A selective GPR55 antagonist
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Product Categories

Product Type

Small Molecule Modulators
Receptor Pharmacology
Antagonists

Research Area

ML-192

Item No. 15183

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
2-furanyl[4-(5,6,7,8-tetrahydro-2-methyl[1]benzothieno[2,3-d]pyrimidin-4-yl)-1-piperazinyl]-methanone
CAS Number
460331-61-7
Synonyms
  • CID-1434953
Molecular Formula
C20H22N4O2S
Formula Weight
382.5
Purity
≥98%
Formulation
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 10 mg/mlDMSO: 5 mg/mlEthanol: 15 mg/mlEthanol:PBS (pH 7.2)(1:2): 0.30 mg/ml
λmax
235, 292 nm
SMILES
O=C(C1=CC=CO1)N2CCN(C3=C4C(SC5=C4CCCC5)=NC(C)=N3)CC2
InChi Code
InChI=1S/C20H22N4O2S/c1-13-21-18(17-14-5-2-3-7-16(14)27-19(17)22-13)23-8-10-24(11-9-23)20(25)15-6-4-12-26-15/h4,6,12H,2-3,5,7-11H2,1H3
InChi Key
GDPDARVUXXOYAJ-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
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    1 mg

    $80

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    5 mg

    $293

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    10 mg

    $467

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    Product Description

    ML-192 is an antagonist of GPR55 (IC50 = 702 nM).1 It is selective for GPR55 over the cannabinoid (CB) receptors CB1 and CB2, as well as GPR35 (IC50s = >32 μM).

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Heynen-Genel, S., Dahl, R., Shi, S., et al. Selective GPR55 antagonists: Screening for selective ligands for GPR55. Probe Reports from the NIH Molecular Libraries Program (2011).