An N-type calcium channel blocker
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PD 173212

Item No. 29447

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
N-[[4-(1,1-dimethylethyl)phenyl]methyl]-N-methyl-L-leucyl-N-(1,1-dimethylethyl)-O-(phenylmethyl)-L-tyrosinamide
CAS Number
217171-01-2
Molecular Formula
C38H53N3O3
Formula Weight
599.9
Purity
≥95%
Formulation
A solid
Solubility(Learn about Variance in Solubility)
DMSO: 100 mMEthanol: 100 mM
SMILES
CC(C)(C)C1=CC=C(CN(C)[C@@H](CC(C)C)C(N[C@@H](CC2=CC=C(OCC3=CC=CC=C3)C=C2)C(NC(C)(C)C)=O)=O)C=C1
InChi Code
InChI=1S/C38H53N3O3/c1-27(2)23-34(41(9)25-29-15-19-31(20-16-29)37(3,4)5)36(43)39-33(35(42)40-38(6,7)8)24-28-17-21-32(22-18-28)44-26-30-13-11-10-12-14-30/h10-22,27,33-34H,23-26H2,1-9H3,(H,39,43)(H,40,42)/t33-,34-/m0/s1
InChi Key
GCDHMGROXQUFNR-HEVIKAOCSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    500 µg

    $37

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    1 mg

    $66

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    5 mg

    $194

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    Product Description

    PD 173212 is an N-type calcium channel blocker (IC50 = 36 nM).1 It prevents audiogenic seizures in mice when administered at a dose of 30 mg/kg.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Hu, L.-Y., Ryder, T.R., Rafferty, M.F., et al. Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers. Bioorg. Med. Chem. Lett. 9(15), 2151-2156 (1999).