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Displaying 1 - 25 of 374 Results
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Calcitriol

An agonist of the vitamin D3 receptor and active metabolite of vitamin D3

CAS No. 32222-06-3

Item No. 71820


Formulation: A crystalline solid
Purity: ≥97%
  • 1,25-dihydroxy Cholecalciferol
  • 1α,25-dihydroxy Cholecalciferol
  • 1,25-dihydroxy Vitamin D3
  • 1α,25-dihydroxy Vitamin D3

1 mg

$98

Add

5 mg

$368

Add

10 mg

$686

Add

4-hydroxy Diclofenac

An active metabolite of diclofenac

CAS No. 64118-84-9

Item No. 10008518


Formulation: A crystalline solid
Purity: ≥95%

    1 mg

    $138

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    5 mg

    $516

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    10 mg

    $895

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    α-hydroxy Midazolam

    A CYP3A metabolite of midazolam

    CAS No. 59468-90-5

    Item No. 10385


    Formulation: A crystalline solid
    Purity: ≥95%
    • 1’-hydroxy Midazolam
    • Ro 21-6347

    1 mg

    $160

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    5 mg

    $240

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    (E/Z)-4-hydroxy Tamoxifen

    A mixture of (E)-4-hydroxy tamoxifen and (Z)-4-hydroxy tamoxifen

    CAS No. 68392-35-8

    Item No. 17308


    Formulation: A crystalline solid
    Purity: ≥98% (mixture of isomers)
    • Afimoxifene
    • 4-OHT

    5 mg

    $42

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    10 mg

    $80

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    25 mg

    $189

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    50 mg

    $293

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    (Z)-4-hydroxy Tamoxifen

    An active metabolite of tamoxifen

    CAS No. 68047-06-3

    Item No. 14854


    Formulation: A crystalline solid
    Purity: ≥98%
    • ICI 79280
    • trans-4-hydroxy Tamoxifen

    1 mg

    $43

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    5 mg

    $161

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    10 mg

    $215

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    25 mg

    $483

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    (S)-Mephenytoin

    A substrate of CYP2C19

    CAS No. 70989-04-7

    Item No. 11913


    Formulation: A crystalline solid
    Purity: ≥98%
    • (+)-Mephenytoin
    • (S)-5-ethyl-3-methyl-5-Phenylhydantoin

    1 mg

    $47

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    5 mg

    $116

    Add

    10 mg

    $208

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    25 mg

    $462

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    Paclitaxel

    A potent mitotic inhibitor

    CAS No. 33069-62-4

    Item No. 10461


    Formulation: A crystalline solid
    Purity: ≥98%
    • NSC 125973

    5 mg

    $39

    Add

    25 mg

    $106

    Add

    50 mg

    $193

    Add

    100 mg

    $308

    Add

    6α-hydroxy Paclitaxel

    A metabolite of paclitaxel

    CAS No. 153212-75-0

    Item No. 10009027


    Formulation: A crystalline solid
    Purity: ≥95%
    • 6α-hydroxy Taxol

    500 µg

    $275

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    1 mg

    $385

    Add

    5 mg

    $1,788

    Add

    CH 223191

    A potent antagonist of AhR

    CAS No. 301326-22-7

    Item No. 16154


    Formulation: A crystalline solid
    Purity: ≥95%

      5 mg

      $76

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      10 mg

      $145

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      25 mg

      $343

      Add

      50 mg

      $608

      Add

      (±)17(18)-EpETE

      An active metabolite of eicosapentaenoic acid and an S1P1 agonist

      Item No. 50861


      Formulation: A 100 µg/ml solution in ethanol
      Purity: ≥90%
      • (±)17(18)-EEQ
      • (±)17(18)-epoxy-5(Z),8(Z)
      • (±)17(18)-epoxy-all-cis-5,8,11,14-Eicosatetraenoic Acid
      • (±)17(18)-Epoxyeicosatetraenoic Acid
      • 11(Z),14(Z)-ETE
      • FA 20:5;O

      25 µg

      $69

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      50 µg

      $130

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      100 µg

      $233

      Add

      500 µg

      $955

      Add

      Gemfibrozil 1-O-β-Glucuronide

      A major metabolite of gemfibrozil

      CAS No. 91683-38-4

      Item No. 19080


      Formulation: A solid
      Purity: ≥85%

        500 µg

        $267

        Add

        1 mg

        $505

        Add

        25-hydroxy Vitamin D3

        A vitamin D intermediate

        CAS No. 19356-17-3

        Item No. 9000683


        Formulation: A crystalline solid
        Purity: ≥98%
        • 25-hydroxy Cholecalciferol
        • RO 8-8892
        • U 32070E

