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Analytical Chemistry (1)
Biochemicals (35)
Antiparasitics (1)
Antivirals (1)
Antioxidants (1)
Kinase Inhibitors (35)
Aurora (1)
CaMKs (2)
Checkpoint Kinases (1)
ERK (2)
GSK3 (1)
MEK (35)
PDGFR Family (1)
PDPK1/PDK1 (1)
PKA (1)
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Displaying 1 - 25 of 35 Results
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PD 0325901

A MEK inhibitor that sustains stem cell renewal

CAS No. 391210-10-9

Item No. 13034


Formulation: A crystalline solid
Purity: ≥90%
  • Mirdametinib

5 mg

$54

Add

10 mg

$97

Add

25 mg

$175

Add

50 mg

$270

Add

U-0126

A MEK inhibitor and AMPK activator

CAS No. 109511-58-2

Item No. 70970


Formulation: A crystalline solid
Purity: ≥98%

    1 mg

    $49

    Add

    5 mg

    $130

    Add

    10 mg

    $236

    Add

    25 mg

    $412

    Add

    KT 5720

    A potent inhibitor of PKA

    CAS No. 108068-98-0

    Item No. 10011011


    Formulation: A clear film
    Purity: ≥98%

      50 µg

      $90

      Add

      100 µg

      $142

      Add

      250 µg

      $328

      Add

      500 µg

      $479

      Add

      Trametinib

      An inhibitor of MEK1 and MEK2

      CAS No. 871700-17-3

      Item No. 16292


      Formulation: A crystalline solid
      Purity: ≥95%
      • GSK1120212
      • JTP-74057

      25 mg

      $75

      Add

      50 mg

      $105

      Add

      100 mg

      $165

      Add

      250 mg

      $374

      Add

      Myricetin

      A potent antioxidant

      CAS No. 529-44-2

      Item No. 10012600


      Formulation: A crystalline solid
      Purity: ≥98%
      • Cannabiscetin
      • LDN-0014058
      • NSC 407290

      10 mg

      $43

      Add

      25 mg

      $103

      Add

      50 mg

      $161

      Add

      100 mg

      $237

      Add

      PD 184161

      A potent MEK1/2 inhibitor

      CAS No. 212631-67-9

      Item No. 10012431


      Formulation: A crystalline solid
      Purity: ≥98%

        1 mg

        $31

        Add

        5 mg

        $129

        Add

        10 mg

        $228

        Add

        25 mg

        $493

        Add

        AZD 6244

        A highly selective inhibitor of MEK1/2

        CAS No. 606143-52-6

        Item No. 11599


        Formulation: A crystalline solid
        Purity: ≥95%
        • ARRY-142886
        • CL 1,040
        • NSC 741O78
        • Selumetinib

        10 mg

        $36

        Add

        25 mg

        $61

        Add

        50 mg

        $95

        Add

        100 mg

        $120

        Add

        Cobimetinib

        A potent, orally available MEK1 inhibitor

        CAS No. 934660-93-2

        Item No. 19563


        Formulation: A crystalline solid
        Purity: ≥98%
        • GDC-0973
        • RG-7420
        • XL518

        1 mg

        $54

        Add

        5 mg

        $197

        Add

        10 mg

        $367

        Add

        25 mg

        $783

        Add

        Trametinib-13C-d3

        An internal standard for the quantification of trametinib

        CAS No. 2712126-59-3

        Item No. 29144


        Formulation: A solid
        Purity: ≥99% deuterated forms (d1-d3)

          1 mg

          $436

          Add

          Binimetinib

          A MEK1/2 inhibitor

          CAS No. 606143-89-9

          Item No. 16996


          Formulation: A crystalline solid
          Purity: ≥98%
          • ​ARRY-438162
          • MEK162

          5 mg

          $35

          Add

          10 mg

          $53

          Add

          50 mg

          $123

          Add

          100 mg

          $228

          Add

          CI-1040

          A potent MEK inhibitor

          CAS No. 212631-79-3

          Item No. 11580


          Formulation: A crystalline solid
          Purity: ≥98%
          • PD 184352

          5 mg

          $90

          Add

          10 mg

          $158

          Add

          25 mg

          $349

          Add

          50 mg

          $653

          Add

          BIX02189

          An inhibitor of MEK5 and ERK5

          CAS No. 1265916-41-3

          Item No. 16999


          Formulation: A crystalline solid
          Purity: ≥98%

            5 mg

            $129

            Add

            10 mg

            $231

            Add

            25 mg

            $319

            Add

            Refametinib

            An allosteric inhibitor of MEK1/2

            CAS No. 923032-37-5

            Item No. 16997


            Formulation: A crystalline solid
            Purity: ≥95%
            • BAY 86-9766
            • RDEA119

