An LSD1 inhibitor
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S 2101

Item No. 19802

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
(1R,2S)-rel-2-[3,5-difluoro-2-(phenylmethoxy)phenyl]-cyclopropanamine, monohydrochloride
CAS Number
1239262-36-2
Synonyms
  • KDM1 inhibitor II
  • LSD1 inhibitor II
  • Lysine-specific Demethylase 1 Inhibitor II
Molecular Formula
C16H15F2NO • HCl
Formula Weight
311.8
Purity
≥98%
Formulation
A solid
Solubility(Learn about Variance in Solubility)
Water: Soluble
SMILES
FC1=C(OCC2=CC=CC=C2)C([C@@H]3C[C@H]3N)=CC(F)=C1.Cl
InChi Code
InChI=1S/C16H15F2NO.ClH/c17-11-6-13(12-8-15(12)19)16(14(18)7-11)20-9-10-4-2-1-3-5-10;/h1-7,12,15H,8-9,19H2;1H/t12-,15+;/m0./s1
InChi Key
CTSUZAFTJVLOIX-SBKWZQTDSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
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    1 mg

    $41

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    5 mg

    $184

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    10 mg

    $266

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    25 mg

    $611

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    Product Description

    S 2101 is an inhibitor of lysine-specific demethylase 1 (LSD1; Ki = 0.61 µM).1 It is selective for LSD1 over monoamine oxidase A (MAO-A) and MAO-B (Kis = 17 and 110 µM, respectively).

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Mimasu, S., Umezawa, N., Sato, S., et al. Structurally designed trans-2-phenylcyclopropylamine derivatives potently inhibit histone demethylase LSD1/KDM1. Biochemistry 49(30), 6494-6503 (2010).