A STAT5a inhibitor
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Stafia-1

Item No. 43191

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
CAS Number
2582757-90-0
Molecular Formula
C24H27O10P
Formula Weight
506.4
Purity
≥95%
Formulation
A solid
Solubility(Learn about Variance in Solubility)
DMSO: Slightly Soluble: 0.1-1 mg/mlEthanol: Sparingly Soluble: 1-10 mg/ml
SMILES
COC1=CC(C2=CC(C3=CC(OC)=C(OC)C(OC)=C3)=CC(OP(O)(O)=O)=C2)=CC(OC)=C1OC
InChi Code
InChI=1S/C24H27O10P/c1-28-19-10-16(11-20(29-2)23(19)32-5)14-7-15(9-18(8-14)34-35(25,26)27)17-12-21(30-3)24(33-6)22(13-17)31-4/h7-13H,1-6H3,(H2,25,26,27)
InChi Key
UGUOUFLCZFMHNI-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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Certificates of Analysis & Batch Specific Data

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    5 mg

    $285

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    10 mg

    $456

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    25 mg

    $927

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    50 mg

    $1,425

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    Product Description

    Stafia-1 is an inhibitor of STAT5a (Ki = 10.9 µM).1 It is selective for STAT5a over STAT5b and STAT3 (Kis = >200 µM for both).

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Natarajan, K., Müller-Klieser, D., Rubner, S., et al. Stafia-1: A STAT5a-selective inhibitor developed via docking-based screening of in silico o-phosphorylated fragments. Chemistry 26(1), 148-154 (2020).