            1 mg

            $42

            Add

            5 mg

            $123

            Add

            10 mg

            $183

            Add

            50 mg

            $602

            Add

            Hypothemycin

            A resorcylic acid lactone polyketide with diverse biological activities

            CAS No. 76958-67-3

            Item No. 27913


            Formulation: A solid
            Purity: ≥95%
            • NSC 354462

            1 mg

            $219

            Add

            5 mg

            $1,040

            Add

            U-0124

            An inactive analog of U-0126

            CAS No. 108923-79-1

            Item No. 34871


            Formulation: A solid
            Purity: ≥95%

              500 µg

              $95

              Add

              1 mg

              $167

              Add

              AS-703026

              A MEK1/2 inhibitor

              CAS No. 1236699-92-5

              Item No. 11226


              Formulation: A crystalline solid
              Purity: ≥95%
              • MSC1936369B
              • Pimasertib

              1 mg

              $28

              Add

              5 mg

              $83

              Add

              10 mg

              $125

              Add

              25 mg

              $207

              Add

              GDC-0623

              A potent, ATP-uncompetitive inhibitor of MEK1

              CAS No. 1168091-68-6

              Item No. 19479


              Formulation: A crystalline solid
              Purity: ≥98%

                1 mg

                $46

                Add

                5 mg

                $134

                Add

                10 mg

                $222

                Add

                25 mg

                $333

                Add

                PD 198306

                A potent inhibitor of MEK1/2

                CAS No. 212631-61-3

                Item No. 23966


                Formulation: A solid
                Purity: ≥98%

                  1 mg

                  $74

                  Add

                  5 mg

                  $255

                  Add

                  10 mg

                  $399

                  Add

                  SL 327

                  A selective MEK1/2 inhibitor

                  CAS No. 305350-87-2

                  Item No. 15598


                  Formulation: A crystalline solid
                  Purity: ≥95% (mixture of cis/trans isomers)

                    1 mg

                    $63

                    Add

                    5 mg

                    $90

                    Add

                    10 mg

                    $153

                    Add

                    25 mg

                    $303

                    Add

                    TAK-733

                    A MEK1 inhibitor

                    CAS No. 1035555-63-5

                    Item No. 16998


                    Formulation: A crystalline solid
                    Purity: ≥98%

                      500 µg

                      $37

                      Add

                      1 mg

                      $66

                      Add

                      5 mg

                      $229

                      Add

                      10 mg

                      $418

                      Add

                      BIX02188

                      A potent MEK5 inhibitor

                      CAS No. 334949-59-6

                      Item No. 16238


                      Formulation: A crystalline solid
                      Purity: ≥95%

                        1 mg

                        $49

                        Add

                        5 mg

                        $178

                        Add

                        10 mg

                        $306

                        Add

                        25 mg

                        $645

                        Add

                        RO4987655

                        A MEK inhibitor

                        CAS No. 874101-00-5

                        Item No. 19488


                        Formulation: A crystalline solid
                        Purity: ≥98%
                        • CH4987655

                        1 mg

                        $65

                        Add

                        5 mg

                        $195

                        Add

                        10 mg

                        $293

                        Add

                        25 mg

                        $568

                        Add

                        HI TOPK 032

                        An inhibitor of TOPK, Chk1, and MEK1 kinases

                        CAS No. 487020-03-1

                        Item No. 19815


                        Formulation: A crystalline solid
                        Purity: ≥95%

                          1 mg

                          $38

                          Add

                          5 mg

                          $102

                          Add

                          10 mg

                          $165

                          Add

                          BI-847325

                          A selective dual MEK/Aurora kinase inhibitor

                          CAS No. 1207293-36-4

                          Item No. 18301


                          Formulation: A crystalline solid
                          Purity: ≥98%

                            1 mg

                            $81

                            Add

                            5 mg

                            $189

                            Add

                            HRX215

                            An MKK4 inhibitor

                            CAS No. 2369583-33-3

                            Item No. 41238


                            Formulation: A solid
                            Purity: ≥98%
                            • Darizmetinib
                            • LN3348

                            1 mg

                            $138

                            Add

                            5 mg

                            $471

                            Add

                            10 mg

                            $825

                            Add

                            25 mg

                            $1,375

                            Add

                            Displaying 1 - 25 of 35 Results
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