A convenient fluorescence-based method for screening FAAH inhibitors
Features
  • Screen for inhibitors of FAAH
  • Assay 45 samples in duplicate
  • Includes JZL 195 positive control
  • Plate-based fluorometric measurement (ex 340-360 nm, em 450-465 nm)
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Fatty Acid Amide Hydrolase Inhibitor Screening Assay Kit

Item No. 10005196

Kit Booklet (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Synonyms
  • Anandamide Amidohydrolase 1
  • FAAH
  • Oleamide Hydrolase 1
  • PSAB
Emission
450-465 nm
Excitation
340-360 nm
Shipping & Storage Information
Storage
-80°C
Shipping
Dry ice in continental US; may vary elsewhere
Recommended Products

Certificates of Analysis & Batch Specific Data

Provide batch numbers separated by commas to download or request available product inserts, QC sheets, certificates of analysis, data packs, and GC-MS data.

    96 wells

    $413

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    Product Description

    Cayman’s FAAH Inhibitor Screening Assay Kit provides a convenient fluorescence-based method for screening FAAH inhibitors. FAAH hydrolyzes AMC arachidonoyl amide resulting in the release of the fluorescent product, 7-amino-4-methylcoumarin (AMC). The fluorophore can be easily analyzed using an excitation wavelength of 340-360 nm and an emission wavelength of 450-465 nm.

    Needed but not supplied: Please download the kit booklet to verify if UltraPure Water (Milli-Q or equivalent) or any other components are needed for this assay.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Citations

    Azar, S., Udi, S., Drori, A., et al. Reversal of diet-induced hepatic steatosis by peripheral CB1 receptor blockade in mice is p53/miRNA-22/SIRT1/PPARα dependent. Mol. Metab. (2020).

    El-Alfy, A., Abourashed, E.A., Patel, C.A., et al. Phenolic compounds from nutmeg (Myristica fragrans Houtt.) inhibit the endocannabinoid-modulating enzyme fatty acid amide hydrolase. J. Pharm. Pharmacol. 71(12), 1879-1889 (2019).

    Jaiswal, S., Tripathi, R.K.P., and Ayyannan, S.R. Scaffold hopping-guided design of some isatin based rigid analogs as fatty acid amide hydrolase inhibitors: Synthesis and evaluation. Biomed. Pharmacother. 107, 1611-1623 (2018).