-5

      Item No. 23651


      Formulation: A solid
      Purity: ≥95%
      • ORG 2969

      5 mg

      $68

      Add

      10 mg

      $118

      Add

      25 mg

      $179

      Add

      Robinetin

      A flavonol with diverse biological activities

      CAS No. 490-31-3

      Item No. 35272


      Formulation: A solid
      Purity: ≥98%
      • NSC 407331
      • NSC 656274
      • 3,7,3′,4′,5′-Pentahydroxyflavone

      5 mg

      $49

      Add

      10 mg

      $87

      Add

      25 mg

      $194

      Add

      50 mg

      $315

      Add

      Benzoylaconine

      An aconitine-type diterpenoid alkaloid

      CAS No. 466-24-0

      Item No. 25687


      Formulation: A crystalline solid
      Purity: ≥95%

        1 mg

        $49

        Add

        5 mg

        $223

        Add

        10 mg

        $423

        Add

        25 mg

        $820

        Add

        Atorvastatin lactone-d5

        An internal standard for the quantification of atorvastatin lactone

        Item No. 35171


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d5)

          500 µg

          $174

          Add

          1 mg

          $329

          Add

          Displaying 1 - 25 of 28 Results
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