An Analytical Reference Standard
Related Products
Certified Reference Material(s)
35880Tianeptine (sodium salt) (CRM)
Research Tool(s)
17561Tianeptine (sodium salt)
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Tianeptine (sodium salt)

Item No. 25950

Product Insert (PDF)GC-MS (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
7-[(3-chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]-heptanoic acid, monosodium salt
CAS Number
30123-17-2
Molecular Formula
C21H24ClN2O4S • Na
Formula Weight
458.9
Purity
≥98%
Formulation
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 30 mg/mlDMSO: 20 mg/mlEthanol: 10 mg/mlPBS (pH 7.2): 10 mg/ml
SMILES
[O-]C(CCCCCCNC(C1=C2C=C(Cl)C=C1)C(C=CC=C3)=C3N(C)S2(=O)=O)=O.[Na+]
InChi Code
InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);/q;+1/p-1
InChi Key
ZLBSUOGMZDXYKE-UHFFFAOYSA-M
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    Product Description

    Tianeptine (sodium salt) (Item No. 25950) is an analytical reference standard categorized as an opioid.1 Tianeptine has been abused and associated with overdose and death.2 Formulations containing tianeptine have been used in the treatment of depression.3 This product is intended for use in analytical forensic applications. This product is also available as a general research tool (Item No. 17561).

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Gassaway, M.M., Rives, M.L., Kruegel, A.C., et al. The atypical antidepressant and neurorestorative agent tianeptine is a μ-opioid receptor agonist. Transl. Psychiatry 4(7), e411 (2014).

    2. Lauhan, R., Hsu, A., Alam, A., et al. Tianeptine abuse and dependence: Case report and literature review. Psychosomatics 59(6), 547-553 (2018).

    3. McEwen, B.S., Chattarji, S., Diamond, D.M., et al. The neurobiological properties of tianeptine (Stablon): From monoamine hypothesis to glutamatergic modulation. Mol. Psychiatry 15(3), 237-249 (2010).

    Product Citations

    Vandeputte, M.M., Cannaert, A., and Stove, C.P. In vitro functional characterization of a panel of non‑fentanyl opioid new psychoactive substances. Arch. Toxicol. 94(11), 3819-3830 (2020).