A metabolite of febuxostat
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Parent Compound(s)
14127Febuxostat
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Febuxostat Acyl Glucuronide

Item No. 26599

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
1-[2-[3-cyano-4-(2-methylpropoxy)phenyl]-4-methyl-5-thiazolecarboxylate], β-D-glucopyranuronic acid
CAS Number
1351692-92-6
Molecular Formula
C22H24N2O9S
Formula Weight
492.5
Purity
≥98%
Formulation (Request formulation change)
A solid
Solubility(Learn about Variance in Solubility)
DMSO: slightly solubleMethanol: slightly soluble
SMILES
CC(C)COC1=C(C#N)C=C(C2=NC(C)=C(C(O[C@@H]3O[C@H](C(O)=O)[C@@H](O)[C@H](O)[C@H]3O)=O)S2)C=C1
InChi Code
InChI=1S/C22H24N2O9S/c1-9(2)8-31-13-5-4-11(6-12(13)7-23)19-24-10(3)18(34-19)21(30)33-22-16(27)14(25)15(26)17(32-22)20(28)29/h4-6,9,14-17,22,25-27H,8H2,1-3H3,(H,28,29)/t14-,15-,16+,17-,22-/m0/s1
InChi Key
ZRXRMGPMLDOOKN-FVMGUFKOSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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Certificates of Analysis & Batch Specific Data

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    500 µg

    $90

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    1 mg

    $168

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    2.5 mg

    $392

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    Cayman Chemical
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    Product Description

    Febuxostat acyl glucuronide is a metabolite of the xanthine oxidoreductase inhibitor febuxostat (Item No. 14127).1,2 Febuxostat acyl glucuronide is formed via glucuronidation of febuxostat by uridine diphosphate-glucuronosyltransferases (UGTs).2

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Grabowski, B.A., Khosravan, R., Vernillet, L., et al. Metabolism and excretion of [14C] febuxostat, a novel nonpurine selective inhibitor of xanthine oxidase, in healthy male subjects. J. Clin. Pharmacol. 51(2), 189-201 (2011).

    2. Kamel, B., Graham, G.G., Williams, K.M., et al. Clinical pharmacokinetics and pharmacodynamics of febuxostat. Clin. Pharmacokinet. 56(5), 459-475 (2017).