A selective GABAB receptor antagonist
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CGP 54626 (hydrochloride)

Item No. 20121

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
P-(cyclohexylmethyl)-P-[(2S)-3-[[(1S)-1-(3,4-dichlorophenyl)ethyl]amino]-2-hydroxypropyl]-phosphinic acid, monohydrochloride
CAS Number
149184-21-4
Synonyms
  • CGP 54626A
Molecular Formula
C18H28Cl2NO3P • HCl
Formula Weight
444.8
Purity
≥95%
Formulation
A crystalline solid
Solubility(Learn about Variance in Solubility)
DMF: 0.33 mg/mlDMSO: 1 mg/mlDMSO:PBS (pH 7.2) (1:6): 0.14 mg/mlEthanol: 0.2 mg/ml
SMILES
ClC(C=C1)=C(Cl)C=C1[C@H](C)NC[C@H](O)CP(CC2CCCCC2)(O)=O.Cl
InChi Code
InChI=1S/C18H28Cl2NO3P.ClH/c1-13(15-7-8-17(19)18(20)9-15)21-10-16(22)12-25(23,24)11-14-5-3-2-4-6-14;/h7-9,13-14,16,21-22H,2-6,10-12H2,1H3,(H,23,24);1H/t13-,16-;/m0./s1
InChi Key
ZQCFHOVIXCJPLE-LINSIKMZSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    1 mg

    $60

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    5 mg

    $165

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    10 mg

    $270

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    Product Description

    CGP 54626 is a selective antagonist of the GABAB receptor with an IC50 value of 4 nM.1 It can be used to investigate the role of GABAB receptors in neurological signaling.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Kaupmann, K., Malitschek, B., Schuler, V., et al. GABAB-receptor subtypes assemble into functional heteromeric complexes. Nature 396(6712), 683-687 (1998).