A PKCα inhibitor
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PKCα (C2-4) Inhibitor Peptide

Item No. 17478

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Synonyms
  • Protein Kinase Cα (C2-4) Inhibitor Peptide
Molecular Formula
C47H74N14O17
Formula Weight
1107.2
Purity
≥95%
Formulation (Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 1 mg/mlDMSO: 10 mg/mlPBS (pH 7.2): 5 mg/ml
SMILES
O=C[C@H](CO)NN[C@@H](CC(C)C)C(N[C@@H](CC(N)=O)C(N1CCC[C@H]1C(N[C@@H](CCC(O)=O)C(N[C@H](C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CCC(N)=O)C(N[C@]([C@@H](C)O)([H])C=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)=O)=O)=O
InChi Code
InChI=1S/C47H74N14O16/c1-24(2)18-33(60-59-27(21-62)22-63)44(75)57-34(20-38(49)68)46(77)61-17-5-7-36(61)45(76)55-31(13-15-39(69)70)41(72)56-32(19-26-8-10-28(66)11-9-26)43(74)53-29(6-4-16-52-47(50)51)40(71)54-30(12-14-37(48)67)42(73)58-35(23-64)25(3)65
InChi Key
XYGZNIKBSICVGI-FZSOQVDMSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    500 µg

    $106

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    1 mg

    $201

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    5 mg

    $783

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    Product Description

    PKCα (C2-4) inhibitor peptide is a synthetic peptide that blocks PKC activity in HepG2 cells stimulated with calcium and pancreastatin when applied at 10 µM.1

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Gayen, J.R., Saberi, M., Schenk, S., et al. A novel pathway of insulin sensitivity in chromogranin A null mice: A crucial role for pancreastatin in glucose homeostasis. The Journal of Biological Chemisty 248(42), 28498-28509 (2009).