A DPP-4 inhibitor
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CGT-8012

Item No. 45055

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
3R-amino-1-[5,6-dihydro-3-(trifluoromethyl)imidazo[1,5-a]pyrazin-7(8H)-yl]-4-(2,4,5-trifluorophenyl)-1-butanone
CAS Number
1152810-23-5
Synonyms
  • Sheng Gelieting
Molecular Formula
C17H16F6N4O
Formula Weight
406.3
Purity
≥95%
Formulation (Request formulation change)
A 10 mg/ml solution in ethanol
Solubility(Learn about Variance in Solubility)
Acetonitrile: Sparingly Soluble: 1-10 mg/mlEthanol: Soluble: ≥10 mg/ml
SMILES
FC(C=C(C(F)=C1)F)=C1C[C@H](CC(N(C2)CCN3C2=CN=C3C(F)(F)F)=O)N
InChi Code
InChI=1S/C17H16F6N4O/c18-12-6-14(20)13(19)4-9(12)3-10(24)5-15(28)26-1-2-27-11(8-26)7-25-16(27)17(21,22)23/h4,6-7,10H,1-3,5,8,24H2/t10-/m1/s1
InChi Key
AAOHXMMVWCGBJI-SNVBAGLBSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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Certificates of Analysis & Batch Specific Data

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    1 mg

    $65

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    5 mg

    $211

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    Product Description

    CGT-8012 is a dipeptidyl peptidase 4 (DPP-4) inhibitor (IC50 = 0.14 µM).1

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Tang, P.C., Yang, F., Wang, Y., et al. Piperazine derivatives, preparation process and pharmaceutical use thereof. (2007).