A metabolite of trifluoperazine
Related Products
Parent Compound(s)
15068Trifluoperazine (hydrochloride)
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Trifluoperazine N-Glucuronide

Item No. 34299

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
1-β-D-glucopyranuronosyl-1-methyl-4-[3-[2-(trifluoromethyl)-10H-phenothiazin-10-yl]propyl]-piperazinium, inner salt
CAS Number
165602-90-4
Synonyms
  • TFP N-Glucuronide
Molecular Formula
C27H32F3N3O6S
Formula Weight
583.6
Purity
≥70%
Formulation (Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
Methanol: SolubleWater: Soluble
SMILES
C[N+](CC1)([C@H]2[C@H](O)[C@@H](O)[C@@H]([C@@H](C([O-])=O)O2)O)CCN1CCCN3C4=CC(C(F)(F)F)=CC=C4SC5=CC=CC=C53
InChi Code
InChI=1S/C27H32F3N3O6S/c1-33(25-23(36)21(34)22(35)24(39-25)26(37)38)13-11-31(12-14-33)9-4-10-32-17-5-2-3-6-19(17)40-20-8-7-16(15-18(20)32)27(28,29)30/h2-3,5-8,15,21-25,34-36H,4,9-14H2,1H3/t21-,22-,23+,24-,25+/m0/s1
InChi Key
AFYPHWNGUDUHIW-ARXROMJUSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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    500 µg

    $241

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    1 mg

    $457

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    Product Description

    Trifluoperazine N-glucuronide is a metabolite of the antipsychotic agent trifluoperazine (Item No. 15068).1,2 It is formed from trifluoperazine by the UDP-glucuronosyltransferase (UGT) isoform UGT1A4.2

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Luo, H., Hawes, E.M., McKay, G., et al. N(+)-glucuronidation of aliphatic tertiary amines in human: antidepressant versus antipsychotic drugs. Xenobiotica 25(3), 291-301 (1995).

    2. Fujiwara, R., Nakajima, M., Yamanaka, H., et al. Interactions between human UGT1A1, UGT1A4, and UGT1A6 affect their enzymatic activities. Drug Metab. Dispos. 35(10), 1781-1787 (2007).