An atypical antipsychotic
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BMY 14802 (hydrochloride)

Item No. 42264

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
α-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol, monohydrochloride
CAS Number
105565-55-7
Synonyms
  • BMS 181100
Molecular Formula
C18H22F2N4O • HCl
Formula Weight
384.9
Purity
≥98%
Formulation
A solid
Solubility(Learn about Variance in Solubility)
DMSO: Sparingly soluble: 1-10 mg/mlEthanol: Slightly soluble: 0.1-1 mg/ml
SMILES
FC1=CC=C(C(CCCN2CCN(C3=NC=C(F)C=N3)CC2)O)C=C1.Cl
InChi Code
InChI=1S/C18H22F2N4O.ClH/c19-15-5-3-14(4-6-15)17(25)2-1-7-23-8-10-24(11-9-23)18-21-12-16(20)13-22-18;/h3-6,12-13,17,25H,1-2,7-11H2;1H
InChi Key
NIBVEFRJDFVQLM-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
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    5 mg

    $65

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    10 mg

    $124

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    25 mg

    $293

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    50 mg

    $520

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    Product Description

    BMY 14802 is an atypical antipsychotic.1 It selectively binds to σ receptors over α1-adrenergic receptors (α1-ARs) and dopamine D2 receptors (IC50s = 112, 520, and 6,340 nM, respectively). In vivo, BMY 14802 inhibits the conditioned avoidance response and apomorphine-induced stereotypy in rats (ED50s = 26.4 and 33 mg/kg, respectively).

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Yevich, J.P., New, J.S., Lobeck, W.G., et al. Synthesis and biological characterization of ɑ-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol and analogues as potential atypical antipsychotic agents. J. Med. Chem. 35(24), 4516-4525 (1992).