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A-796260

Item No. 11606

Product Insert (PDF)GC-MS (PDF)Safety Data Sheet (SDS) (PDF)
Synonyms
Synonyms
  • LTI-258
Technical Information
Formal Name
[1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone
CAS Number
895155-26-7
Molecular Formula
C22H30N2O2
Formula Weight
354.5
Purity
≥98%
Formulation
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 5 mg/mlDMSO: 3 mg/mlEthanol: 5 mg/mlEthanol:PBS(pH 7.2) (1:5): 0.16 mg/mlMethanol: 1 mg/ml
λmax
218, 246, 303 nm
SMILES
CC(C1(C)C)(C)C1C(C2=CN(CCN3CCOCC3)C4=CC=CC=C42)=O
InChi Code
InChI=1S/C22H30N2O2/c1-21(2)20(22(21,3)4)19(25)17-15-24(18-8-6-5-7-16(17)18)10-9-23-11-13-26-14-12-23/h5-8,15,20H,9-14H2,1-4H3
InChi Key
ZCFHOMLAFTWDFM-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    1 mg

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    Cayman Chemical
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    Product Description

    A-796260 is a synthetic cannabinoid (CB) that shows high selectivity for the CB2 receptor (Ki = 0.77 nM) over the CB1 receptor (Ki = 2,100 nM).1 It also shows efficacy in vivo in models of inflammatory, post-operative, neuropathic, and osteoarthritic pain, activities which are selectively blocked by CB2 receptor-selective antagonists.2 This product is intended for research and forensic uses.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Poso, A., and Huffman, J.W. Targeting the cannabinoid CB2 receptor: Modelling and structural determinants of CB2 selective ligands. Br. J. Pharmacol. 153(2), 335-346 (2008).

    2. Yao, B.B., Hsieh, G.C., Frost, J.M., et al. In vitro and in vivo characterization of A-796260: A selective cannabinoid CB2 receptor agonist exhibiting analgesic activity in rodent pain models. Br. J. Pharmacol. 153(2), 390-401 (2008).