A prodrug form of paliperidone
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Active Metabolite(s)
15556Paliperidone
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Paliperidone Palmitate

Item No. 39644

Product Insert (PDF)Safety Data Sheet (SDS) (PDF)
Technical Information
Formal Name
hexadecanoic acid, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl ester
CAS Number
199739-10-1
Synonyms
  • 9-hydroxy Risperidone Palmitate
  • RO92670
Molecular Formula
C39H57FN4O4
Formula Weight
664.9
Purity
≥98%
Formulation
A solid
Solubility(Learn about Variance in Solubility)
Chloroform: Slightly SolubleMethanol: SolubleWater: Slightly Soluble
SMILES
O=C(N1CCC2)C(CCN3CCC(CC3)C4=NOC5=C4C=CC(F)=C5)=C(C)N=C1C2OC(CCCCCCCCCCCCCCC)=O
InChi Code
InChI=1S/C39H57FN4O4/c1-3-4-5-6-7-8-9-10-11-12-13-14-15-18-36(45)47-34-17-16-24-44-38(34)41-29(2)32(39(44)46)23-27-43-25-21-30(22-26-43)37-33-20-19-31(40)28-35(33)48-42-37/h19-20,28,30,34H,3-18,21-27H2,1-2H3
InChi Key
VOMKSBFLAZZBOW-UHFFFAOYSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Room temperature in continental US; may vary elsewhere
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Certificates of Analysis & Batch Specific Data

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    100 mg

    $109

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    250 mg

    $164

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    1 g

    $491

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    Product Description

    Paliperidone palmitate is a prodrug form of the atypical antipsychotic paliperidone (Item No. 15556).1,2 Formulations containing paliperidone palmitate have been used in the treatment of schizophrenia and schizoaffective disorder.

    WARNING This product is not for human or veterinary use.

    References & Product Citations
    Product Description References

    1. Chen, A., Cai, P., Peng, Y., et al. The role of alkyl chain length in the melt and solution crystallization of paliperidone aliphatic prodrugs. IUCrJ 11(Pt. 1), 23-33 (2024).

    2. Patel, H., Patel, P., Modi, N., et al. Rats and rabbits as pharmacokinetic screening tools for long acting intramuscular depots: Case study with paliperidone palmitate suspension. Xenobiotica 49(4), 415-421 (2019).