        1 mg

        $94

        Add

        5 mg

        $328

        Add

        10 mg

        $561

        Add

        Paclitaxel-d5

        An internal standard for the quantification of paclitaxel

        CAS No. 1129540-33-5

        Item No. 22092


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d5)

          1 mg

          $502

          Add

          Pregnenolone Carbonitrile

          A rodent PXR agonist

          CAS No. 1434-54-4

          Item No. 16343


          Formulation: A crystalline solid
          Purity: ≥97%
          • PCN
          • Pregnenolone 16α-carbonitrile
          • SC-4674

          25 mg

          $47

          Add

          50 mg

          $74

          Add

          100 mg

          $120

          Add

          250 mg

          $255

          Add

          Tienilic Acid

          Suicide substrate of CYP 2C9

          CAS No. 40180-04-9

          Item No. 10008517


          Formulation: A crystalline solid
          Purity: ≥99%

            5 mg

            $80

            Add

            10 mg

            $132

            Add

            25 mg

            $351

            Add

            50 mg

            $622

            Add

            Urolithin A

            A metabolite of ellagic acid with diverse biological activities

            CAS No. 1143-70-0

            Item No. 22607


            Formulation: A crystalline solid
            Purity: ≥98%
            • 2',7-Dihydroxy-3,4-benzocoumarin
            • 3,8-Dihydroxy Urolithin

            1 mg

            $25

            Add

            5 mg

            $44

            Add

            10 mg

            $75

            Add

            25 mg

            $156

            Add

            5-hydroxy Omeprazole

            A metabolite of omeprazole

            CAS No. 92340-57-3

            Item No. 10009028


            Formulation: A solid
            Purity: ≥98%
            • 5-hydroxy OMEP
            • 5-hydroxy OMP
            • 5-hydroxy OMZ

            500 µg

            $336

            Add

            1 mg

            $535

            Add

            Bufuralol (hydrochloride)

            An antagonist of β-adrenergic receptors

            CAS No. 60398-91-6

            Item No. 17794


            Formulation: A crystalline solid
            Purity: ≥95%
            • (±)-Bufuralol
            • DL-Bufuralol
            • Ro 3-4787

            1 mg

            $90

            Add

            5 mg

            $392

            Add

            10 mg

            $556

            Add

            Azamulin

            A selective CYP3A inhibitor

            CAS No. 76530-44-4

            Item No. 18748


            Formulation: A crystalline solid
            Purity: ≥98%
            • Antibiotic TDM 85-530
            • SA 85530b

            500 µg

            $50

            Add

            1 mg

            $81

            Add

            5 mg

            $198

            Add

            (−)-Warfarin

            An anticoagulant

            CAS No. 5543-57-7

            Item No. 13531


            Formulation: A crystalline solid
            Purity: ≥98%
            • (S)-Warfarin

            1 mg

            $82

            Add

            5 mg

            $266

            Add

            10 mg

            $489

            Add

            25 mg

            $1,018

            Add

            N-Acetyl-4-benzoquinone imine

            A reactive CYP450 metabolite of acetaminophen

            CAS No. 50700-49-7

            Item No. 16115


            Formulation: A crystalline solid
            Purity: ≥90%
            • NAPQI
            • N-Acetyl-p-benzoquinonimine

            500 µg

            $129

            Add

            1 mg

            $245

            Add

            5 mg

            $1,016

            Add

            Norfluoxetine (hydrochloride)

            An active metabolite of fluoxetine

            CAS No. 57226-68-3

            Item No. 15900


            Formulation: A crystalline solid
            Purity: ≥98%
            • Desmethylfluoxetine

            1 mg

            $50

            Add

            5 mg

            $218

            Add

            10 mg

            $305

            Add

            Furafylline

            An inhibitor of CYP1A2

            CAS No. 80288-49-9

            Item No. 9000058


            Formulation: A crystalline solid
            Purity: ≥95%

              500 µg

              $90

              Add

              1 mg

              $142

              Add

              5 mg

              $349

              Add

              6,7-dihydroxy Bergamottin

              A potent CYP3A4 inhibitor

              CAS No. 145414-76-2

              Item No. 10009598


              Formulation: A crystalline solid
              Purity: ≥98%
              • 6,7-DHB

              1 mg

              $55

              Add

              5 mg

              $193

              Add

              10 mg

              $358

              Add

              25 mg

              $825

              Add

              6-hydroxy Chlorzoxazone

              A metabolite of chlorzoxazone

              CAS No. 1750-45-4

              Item No. 10009029


              Formulation: A solid
              Purity: ≥95%
              • NSC 24955

              1 mg

              $116

              Add

              5 mg

              $260

              Add

              10 mg

              $462

              Add

              Displaying 1 - 25 of 374 Results
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