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4-bromo-2,5-DMA (hydrochloride)

Item No. 11142

Restricted Product (Schedule I)
Product Insert (PDF)GC-MS (PDF)Safety Data Sheet (SDS) (PDF)
Synonyms
Synonyms
  • 4-bromo-2,5-Dimethoxyamphetamine
  • Dimethoxybromoamphetamine
  • DOB
Technical Information
Formal Name
4-bromo-2,5-dimethoxy-α-methyl-benzeneethanamine, monohydrochloride
CAS Number
29705-96-2
Molecular Formula
C11H16BrNO2 • HCl
Formula Weight
310.6
Purity
≥98%
Formulation
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 10 mg/mlDMSO: 5 mg/mlEthanol: 5 mg/mlPBS (pH 7.2): 5 mg/ml
λmax
206, 297 nm
SMILES
COC1=C(CC(N)C)C=C(OC)C(Br)=C1.Cl
InChi Code
InChI=1S/C11H16BrNO2.ClH/c1-7(13)4-8-5-11(15-3)9(12)6-10(8)14-2;/h5-7H,4,13H2,1-3H3;1H
InChi Key
SPBBKPOIDQIWDZ-UHFFFAOYSA-N
Regulatory Information
DEA Schedule
I
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    5 mg

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    Product Description

    4-bromo-2,5-DMA is a common hallucinogenic designer drug which avidly binds and activates serotonin receptors (Ki = 2.2 and 2.8 nM for 5-HT2A and 5-HT2C, respectively).1,2 Methods have been developed for the identification of this compound in serum and in urine.3,4 4-bromo-2,5-DMA is regulated as a Schedule I compound in the United States. This product is intended for research and forensic applications.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. de Boer, D., and Bosman, I. A new trend in drugs-of-abuse; the 2C-series of phenethylamine designer drugs. Pharm. World Sci. 26(2), 110-113 (2004).

    2. Chambers, J.J., Kurrasch-Orbaugh, D.M., Parker, M.A., et al. Enantiospecific synthesis and pharmacological evaluation of a series of super-potent, conformationally restricted 5-HT2A/2C receptor agonists. J. Med. Chem. 44(6), 1003-1010 (2001).

    3. Wohlfarth, A., Weinmann, W., and Dresen, S. LC-MS/MS screening method for designer amphetamines, tryptamines, and piperazines in serum. Anal. Bioanal. Chem. 396(7), 2403-2414 (2010).

    4. Kerrigan, S., Banuelos, S., Perrella, L., et al. Simultaneous detection of ten psychedelic phenethylamines in urine by gas chromatography-mass spectrometry. J. Anal. Toxicol. 35(7), 459-469 (2011).

    Product Citations

    Halberstadt, A.L., Chatha, M., Stratford, A., et al. Comparison of the behavioral responses induced by phenylalkylamine hallucinogens and their tetrahydrobenzodifuran (“FLY”) and benzodifuran (“DragonFLY”) analogs. Neuropharmacology 144, 368-376 (2019).